Hydroxy- and alkoxyanilides of 6-hydroxy-2-methyl-4-oxo-2,4-dihydro-1H-pyrrolo[3,2,1-ij]quinoline-5-carboxylic acids have been synthesized as potential diuretic agents. Features of their purification, their steric structure, and biological activity are discussed.
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*For Communication 200, see [1].
Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 9, pp. 1364–1371, September, 2011.
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Ukrainets, I.V., Golik, N.Y., Shemchuk, A.L. et al. 4-hydroxy-2-quinolones. 201*. Synthesis, structure, and diuretic activity of hydroxy- and alkoxy- anilides of 6-hydroxy-2-methyl-4-oxo-2,4-dihydro- 1H-pyrrolo[3,2,1-ij]quinoline-5-carboxylic acid. Chem Heterocycl Comp 47, 1122–1127 (2011). https://doi.org/10.1007/s10593-011-0882-1
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DOI: https://doi.org/10.1007/s10593-011-0882-1