Volume 27, Issue 5

Search all Medicinal Chemistry Research articles

May 2018

22 articles in this issue

The synthetic and therapeutic expedition of isoxazole and its analogs
Neetu Agrawal
Pradeep Mishra
Review Paper 27 February 2018 Pages: 1309 - 1344
Antimalarial activity of phytol derivatives: in vitro and in vivo study
Archana Saxena
Harish C. Upadhyay
Dnyaneshwar U. Bawankule
Original Research 03 March 2018 Pages: 1345 - 1354
Synthesis, cytotoxic activity and binding model analysis of novel isoxazole-docetaxel analogues with C3′-N modification
Ming Chen
Jiyuan Liu
Shengyong Zhang
Original Research 03 March 2018 Pages: 1355 - 1365
Design, synthesis and neuroprotective activities of novel cinnamide derivatives containing benzylpiperazine moiety
Yan Zhong
Xiaofeng Li
Bin Wu
Original Research 22 February 2018 Pages: 1366 - 1373
Synthesis, crystal structure, and antinociceptive effects of some new riluzole derivatives
Xiang-Long Wu
Liu Liu
Qi-Bing Mei
Original Research 02 March 2018 Pages: 1374 - 1383
Synthesis and anticancer activity of multisubstituted purines and xanthines with one or two propynylthio and aminobutynylthio groups
Alicja Kowalska
Krystian Pluta
Małgorzata Latocha
Original Research Open access 06 March 2018 Pages: 1384 - 1395
Heterocycles 44. Synthesis, characterization and anticancer activity of new thiazole ortho-hydroxychalcones
Fana-Maria Coman
Armelle T. Mbaveng
Valentin Zaharia
Original Research 28 February 2018 Pages: 1396 - 1407
Insulin releasing effect of some pure compounds from Moringa oleifera on mice islets
Rahman M. Hafizur
Kiran Maryam
Shaheen Faizi
Original Research 03 March 2018 Pages: 1408 - 1418
Synthesis, characterization, and bioactivity of new bisamidrazone derivatives as possible anticancer agents
Malath A. Al-Qtaitat
Mustafa M. El-Abadelah
Mohammad S. Mubarak
Original Research 28 February 2018 Pages: 1419 - 1431
Collection of alkenylcoumarin derivatives as Taq DNA polymerase inhibitors: SAR and in silico simulations
Ezequiel Bruna-Haupt
Hugo A. Garro
Carlos R. Pungitore
Original Research 07 March 2018 Pages: 1432 - 1442
Potentiation effects by usnic acid in combination with antibiotics on clinical multi-drug resistant isolates of methicillin-resistant Staphylococcus aureus (MRSA)
Guo-Ying Zuo
Rui-Chun Fu
Gen-Chun Wang
Original Research 09 March 2018 Pages: 1443 - 1448
The protective effects of MPLC isolated glycyrrhizin and mangiferin against brain toxicity in rats
Sylvia A. Boshra
Alaadin E. El-Haddad
Original Research 08 March 2018 Pages: 1449 - 1459
Inhibitory effects of α, β-unsaturated carbonyl-based compounds and their pyrazoline derivatives on the phagocytosis of human neutrophils
Laiba Arshad
Ibrahim Jantan
Shajarahtunnur Jamil
Original Research 07 March 2018 Pages: 1460 - 1471
Study of the effect of thiourea and N-ethyl groups on antibacterial activity of rhodamine-labeled 3,4-HPO iron chelators against Gram (+/−) bacteria
Tânia Moniz
Maria Feio
Maria Rangel
Original Research 12 March 2018 Pages: 1472 - 1477
Optimal axial alkylpyridinium-bonded tricationic P-porphyrin in photodynamic inactivation of Escherichia coli
Jin Matsumoto
Masahide Yasuda
Original Research 28 March 2018 Pages: 1478 - 1484
Derivatives of 4,5-dihydro (1H) pyrazoles as possible MAO-A inhibitors in depression and anxiety disorders: synthesis, biological evaluation and molecular modeling studies
Avinash C. Tripathi
Savita Upadhyay
Shailendra K. Saraf
Original Research 23 March 2018 Pages: 1485 - 1503
Dipeptides as linker for multicomponent presentation—a facile, robust, and high-bioactivity yielding strategy
Honnegowdanahally K. Kumara
Suhas Ramesh
Dase Channe Gowda
Original Research 23 March 2018 Pages: 1504 - 1516
Synthesis of nucleobase-neomycin conjugates and evaluation of their DNA binding, cytotoxicities, and antibacterial properties
Siwen Wang
Mandeep Singh
Liang Xue
Original Research 27 March 2018 Pages: 1517 - 1527
Synthesis and enzyme inhibitory kinetics of some novel 3-(substituted benzoyl)-2-thioxoimidazolidin-4-one derivatives as α-glucosidase/α-amylase inhibitors
Rabia Qamar
Aamer Saeed
Sung Yum Seo
Original Research 28 March 2018 Pages: 1528 - 1537
Evidences for the antitumor potentiality of Hemimycale arabica and Negombata magnifica mesohyls in hepatocellular carcinoma rat model
Hanaa H. Ahmed
Hanaa M. Rady
Soheir E. Kotob
Original Research 29 March 2018 Pages: 1538 - 1548
Effects of acetazolamide on the conformations and activities of digestive enzymes: pepsin and trypsin
Ting Liu
Xiaopeng Chen
Zhiqiang Ge
Original Research 28 March 2018 Pages: 1549 - 1557
Correction to: Antiacetylcholinesterase activity and docking studies with chlorogenic acid, cynarin and arzanol from Helichrysum stoechas (Asteraceae)
Letícia Silva
Ana Margarida Rodrigues
Maria Luísa Marques Serralheiro
Author Correction 02 March 2018 Pages: 1558 - 1558

