Volume 24, Issue 1

Search all Molecular Diversity articles

February 2020

26 articles in this issue

One-pot organocatalytic/multicomponent approach for the preparation of novel enantioenriched non-natural selenium-based peptoids and peptide–peptoid conjugates
Alexander F. de la Torre
Akbar Ali
Márcio W. Paixão
Original Article 18 February 2019 Pages: 1 - 10
Substituent effect on inter-ring interaction in paracyclophanes
Irena Majerz
Teresa Dziembowska
Original Article Open access 19 February 2019 Pages: 11 - 20
Lupenone is a good anti-inflammatory compound based on the network pharmacology
Feng Xu
Liubo Yang
Hongmei Wu
Original Article 22 February 2019 Pages: 21 - 30
The periodic table of urea derivative: small molecules of zinc(II) and nickel(II) of diverse antimicrobial and antiproliferative applications
Christina N. Banti
Mehmet Poyraz
Sotiris K. Hadjikakou
Original Article 23 February 2019 Pages: 31 - 43
Combining ligand- and structure-based in silico methods for the identification of natural product-based inhibitors of Akt1
Priya Mahajan
Bhumika Wadhwa
Amit Nargotra
Original Article 23 February 2019 Pages: 45 - 60
Single-stage synthesis of heterocyclic alkaloid-like compounds from (+)-camphoric acid and their antiviral activity
Vladimir V. Chernyshov
Olga I. Yarovaya
Nariman F. Salakhutdinov
Original Article 28 February 2019 Pages: 61 - 67
Design and synthesis of new imidazo[1,2-b]pyrazole derivatives, in vitro α-glucosidase inhibition, kinetic and docking studies
Fariba Peytam
Mehdi Adib
Bagher Larijani
Original Article 02 March 2019 Pages: 69 - 80
Four-component green synthesis of benzochromene derivatives using nano-KF/clinoptilolite as basic catalyst: study of antioxidant activity
Elham Ezzatzadeh
Zinatossadat Hossaini
Original Article 04 March 2019 Pages: 81 - 91
A quick accelerating microwave-assisted sustainable technique: permutated spiro-casing for imaging experiment
Animesh Mondal
Barnali Naskar
Chhanda Mukhopadhyay
Original Article 06 March 2019 Pages: 93 - 106
Regioselective synthesis of pyrimidine-fused tetrahydropyridines and pyridines by microwave-assisted one-pot reaction
Pooja Kumari
Rahul Yadav
Tasneem Parvin
Original Article 07 March 2019 Pages: 107 - 117
Synthesis and plant growth regulatory activities of 2′,3′-PhABA and iso-2′,3′-PhABA esters
Chuan Wan
Jiaqi Li
Zhaohai Qin
Original Article 09 March 2019 Pages: 119 - 130
Iodine/potassium iodide catalyst for the synthesis of trifluoromethylated quinazolines via intramolecular cyclization of 2,2,2-trifluoro-N-benzyl-N′-arylacetimidamides
Ali Darehkordi
Elham Kazemi
Original Article 13 March 2019 Pages: 131 - 139
Two- and three-dimensional QSAR studies on hURAT1 inhibitors with flexible linkers: topomer CoMFA and HQSAR
Tingting Zhao
Zean Zhao
Yuanxin Tian
Original Article 13 March 2019 Pages: 141 - 154
Synthesis and process optimization of symmetric and unsymmetric barbiturates C5-coupled with 2,1-benzisoxazoles
João L. Serrano
Pedro F. Soeiro
Paulo Almeida
Original Article 14 March 2019 Pages: 155 - 166
Application of 2,4-bis(halomethyl)quinoline: synthesis and biological activities of 2,4-bis(benzofuran-2-yl)- and 2,4-bis(aroxymethyl)quinolines
Yang Li
Qiqi Xu
Yu Chen
Original Article 20 March 2019 Pages: 167 - 178
Novel fused 1,2,3-triazolo-benzodiazepine derivatives as potent anticonvulsant agents: design, synthesis, in vivo, and in silico evaluations
Arefeh Shafie
Maryam Mohammadi-Khanaposhtani
Ahmad Reza Dehpour
Original Article 20 March 2019 Pages: 179 - 189
DBU-mediated annulation of 2-aryl-3-nitro-2H-chromenes with 1,3-cyclohexanediones for the synthesis of benzofuro[2,3-c]chromenone derivatives
Chenlu Dai
Zengyang Xie
Cunde Wang
Original Article 23 March 2019 Pages: 191 - 200
Preparation and characterization of a novel spherical cellulose–copper(II) oxide composite particles: as a heterogeneous catalyst for the click reaction
Seyedeh Fazileh Hamzavi
Sanaz Gerivani
Gholamhossein Shahverdizadeh
Original Article 26 March 2019 Pages: 201 - 209
Design, synthesis, in vivo and in vitro studies of 1,2,3,4-tetrahydro-9H-carbazole derivatives, highly selective and potent butyrylcholinesterase inhibitors
Roshanak Ghobadian
Roghaieh Esfandyari
Mohsen Amini
Original Article 29 March 2019 Pages: 211 - 223
A novel protocol for catalyst-free synthesis of fused six-member rings to triazole and pyrazole
Sedigheh Akrami
Bahador Karami
Mahnaz Farahi
Original Article 01 April 2019 Pages: 225 - 231
Identification of pyrrolo-pyridine derivatives as novel class of antibacterials
Mark S. Veselov
Yan A. Ivanenkov
Olga A. Dontsova
Original Article 04 April 2019 Pages: 233 - 239
Facile, efficient and one-pot access to diverse new functionalized aminoalkyl and amidoalkyl naphthol scaffolds via green multicomponent reaction using triethylammonium hydrogen sulfate ([Et₃NH][HSO₄]) as an acidic ionic liquid under solvent-free conditions
Elahe Hadadianpour
Behjat Pouramiri
Original Article 05 April 2019 Pages: 241 - 252
Adamantyl pyran-4-one derivatives and their in vitro antiproliferative activity
Vesna Petrović Peroković
Željka Car
Srđanka Tomić
Original Article 05 April 2019 Pages: 253 - 263
Synthesis, anti-proliferative activity, theoretical and ¹H NMR experimental studies of Morita–Baylis–Hillman adducts from isatin derivatives
Vinicius B. M. Brito
Gilmar F. Santos
Edilson B. Alencar-Filho
Original Article 06 April 2019 Pages: 265 - 281
Amine-functionalized graphene oxide nanosheets (AFGONs): an efficient bifunctional catalyst for selective formation of 1,4-dihydropyridines, acridinediones and polyhydroquinolines
Prasun Choudhury
Pranab Ghosh
Basudeb Basu
Short Communication 06 April 2019 Pages: 283 - 294
5-Endo-dig cyclizations in organic syntheses
Muhammad Aamir Sajid
Zulfiqar Ali Khan
Muhammad Usman
Comprehensive Review 05 March 2019 Pages: 295 - 317

