1. Design and synthesis of new coumarin–chalcone/NO hybrids of potential biological activity

   • Hany A. El-Sherief
   • Gamal El-Din A. Abuo-Rahma
   • Rehab M. Abdel-baky

   Original Research 17 August 2017 Pages: 3077 - 3090

   

2. Albizia harveyi: phytochemical profiling, antioxidant, antidiabetic and hepatoprotective activities of the bark extract

   • Mansour Sobeh
   • Mona F. Mahmoud
   • Michael Wink

   Original Research 31 August 2017 Pages: 3091 - 3105

   

3. Synthesis and biological evaluation of some undecanone derivatives

   • Bharani Meka
   • Suryachandra Rao Ravada
   • Trimurtulu Golakoti

   Original Research 17 August 2017 Pages: 3106 - 3124

4. 3D QSAR and molecular docking studies of 4-alkoxy- and 4-acyloxy –phenyl ethylene thiosemicarbazone derivatives as tyrosinase inhibitors

   • Madhavi Madhavaram
   • Parthasarathy Tigulla

   Original Research 24 August 2017 Pages: 3125 - 3135

   

5. Synthesis, biological evaluation and in silico study of bis-thiourea derivatives as anticancer, antimalarial and antimicrobial agents

   • Ratchanok Pingaew
   • Nujarin Sinthupoom
   • Virapong Prachayasittikul

   Original Research 05 September 2017 Pages: 3136 - 3148

   

6. Radiosynthesis and biodistribution of ^99mTc-Sulfamethoxazole: a novel molecule for in-vivo infection imaging

   • Özge Uyaroğlu
   • Hasan Demiroğlu
   • Uğur Avcıbaşı

   Original Research 17 August 2017 Pages: 3149 - 3157

   

7. Design and synthesis of novel 2-(5-(4-aryl)-4,5-dihydro-1H-pyrazol-3-yl)-1-(substituted aminomethyl)-1H-benzimidazole as potent anticonvulsants

   • Pullagura Mallikarjuna Krishna Prasad
   • Raja Sundararajan

   Original Research 17 August 2017 Pages: 3158 - 3172

   

8. Discovery of tetrahydro-ß-carboline derivatives as a new class of phosphodiesterase 4 inhibitors

   • Ahmad Abdelwaly
   • Ismail Salama
   • Mohamed A. Helal

   Original Research 18 August 2017 Pages: 3173 - 3187

   

9. New quaternary ammonium pyridoxine derivatives: synthesis and antibacterial activity

   • Sergey V. Sapozhnikov
   • Nikita V. Shtyrlin
   • Yurii G. Shtyrlin

   Original Research 24 August 2017 Pages: 3188 - 3202

   

10. QSAR of antimycobacterial activity of benzoxazoles by optimal SMILES-based descriptors

    • Karel Nesměrák
    • Andrey A. Toropov
    • Ilkay Yildiz

    Original Research 17 August 2017 Pages: 3203 - 3208

11. α-Amylase and α-glucosidase inhibitory activities of the herbs of Artemisia dracunculus L. and its active constituents

    • Zühal Güvenalp
    • Hilal Özbek
    • Ömür L. Demirezer

    Original Research 17 August 2017 Pages: 3209 - 3215

    

12. Microwave-assisted synthesis, characterization and bioassay of acylhydrazone derivatives as influenza neuraminidase inhibitors

    • Mengwu Xiao
    • Jiao Ye
    • Aixi Hu

    Original Research 18 August 2017 Pages: 3216 - 3227

    

13. In silico studies on 2-substituted phenol quinazoline derivatives as RET receptor tyrosine kinase antagonists

    • Swapnil P. Bhujbal
    • Pavithra K. Balasubramanian
    • Seung Joo Cho

    Original Research 19 September 2017 Pages: 3228 - 3239

    

14. Evaluation of nitric oxide inhibition effect in LPS-stimulated RAW 264.7 macrophages by phytochemical constituents from Mesua beccariana, Mesua congestiflora, and Mesua ferrea

    • Soek Sin Teh
    • Gwendoline Cheng Lian Ee
    • Siau Hui Mah

    Original Research 09 August 2017 Pages: 3240 - 3246

    

15. Molecular docking and glucosidase inhibition studies of novel N-arylthiazole-2-amines and Ethyl 2-[aryl(thiazol-2-yl)amino]acetates

    • Ayesha Babar
    • Muhammad Yar
    • Ather Farooq Khan

    Original Research 18 August 2017 Pages: 3247 - 3261

    

