New acetylenic derivatives of betulin and betulone, synthesis and cytotoxic activity Ewa BębenekMonika Kadela-TomanekStanisław Boryczka Review Article Open access 01 September 2016 Pages: 1 - 8
Physicochemical characterization of two new Nitazoxanide analogs with antiparasitic activity Adriana Valladares-MéndezMirna García-FloresJulio C Rivera-Leyva Review Article 18 November 2016 Pages: 9 - 18
Geraniol attenuates osteoclast differentiation by suppressingNF-kB activity and expression of osteoclastogenic genes Vishwa DeepakMarlena C KrugerMagdalena Coetzee Original Research 27 August 2016 Pages: 19 - 26
Synthesis and in vitro evaluation of novel triazole/azide chalcones Fernanda C. G. EvangelistaMaralice O. BandeiraFernando P. Varotti Original Research 23 September 2016 Pages: 27 - 43
Synthesis and evaluation of novel benzene-ethanol bearing 1,2,4-triazole derivatives as potential antimicrobial agents Bochao LiDawei ZhangFeng Lin Original Research 23 September 2016 Pages: 44 - 51
Structural exploration of PPARγ modulators through pharmacophore mapping, fragment-based design, docking, and molecular dynamics simulation analyses Ashis NandyKunal RoyAchintya Saha Original Research 05 October 2016 Pages: 52 - 63
Cytotoxic activity of genistein-8-C-glucoside form Lupinus luteus L. and genistein against human SK-OV-3 ovarian carcinoma cell line Agata AntosiakKatarzyna MilowskaTeresa Gabryelak Original Research Open access 03 October 2016 Pages: 64 - 73
Discovery of novel small molecule EGFR inhibitory leads by structure and ligand-based virtual screening Priya MahajanNitasha SuriAmit Nargotra Original Research 07 October 2016 Pages: 74 - 92
TNF-α and IL-6 inhibitory effects of cyclic dipeptides isolated from marine bacteria Streptomyces sp Yedukondalu NalliShilpa GuptaAsif Ali Original Research 07 October 2016 Pages: 93 - 100
Anti-human immunodeficiency activity of novel 2-arylpyrrolidine analogs Ashot H. MartirosyanSahak P. GasparyanRaymond F. Schinazi Original Research 17 October 2016 Pages: 101 - 108
Synthesis and antimicrobial activity of novel quinoline derivatives bearing pyrazoline and pyridine analogues Nisheeth C. DesaiBonny Y. PatelBharti P. Dave Original Research 19 October 2016 Pages: 109 - 119
Synthesis of novel 1, 2, 4-triazolopyrimidines and their evaluation as antimicrobial agents Ameen A. Abu-HashemHoda A. R. HusseinKhadeja M. Abu-zied Original Research 21 October 2016 Pages: 120 - 130
Synthesis and in vitro evaluation of leishmanicidal activity of 7-hydroxy-4-phenylcoumarin derivatives Isael A. RosaLetícia de AlmeidaMarcelo H. dos Santos Original Research 27 October 2016 Pages: 131 - 139
1,5-Diaryl-3-oxo-1,4-pentadienes based on (4-oxopiperidin-1-yl)(aryl)methyl phosphonate scaffold: synthesis and antitumor properties Mikhail V. MakarovEkaterina Yu. RybalkinaValery K. Brel Original Research 01 November 2016 Pages: 140 - 152
Exploring the possible binding mode of trisubstituted benzimidazoles analogues in silico for novel drug designtargeting Mtb FtsZ Ding LiBo ChiJian Wan Original Research 05 November 2016 Pages: 153 - 169
Cyclic peroxides as promising anticancer agents: in vitro cytotoxicity study of synthetic ozonides and tetraoxanes on human prostate cancer cell lines Ivan A. YaremenkoMikhail A. SyroeshkinAlexander O. Terent’ev Original Research 09 November 2016 Pages: 170 - 179
In silico investigation of morpholines as novel class of trypanosomal triosephosphate isomerase inhibitors Akachukwu IbezimNgozi Justina NwodoChika J. Mba Original Research 09 November 2016 Pages: 180 - 189
Design, synthesis and biological evaluation of 1,3,4-oxadiazoles as promising anti-inflammatory agents Vishwanathan Balasubramanya IyerBannimath GurupadayyaRavandur Shivanna Chandan Original Research 10 November 2016 Pages: 190 - 204
Identification of new insulin growth factor receptor-1 (IGF-1R) inhibitors via exploring ATPas kinase domain of IGF-1R through virtual screening Mansi GargMonika ChauhanRaj Kumar Original Research 14 November 2016 Pages: 205 - 219
Chemical constituents of Piper aduncum and their inhibitory effects on soluble epoxide hydrolase and tyrosinase Bui Thi Thuy LuyenNguyen Phuong ThaoYoung Ho Kim Original Research 15 November 2016 Pages: 220 - 226
5-farnesyloxycoumarin: a potent 15-LOX-1 inhibitor, prevents prostate cancer cell growth Ala OrafaieHamid SadeghianMaryam M. Matin Original Research 15 November 2016 Pages: 227 - 234
Benzenesulfonamides bearing pyrrolidinone moiety as inhibitors of carbonic anhydrase IX: synthesis and binding studies Kęstutis RutkauskasAsta ZubrienėDaumantas Matulis Original Research 15 November 2016 Pages: 235 - 246
Dihydrofolate reductase inhibitors: a quantitative structure–activity relationship study using 2D-QSAR and 3D-QSAR methods Juan C. Garro MartinezMatias F. AndradaMario R. Estrada Original Research 15 November 2016 Pages: 247 - 261
Synthesis of novel α,α-difluoro-β-hydroxycarbonyl pyrazole derivatives as antioxidant, anti-inflammatory and anticancer agents Salman MukarramBabasaheb P. BandgarHemant V. Chavan Original Research 16 November 2016 Pages: 262 - 273
Natural diarylheptanoid compounds from Curcuma comosa Roxb. promote differentiation of mouse myoblasts C2C12 cells selectively via ER alpha receptors Chittipong TipbunjongYindee KitiyanantChumpol Pholpramool Original Research 18 November 2016 Pages: 274 - 286