1. Quinoxaline 1,4-di-N-oxides: a review of the importance of their structure in the development of drugs against infectious diseases and cancer

   • Socorro Leyva-Ramos
   • Alberto Pedraza-Alvarez

   Review Article 05 May 2021 Pages: 1175 - 1184

   

2. New synthetic 1H-1,2,3-triazole derivatives of 3-O-acetyl-β-boswellic acid and 3-O-acetyl-11-keto-β-boswellic acid from Boswellia sacra inhibit carbonic anhydrase II in vitro

   • Satya Kumar Avula
   • Najeeb Ur Rehman
   • Ahmed Al-Harrasi

   Original Research 31 March 2021 Pages: 1185 - 1198

   

3. Diversifying the xanthine scaffold for potential phosphodiesterase 9A inhibitors: synthesis and validation

   • Nivedita Singh
   • Akhtar Hussain Malik
   • Sanjukta Patra

   Original Research 10 April 2021 Pages: 1199 - 1219

   

4. Synthesis, molecular docking, and biological evaluation of nitroimidazole derivatives as potent urease inhibitors

   • Meysam Talebi
   • Elham Hamidian
   • Massoud Amanlou

   Original Research 12 April 2021 Pages: 1220 - 1229

   

5. A comparative study of the recent most potent small-molecule PD-L1 inhibitors: what can we learn?

   • Mei Liu
   • Yu Zhang
   • Xiaowu Dong

   Original Research 13 April 2021 Pages: 1230 - 1239

   

6. Syntheses and anticancer activities of novel glucosylated (−)-epigallocatechin-3-gallate derivatives linked via triazole rings

   • Bo-Ya Shi
   • Ze-Hao Wang
   • Jun Sheng

   Original Research 26 April 2021 Pages: 1240 - 1248

   

7. 2-(3-Hydroxybenzyl)benzo[d]isothiazol-3(2H)-one Mannich base derivatives as potential multifunctional anti-Alzheimer’s agents

   • Yuxi He
   • Ganyuan Xiao
   • Yong Deng

   Original Research 28 April 2021 Pages: 1249 - 1264

   

8. Ginkgolide B derivative synthesis and their effects on the viability of SKOV3 cells

   • ZiLi Feng
   • ZhiBin Zhu
   • ZhengDong Zhao

   Original Research 07 May 2021 Pages: 1265 - 1272

   

9. Synthesis, in vitro and in silico enzymatic inhibition assays, and toxicity evaluations of new 4,5-diphenylimidazole-N-phenylacetamide derivatives as potent α-glucosidase inhibitors

   • Maryam Mohammadi-Khanaposhtani
   • Atefeh Nikraftar
   • Mohammad Mahdavi

   Original Research 15 May 2021 Pages: 1273 - 1283

   

10. Novel ferrocenyl chalcone derivatives as antibacterial agents: is there a solution to the problem?

    • Elecia J. Henry
    • Charles Thomas Bennett
    • John P. Cassella

    Original Research 17 May 2021 Pages: 1284 - 1293

    

11. Discovery of N-phenyl-1-(phenylsulfonamido)cyclopropane-1-carboxamide analogs as NLRP3 inflammasome inhibitors

    • Wanwan Li
    • Zhongqiang Cao
    • Na Ye

    Original Research 16 May 2021 Pages: 1294 - 1308

    

12. Synthesis and evaluation of cyclic nitrone derivatives as potential anti-cancer agents

    • Wei Zhou
    • Dongyan Ju
    • Jinbo Zhao

    Original Research 18 May 2021 Pages: 1309 - 1316