1. Halogenated 2-amino-4H-benzo[h]chromene derivatives as antitumor agents and the relationship between lipophilicity and antitumor activity

   • Ahmed M. El-Agrody
   • Ahmed M. Fouda
   • Essam Shawky A. E. H. Khattab

   Original Research 21 January 2017 Pages: 691 - 700

   

2. Identification of novel MEK1 inhibitors by pharmacophore and docking based virtual screening

   • Fangxia Zou
   • Yifei Yang
   • Xiaoming Zha

   Original Research 21 January 2017 Pages: 701 - 713

   

3. Design, synthesis and anti-cancer evaluation of a novel series of pyrazolo [1, 5-a] pyrimidine substituted diamide derivatives

   • A.K. Ajeesh Kumar
   • Yadav D. Bodke
   • Kishore G. Bhat

   Original Research 23 January 2017 Pages: 714 - 744

   

4. Novel indole-2-carboxylic acid linked 3-phenyl-2-alkoxy propanoic acids: Synthesis, molecular docking and in vivo antidiabetic studies

   • Amanjot Singh
   • Raman K. Verma
   • Rajiv Mall

   Original Research 23 January 2017 Pages: 745 - 759

   

5. Molecular modeling and structure–activity relationships studies of bioisoster hybrids of N-acylhydrazone and furoxan groups on cruzain

   • Ricardo A. M. Serafim
   • Tiago F. de Oliveira
   • Elizabeth I. Ferreira

   Original Research 24 January 2017 Pages: 760 - 769

   

6. Antituberculosis agents bearing the 1,2-disubstituted benzimidazole scaffold

   • Keng Yoon Yeong
   • Chee Wei Ang
   • Soo Choon Tan

   Original Research 24 January 2017 Pages: 770 - 778

   

7. Synthesis and anticancer activity evaluation of new isoindole analogues

   • Aytekin Köse
   • Yıldız Bal
   • Yunus Kara

   Original Research 25 January 2017 Pages: 779 - 786

   

8. Enantioselective synthesis and evaluation of 4-styryldihydropyrimidin-2-thiones as anti-proliferative agents

   • Han Yu
   • Guoyong Dai
   • Jiang-Jiang Tang

   Original Research 28 January 2017 Pages: 787 - 795

   

9. QSAR study of dipeptidyl peptidase-4 inhibitors based on the Monte Carlo method

   • Dušan Sokolović
   • Jasmina Ranković
   • Aleksandar M. Veselinović

   Original Research 28 January 2017 Pages: 796 - 804

   

10. Antidiabetic and allied biochemical roles of new chromeno-pyrano pyrimidine compounds: synthesis, in vitro and in silico analysis

    • Shrikant V. Hese
    • Rohan J. Meshram
    • Bhaskar S. Dawane

    Original Research 07 February 2017 Pages: 805 - 818

    

11. Design, synthesis and molecular docking of novel structural hybrids of substituted isatin based pyrazoline and thiadiazoline as antitumor agents

    • Kiran Gangarapu
    • Gouthami Thumma
    • Sriram Rekulapally

    Original Research 08 February 2017 Pages: 819 - 829

    

12. Synthesis, anti-17β-HSD and antiproliferative activity of new substituted 5-nitrosopyrimidine analogs

    • Nabeel A. Abdul-Rida
    • Tiba I. Mohammed
    • Martin Frotscher

    Original Research 10 February 2017 Pages: 830 - 840

    

13. A potential anticancer ability of 1,2-di(quinazolin-4-yl)diselane against gastric cancer cells through ROS signaling pathway

    • Jun Wei
    • Yong Yang
    • Danbin Jiang

    Original Research 13 February 2017 Pages: 841 - 848

    

14. α-Glucosidase inhibitory and antioxidant activity of furanocoumarins from Heracleum persicum

    • Hossein Dehghan
    • Yaghoub Sarrafi
    • Samad Nejad Ebrahimi

    Original Research 15 February 2017 Pages: 849 - 855

    

15. Synthesis of prenyloxy coumarin analogues and evaluation of their antioxidant, lipoxygenase (LOX) inhibitory and cytotoxic activity

    • Eleni Kavetsou
    • Leonidas Gkionis
    • Anastasia Detsi

    Original Research 17 February 2017 Pages: 856 - 866