Volume 24, Issue 1

One-pot organocatalytic/multicomponent approach for the preparation of novel enantioenriched non-natural selenium-based peptoids and peptide–peptoid conjugates

Substituent effect on inter-ring interaction in paracyclophanes

Lupenone is a good anti-inflammatory compound based on the network pharmacology

The periodic table of urea derivative: small molecules of zinc(II) and nickel(II) of diverse antimicrobial and antiproliferative applications

Combining ligand- and structure-based in silico methods for the identification of natural product-based inhibitors of Akt1

Single-stage synthesis of heterocyclic alkaloid-like compounds from (+)-camphoric acid and their antiviral activity

Design and synthesis of new imidazo[1,2-b]pyrazole derivatives, in vitro α-glucosidase inhibition, kinetic and docking studies

Four-component green synthesis of benzochromene derivatives using nano-KF/clinoptilolite as basic catalyst: study of antioxidant activity

A quick accelerating microwave-assisted sustainable technique: permutated spiro-casing for imaging experiment

Regioselective synthesis of pyrimidine-fused tetrahydropyridines and pyridines by microwave-assisted one-pot reaction

Synthesis and plant growth regulatory activities of 2′,3′-PhABA and iso-2′,3′-PhABA esters

Iodine/potassium iodide catalyst for the synthesis of trifluoromethylated quinazolines via intramolecular cyclization of 2,2,2-trifluoro-N-benzyl-N′-arylacetimidamides

Two- and three-dimensional QSAR studies on hURAT1 inhibitors with flexible linkers: topomer CoMFA and HQSAR

Synthesis and process optimization of symmetric and unsymmetric barbiturates C5-coupled with 2,1-benzisoxazoles

Application of 2,4-bis(halomethyl)quinoline: synthesis and biological activities of 2,4-bis(benzofuran-2-yl)- and 2,4-bis(aroxymethyl)quinolines

Novel fused 1,2,3-triazolo-benzodiazepine derivatives as potent anticonvulsant agents: design, synthesis, in vivo, and in silico evaluations

DBU-mediated annulation of 2-aryl-3-nitro-2H-chromenes with 1,3-cyclohexanediones for the synthesis of benzofuro[2,3-c]chromenone derivatives

Preparation and characterization of a novel spherical cellulose–copper(II) oxide composite particles: as a heterogeneous catalyst for the click reaction

Design, synthesis, in vivo and in vitro studies of 1,2,3,4-tetrahydro-9H-carbazole derivatives, highly selective and potent butyrylcholinesterase inhibitors

A novel protocol for catalyst-free synthesis of fused six-member rings to triazole and pyrazole

Identification of pyrrolo-pyridine derivatives as novel class of antibacterials

Facile, efficient and one-pot access to diverse new functionalized aminoalkyl and amidoalkyl naphthol scaffolds via green multicomponent reaction using triethylammonium hydrogen sulfate ([Et₃NH][HSO₄]) as an acidic ionic liquid under solvent-free conditions

Adamantyl pyran-4-one derivatives and their in vitro antiproliferative activity

Synthesis, anti-proliferative activity, theoretical and ¹H NMR experimental studies of Morita–Baylis–Hillman adducts from isatin derivatives

Amine-functionalized graphene oxide nanosheets (AFGONs): an efficient bifunctional catalyst for selective formation of 1,4-dihydropyridines, acridinediones and polyhydroquinolines

5-Endo-dig cyclizations in organic syntheses

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