1. Pyrrolo[2,1-f][1,2,4]triazine: a promising fused heterocycle to target kinases in cancer therapy

   • Sarbjit Singh
   • Divya Utreja
   • Vimal Kumar

   Review Article 13 November 2021 Pages: 1 - 25

   

2. Drug repositioning of benzimidazole anthelmintics in the treatment of cryptococcosis: a review

   • Emanuel A. M. Oliveira
   • Gabriella F. Ferreira
   • Karen L. Lang

   Review Article 23 November 2021 Pages: 26 - 39

   

3. A review of natural products, their effects on SARS-CoV-2 and their utility as lead compounds in the discovery of drugs for the treatment of COVID-19

   • Robert L. Chapman
   • Shridhar V. Andurkar

   Review Article 02 December 2021 Pages: 40 - 51

   

4. Synthesis of new calix[4]arene derivatives and evaluation of their cytotoxic activity

   • Mehmet Oguz
   • Ayse Yildirim
   • Mustafa Yilmaz

   Original Research 28 October 2021 Pages: 52 - 59

   

5. Synthesis and potential antimicrobial activity of novel α-aminophosphonates derivatives bearing substituted quinoline or quinolone and thiazole moieties

   • Bilal Litim
   • Abdelghani Djahoudi
   • Abbes Boukhari

   Original Research 02 November 2021 Pages: 60 - 74

   

6. Conjugates of Tetramethylpyrazine’ metabolites and amino acid as potential antiplatelet agents

   • Yongxi Dong
   • Shuxia Wu
   • Li Dong

   Original Research 12 November 2021 Pages: 75 - 84

   

7. Sorbents for treatment of hereditary hemochromatosis

   • Anna Wilson
   • Leslie Laguna
   • Mark B. Shiflett

   Original Research 13 November 2021 Pages: 85 - 93

   

8. Design, synthesis, and antifungal activity evaluation of novel 2-cyano-5-oxopentanoic acid derivatives as potential succinate dehydrogenase inhibitors

   • Xue-song Wang
   • Xiao-rong Tang
   • Yong-zhan Mai

   Original Research 13 November 2021 Pages: 94 - 107

   

9. Synthesis and biological activities of new phthalimide and thiazolidine derivatives

   • Flaviana A. Santos
   • Marcel L. Almeida
   • Ivan da Rocha Pitta

   Original Research 17 November 2021 Pages: 108 - 119

   

10. Synthesis, antiproliferative, and antimicrobial properties of novel phthalimide derivatives

    • Chun-Lan Chi
    • Lu Xu
    • Bao-Quan Chen

    Original Research 23 November 2021 Pages: 120 - 131

    

11. Design, synthesis, and evaluation of functionalized 5-(4-arylpiperazin-1-yl)-N-arylpentanamides as selective dopamine D₃ receptor ligands

    • Benjamin E. Blass
    • Peng-Jen Chen
    • Robert R. Luedtke

    Original Research 26 November 2021 Pages: 132 - 145

    

12. Synthesis, in vitro and in silico enzyme (COX-1/2 & LOX-5), free radical scavenging and cytotoxicity profiling of the 2,4-dicarbo substituted quinazoline 3-oxides

    • Malose J. Mphahlele
    • Eugene E. Onwu
    • Yee Siew Choong

    Original Research 26 November 2021 Pages: 146 - 164

    

13. Phloroglucinol derivatives as anti-tumor agents: synthesis, biological activity evaluation and molecular docking studies

    • Fuli Zhang
    • Qingfu Lai
    • Lianbao Ye

    Original Research 30 November 2021 Pages: 165 - 176

    

14. Design and synthesis of caffeic acid derivatives and evaluation of their inhibitory activity against Pseudomonas aeruginosa

    • Yun-feng Zeng
    • Ya-lun Su
    • Ping-hua Sun

    Original Research 04 January 2022 Pages: 177 - 194

    

15. Design, synthesis and SAR of novel sulfonylurea derivatives for the treatment of Diabetes mellitus in rats

    • Farid M. Sroor
    • Wahid M. Basyouni
    • Azza F. Arafa

    Original Research 28 November 2021 Pages: 195 - 206