Volume 27, Issue 5

The synthetic and therapeutic expedition of isoxazole and its analogs

Antimalarial activity of phytol derivatives: in vitro and in vivo study

Synthesis, cytotoxic activity and binding model analysis of novel isoxazole-docetaxel analogues with C3′-N modification

Design, synthesis and neuroprotective activities of novel cinnamide derivatives containing benzylpiperazine moiety

Synthesis, crystal structure, and antinociceptive effects of some new riluzole derivatives

Synthesis and anticancer activity of multisubstituted purines and xanthines with one or two propynylthio and aminobutynylthio groups

Heterocycles 44. Synthesis, characterization and anticancer activity of new thiazole ortho-hydroxychalcones

Insulin releasing effect of some pure compounds from Moringa oleifera on mice islets

Synthesis, characterization, and bioactivity of new bisamidrazone derivatives as possible anticancer agents

Collection of alkenylcoumarin derivatives as Taq DNA polymerase inhibitors: SAR and in silico simulations

Potentiation effects by usnic acid in combination with antibiotics on clinical multi-drug resistant isolates of methicillin-resistant Staphylococcus aureus (MRSA)

The protective effects of MPLC isolated glycyrrhizin and mangiferin against brain toxicity in rats

Inhibitory effects of α, β-unsaturated carbonyl-based compounds and their pyrazoline derivatives on the phagocytosis of human neutrophils

Study of the effect of thiourea and N-ethyl groups on antibacterial activity of rhodamine-labeled 3,4-HPO iron chelators against Gram (+/−) bacteria

Optimal axial alkylpyridinium-bonded tricationic P-porphyrin in photodynamic inactivation of Escherichia coli

Derivatives of 4,5-dihydro (1H) pyrazoles as possible MAO-A inhibitors in depression and anxiety disorders: synthesis, biological evaluation and molecular modeling studies

Dipeptides as linker for multicomponent presentation—a facile, robust, and high-bioactivity yielding strategy

Synthesis of nucleobase-neomycin conjugates and evaluation of their DNA binding, cytotoxicities, and antibacterial properties

Synthesis and enzyme inhibitory kinetics of some novel 3-(substituted benzoyl)-2-thioxoimidazolidin-4-one derivatives as α-glucosidase/α-amylase inhibitors

Evidences for the antitumor potentiality of Hemimycale arabica and Negombata magnifica mesohyls in hepatocellular carcinoma rat model

Effects of acetazolamide on the conformations and activities of digestive enzymes: pepsin and trypsin

Correction to: Antiacetylcholinesterase activity and docking studies with chlorogenic acid, cynarin and arzanol from Helichrysum stoechas (Asteraceae)

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