Indazole scaffold: a generalist for marketed and clinical drugs Yaquan CaoChunying LuoChunli Wu Review Article 25 November 2020 Pages: 501 - 518
Thiazole-based and thiazolidine-based protein tyrosine phosphatase 1B inhibitors as potential anti-diabetes agents Kexin ChenXu YaoXing Zheng Review Article 25 November 2020 Pages: 519 - 534
DDR1 and DDR2: a review on signaling pathway and small molecule inhibitors as an anticancer agent Gurubasavaraja Swamy Purawarga MatadaArka DasAbhishek Ghara Review Article 12 January 2021 Pages: 535 - 551
Benzilydene and thiourea derivatives as new classes of carbonic anhydrase inhibitors: an in vitro and molecular docking study Shama QaiserMohammad S. MubarakAneela Maalik Original Research 17 November 2020 Pages: 552 - 563
Simple methods of modification of daunorubicin on the daunosamine nitrogen atom Valery K. BrelAleksandra A. MoiseevaZinaida S. Klemenkova Original Research 20 November 2020 Pages: 564 - 573
Biological targets of 92 alkaloids isolated from Papaver genus: a perspective based on in silico predictions Omer BayazeidFunda N. Yalçın Original Research 21 November 2020 Pages: 574 - 585
Synthesis and biological evaluation of novel N-substituted nipecotic acid derivatives with tricyclic cage structures in the lipophilic domain as GABA uptake inhibitors Heinrich-Karl A. RudyGeorg HöfnerKlaus T. Wanner Original Research Open access 22 November 2020 Pages: 586 - 609
Antioxidant and acetylcholinesterase inhibition activity of aliphatic and aromatic edaravone derivatives Victor Wagner Barajas-CarrilloArturo Estolano-CobiánIván Córdova-Guerrero Original Research 23 November 2020 Pages: 610 - 623
Design, synthesis and biological evaluation of Schiff’s base derivatives as multifunctional agents for the treatment of Alzheimer’s disease Jian ShiYi ZhouZhipei Sang Original Research 25 November 2020 Pages: 624 - 634
Design and synthesis of nature-inspired chromenopyrroles as potential modulators of mitochondrial metabolism Paul SchilfVunnam SrinivasuluTaleb H. Al-Tel Original Research 30 November 2020 Pages: 635 - 646
RF-3192C and other polyketides from the marine endophytic Aspergillus niger ASSB4: structure assignment and bioactivity investigation Manar M, MahmoudAhmed S, Abdel-RazekMohamed Shaaban Original Research 01 December 2020 Pages: 647 - 654
Theoretical and experimental verification of molecular properties of novel benzamide derivatives using computational platforms and in vitro antibacterial activity Poonam M. WanjariSantosh N. MokaleVishwas N. Ingle Original Research 05 January 2021 Pages: 655 - 663
Phosphoramidate conjugates of 3′-azido-3′-deoxythymidine glycerolipid derivatives and amino acid esters: synthesis and anti-HIV activity Elizaveta S. DarnotukAndrei E. SiniavinNatal’ya S. Shastina Original Research 05 January 2021 Pages: 664 - 671
Facile one-pot sequential synthesis of novel diaryl urea derivatives and evaluation of their in vitro cytotoxicity on adenocarcinoma cells Fereshteh AzimianMaryam Hamzeh-MivehroudSiavoush Dastmalchi Original Research 07 January 2021 Pages: 672 - 684
Molecular hybridization based design and synthesis of new benzo[5,6]chromeno[2,3-b]-quinolin-13(14H)-one analogs as cholinesterase inhibitors Baswaraju MachaRavindra KulkarniAchaiah Garlapati Original Research 08 January 2021 Pages: 685 - 701
α-Glucosidase and α-amylase inhibition, molecular modeling and pharmacokinetic studies of new quinazolinone-1,2,3-triazole-acetamide derivatives Ali YavariMaryam Mohammadi-KhanaposhtaniMir Hamed Hajimiri Original Research 09 January 2021 Pages: 702 - 711
New amino acid clubbed Schiff bases inhibit carbonic anhydrase II, α-glucosidase, and urease enzymes: in silico and in vitro Kashif RafiqMajid KhanAhmed Al-Harrasi Original Research 09 January 2021 Pages: 712 - 728
Design, synthesis, docking study and urease inhibitory activity evaluation of novel 2-((5-amino-1,3,4-thiadiazol-2-yl)thio)-N-arylacetamide derivatives Mohammad Nazari MontazerMehdi AsadiMassoud Amanlou Original Research 12 January 2021 Pages: 729 - 742
N-(2,3,4,6-tetra-O-acetyl-β-d-glucopyranosyl)thiosemicarbazones of 6-alkoxy-2-oxo-2H-chromene-4-carbaldehydes: synthesis, evaluation of their antibacterial, anti-MRSA, antifungal activity, and docking study Vu Ngoc ToanNguyen Dinh ThanhNguyen Thi Thu Huong Original Research 13 January 2021 Pages: 743 - 759
Design and synthesis of newer N-benzimidazol-2yl benzamide analogues as allosteric activators of human glucokinase Sukhbir SinghSandeep AroraAjmer Singh Grewal Original Research 13 January 2021 Pages: 760 - 770