Structure–activity relationship study of secondary metabolites from Mesua beccariana, Mesua ferrea and Mesua congestiflora for anti-cholinesterase activity Soek Sin TehGwendoline Cheng Lian EeZuraini Ahmad Original Research 20 February 2016 Pages: 819 - 823
Broad-spectrum antiproliferative activity of a series of 6-(4-fluorophenyl)-5-(2-substituted pyrimidin-4-yl)imidazo[2,1-b]thiazole derivatives Mohammed S. Abdel-MaksoudMohammed I. El-GamalChang-Hyun Oh Original Research 23 February 2016 Pages: 824 - 833
QSAR study of diarylalkylimidazole and diarylalkyltriazole aromatase inhibitors Razieh GhodsiBahram Hemmateenejad Original Research 23 February 2016 Pages: 834 - 842
Synthesis, characterization and biological evaluation of some novel fluoroquinolones Neelanjana PanditKamal ShahPradeep Mishra Original Research 23 February 2016 Pages: 843 - 851
An antioxidant mechanism of morphine and related derivatives Rosivaldo S. BorgesJoyce K. L. ValeAlbérico B. F. da Silva Original Research 23 February 2016 Pages: 852 - 857
Design, synthesis and biological evaluation of new tricyclic spiroisoxazoline derivatives as selective COX-2 inhibitors and study of their COX-2 binding modes via docking studies Hoda AbolhasaniSiavoush DastmalchiAfshin Zarghi Original Research 24 February 2016 Pages: 858 - 869
A new class of phenylhydrazinylidene derivatives as inhibitors of Staphylococcus aureus biofilm formation Stella CascioferroBenedetta MaggioGiuseppe Daidone Original Research 24 February 2016 Pages: 870 - 878
Synthesis and in vitro cancer cell growth inhibition evaluation of 11-amino-modified 5-Me-indolo[2,3-b]quinolines and their COMPARE analyses Masashi OkadaZhen-Wu MeiTsutomu Inokuchi Original Research 25 February 2016 Pages: 879 - 892
A convenient synthesis, reactions and biological studies of some novel selenolo[2,3-c]pyrazole compounds as antimicrobial and anti-inflammatory agents Remon M. ZakiYasser A. El-OssailyAhmed A. Geies Original Research 27 February 2016 Pages: 893 - 908
Microwave-assisted synthesis and biological evaluation of carbazole-based chalcones, aurones and flavones D. AshokS. RaviS. D. S. Murthy Original Research 29 February 2016 Pages: 909 - 922
Synthesis, antimicrobial and nematicidal evaluation of a new class of triazolo[4,3-c]quinazolinylthiazolidinones Cherkupally Sanjeeva ReddyGaddam Rajesh KumarBommineni Sunitha Original Research 29 February 2016 Pages: 923 - 931
Synthesis of novel N-acyl-β-d-glucopyranosylamines and ureas as potential lead cytostatic agents Vanessa ParmenopoulouStella MantaDimitri Komiotis Original Research 29 February 2016 Pages: 932 - 940
Synthesis and anticancer activity study of indolyl hydrazide–hydrazones Swapna SundareeBuchi Reddy VaddulaDalip Kumar Original Research 03 March 2016 Pages: 941 - 950
Synthesis and biological evaluation of quinolines, thiazolo[3,2-a]pyrimidines, thiadiazolo[3,2-a]pyrimidines and triazolo[3,4-b][1,3,4]thiadiazepines as antimicrobial agents Seema SahiSatya Paul Original Research 03 March 2016 Pages: 951 - 969
Synthesis and antimicrobial evaluation of hydrazones derived from 4-methylbenzenesulfonohydrazide in aqueous medium Sunita GhiyaYogesh C. Joshi Original Research 03 March 2016 Pages: 970 - 976
Design, synthesis and biological activity evaluation of novel pefloxacin derivatives as potential antibacterial agents Tejeswara Rao AllakaNaveen PolkamJaya Shree Anireddy Original Research 03 March 2016 Pages: 977 - 993
Synthesis and evaluation of some novel N-substituted rhodanines for their anticancer activity Sulaiman Ali MuhammadSubban RaviArumugam Thangamani Original Research 03 March 2016 Pages: 994 - 1004
IDX-184 is a superior HCV direct-acting antiviral drug: a QSAR study Abdo A. ElfikyWael M. Elshemey Original Research 04 March 2016 Pages: 1005 - 1008
Influence of the methyl position on the binding of 5-epi-taiwaniaquinone G to HSA investigated by spectrofluorimetry and molecular modeling Zhigang LiJinqian WangJunbiao Chang Original Research 07 March 2016 Pages: 1009 - 1019
Determination and isolation of potential α-glucosidase and xanthine oxidase inhibitors from Trifolium pratense L. by ultrafiltration liquid chromatography and high-speed countercurrent chromatography Yueqi WangYing TangYuchi Zhang Original Research 07 March 2016 Pages: 1020 - 1029