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4-hydroxy-2-quinolones. 197*. The search for novel diuretics amongst halo-substituted 6-hydroxy-2-methyl-4-oxo-1,2-dihydro-4H-pyrrolo-[3,2,1-ij]quinoline-5-carboxylic acid anilides

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Chemistry of Heterocyclic Compounds Aims and scope

A targeted synthesis of a series of halo-substituted 6-hydroxy-2-methyl-4-oxo-1,2-dihydro-4H-pyrrolo-[3,2,1-ij]quinoline-5-carboxylic acid anilides have been carried out. Peculiarites of the 1H NMR spectra and the results of investigating the diuretic activity of these compounds are discussed.

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Authors and Affiliations

  1. National University of Pharmacy, 53 Pushkinska St., Kharkiv, 61002, Ukraine

    I. V. Ukrainets, N. Yu. Golik, A. L. Shemchuk, O. I. Naboka & Yu. V. Voronina

  2. Taras Shevchenko National University, 64 Volodimirska St., Kyiv, 01033, Ukraine

    A. V. Turov

Authors
  1. I. V. Ukrainets
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  2. N. Yu. Golik
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  3. A. L. Shemchuk
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  4. O. I. Naboka
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  5. Yu. V. Voronina
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  6. A. V. Turov
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Corresponding author

Correspondence to I. V. Ukrainets.

Additional information

*For Communication 196, see [1].

Translated from Khimiya Geterotsiklicheskikh Soedinenii, No. 7, pp. 1009–1017, July, 2011. Original article submitted June 22, 2010.

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Ukrainets, I.V., Golik, N.Y., Shemchuk, A.L. et al. 4-hydroxy-2-quinolones. 197*. The search for novel diuretics amongst halo-substituted 6-hydroxy-2-methyl-4-oxo-1,2-dihydro-4H-pyrrolo-[3,2,1-ij]quinoline-5-carboxylic acid anilides. Chem Heterocycl Comp 47, 826–832 (2011). https://doi.org/10.1007/s10593-011-0842-9

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  • DOI: https://doi.org/10.1007/s10593-011-0842-9

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