Cytotoxicity of some synthetic bis(arylidene) derivatives of cyclic ketones towards cisplatin-resistant human ovarian carcinoma cells Hinal PatelBegum MothiaPeter B. Wyatt Original research Open access 17 April 2020 Pages: 935 - 941
SNX-2112, an Hsp90 inhibitor, suppresses cervical cancer cells proliferation, migration, and invasion by inhibiting the Akt/mTOR signaling pathway Liang-Shun FuHong-Hong QiuZhong Liu Original Research 17 April 2020 Pages: 942 - 953
Synthesis and biological screening of a novel enaminone-grafted trithiocarbonate: a potential anticancer and antimicrobial agent Yahia Nasser MabkhotJamal M. A. KhaledYahya I. Asiri Original Research 21 April 2020 Pages: 954 - 961
Novel allosteric PARP1 inhibitors for the treatment of BRCA-deficient leukemia Elizabeth HewlettMonika TomaTomasz Skorski Original Research 19 April 2020 Pages: 962 - 978
Synthesis and antiviral activity of some pyrrolonyl substituted heterocycles as additives to enhance inactivated Newcastle disease vaccine Alaa R. I. MorsySayed K. RamadanMounir M. Elsafty Original Research 13 April 2020 Pages: 979 - 988
Synthesis and antimicrobial evaluation of new thiazolyl-1,2,3-triazolyl-alcohol derivatives Shivaji JagadaleAbhijit ChavanPravin C. Mhaske Original Research 20 April 2020 Pages: 989 - 999
Multifunctional quinoxaline-hydrazone derivatives with acetylcholinesterase and monoamine oxidases inhibitory activities as potential agents against Alzheimer’s disease Ulviye Acar ÇevikDerya OsmaniyeGülhan Turan Original Research 19 April 2020 Pages: 1000 - 1011
3D-QSAR, HQSAR, molecular docking, and new compound design study of 1,3,6-trisubstituted 1,4-diazepan-7-ones as human KLK7 inhibitors Le FuYi ChenMao Shu Original Research 05 May 2020 Pages: 1012 - 1029
Inhibitory activity on cholinesterases produced by aryl-phthalimide derivatives: green synthesis, in silico and in vitro evaluation Omar Ruiz-MacielItzia I. Padilla-MartínezJosé G. Trujillo-Ferrara Original Research 27 April 2020 Pages: 1030 - 1040
Oxygenated xanthones as P-glycoprotein modulators at the intestinal barrier: in vitro and docking studies Vera SilvaEva Gil-MartinsRenata Silva Original Research 29 April 2020 Pages: 1041 - 1057
Antiproliferative activity of naphthoquinones and indane carboxylic acids from lapachol against a panel of human cancer cell lines Kenneth O. EyongHerve L. KetsemenDaniel Romo Original Research 29 April 2020 Pages: 1058 - 1066
Microwave-assisted synthesis, molecular docking and anti-HIV activities of some drug-like quinolone derivatives Ahmed M. JassemAdil M. DhumadJasim M. Alshawi Original Research 29 April 2020 Pages: 1067 - 1076
Synthesis and evaluation of anticancer effect of a novel molecule based-on pillar[5]arene including multi quinoline units Canan Eroglu GunesMehmet Ali KaraselekErcan Kurar Original Research 27 April 2020 Pages: 1077 - 1083
Antibacterial and antibiofilm activities of synthetic analogs of 3-alkylpyridine marine alkaloids Karina M. S. HerreraFernanda K. da SilvaJaqueline M. S. Ferreira Original Research 04 May 2020 Pages: 1084 - 1089