16. Synthesis, antiprotozoal activity and cytotoxicity in U-937 macrophages of triclosan–hydrazone hybrids

    • Sebastian Vergara
    • Miguel Carda
    • Wilson Cardona Galeano

    Original Research 22 August 2017 Pages: 3262 - 3273

    

17. Discovery of potential neurodegenerative inhibitors in Alzheimer’s disease by casein kinase 1 structure-based virtual screening

    • Ricardo P. Rodrigues
    • Carlos H. T. P. da Silva

    Original Research 22 August 2017 Pages: 3274 - 3285

    

18. Interaction of intravenous immunoglobulin and three 20(S)-camptothecin analogs: maintaining higher circulatory levels of the biologically active species

    • Yongchun Liu
    • Yajun Li
    • Jianning Liu

    Original Research 05 September 2017 Pages: 3286 - 3295

    

19. Antibacterial effect on mature biofilms of oral streptococci and antioxidant activity of 3β,6β,16β-trihydroxylup-20(29)-ene from Combretum leprosum

    • Francisco Flávio Vasconcelos Evaristo
    • Mayron Alves de Vasconcelos
    • Edson Holanda Teixeira

    Original Research 17 August 2017 Pages: 3296 - 3306

    

20. Bioguided chemical characterization of the antiproliferative fraction of edible pseudo bulbs of Malaxis acuminata D. Don by HPLC-ESI-QTOF-MS

    • Deepika Singh
    • Sunil Kumar
    • Brijesh Kumar

    Original Research 18 August 2017 Pages: 3307 - 3314

    

21. Rapid screening, separation, and detection of α-glucosidase inhibitors from Hedyotis diffusa by ultrafiltration–liquid chromatography tandem mass spectrometry–high-speed countercurrent chromatography

    • Xiaojing Yang
    • Lina Chen
    • Senlin Li

    Original Research 24 August 2017 Pages: 3315 - 3322

    

22. Suppression of PGE₂ production via disruption of MAPK phosphorylation by unsymmetrical dicarbonyl curcumin derivatives

    • Mohd Fadhlizil Fasihi Mohd Aluwi
    • Kamal Rullah
    • Kok Wai Lam

    Original Research 18 August 2017 Pages: 3323 - 3335

    

23. In vitro and in silico evaluation of 2-(substituted phenyl) oxazolo[4,5-b]pyridine derivatives as potential antibacterial agents

    • Gagandeep Kour Reen
    • Ashok Kumar
    • Pratibha Sharma

    Original Research 22 August 2017 Pages: 3336 - 3344

    

24. Design, synthesis and activity evaluation study of novel substituted N-sulfonyl homoserine lactone derivatives as bacterial quorum sensing inhibitors

    • Qi Sun
    • Mingming Zhao
    • Fanhao Meng

    Original Research 12 September 2017 Pages: 3345 - 3353

    

25. An efficient synthesis of indolo[2,3-b]quinoline guanidine derivatives with their in vitro and in vivo study

    • Katarzyna Sidoryk
    • Marta Świtalska
    • Marcin Cybulski

    Original Research Open access 05 September 2017 Pages: 3354 - 3366

    

26. Synthesis and biological evaluation of disulfides bearing 1,2,4-triazole moiety as antiproliferative agents

    • Xue-Feng Wang
    • Shuai Zhang
    • Bao-Quan Chen

    Original Research 05 September 2017 Pages: 3367 - 3374

    

27. DNA interaction of bromomethyl-substituted acridines

    • Kazuya Harada
    • Takahiro Imai
    • Keiko Inami

    Original Research 24 August 2017 Pages: 3375 - 3383

    

28. Screening and isolating potential α-glucosidase inhibitors from Rhizoma Coptidis by ultrafiltration LC-PDA-ESI/MS combined with high-speed countercurrent chromatography and reverse-phase medium-pressure liquid chromatography

    • Ying Tang
    • Senlin Li
    • Yuchi Zhang

    Original Research 26 September 2017 Pages: 3384 - 3394

    

29. TQ-B3203, a potent proliferation inhibitor derived from camptothecin

    • Xiquan Zhang
    • Meng Cao
    • Ning Gu

    Original Research 28 August 2017 Pages: 3395 - 3406

    

30. Isolation, characterization and antiproliferative evaluation of constituents from stem extracts of Alafia barteri Oliv. Hook. F.

    • Abdulmumeen A. Hamid
    • Olapeju O. Aiyelaagbe
    • Arvind S. Negi

    Original Research 06 September 2017 Pages: 3407 - 3416