Design and development of oxobenzimidazoles as novel androgen receptor antagonists R. ElancheranK. SaravananJibon Kotoky Original Research 21 January 2016 Pages: 539 - 552
Synthesis, molecular docking and antimicrobial evaluation of novel benzoxazole derivatives Tugba Ertan-Bolelliİlkay YildizSelda Ozgen-Ozgacar Original Research 22 January 2016 Pages: 553 - 567
Synthesis and in vitro biological activities of ferrocenyl–chalcone amides Frans J. SmitJaco J. BezuidenhoutDavid D. N’Da Original Research 25 January 2016 Pages: 568 - 584
Combined pharmacophore models as virtual screening protocol against BRD4(1) inhibitor Yifei YangFangxia ZouJinpei Zhou Original Research 27 January 2016 Pages: 585 - 595
Modulation of indole ring annulation in ergoline template: chemistry, receptor binding and in vivo pharmacology with 6-OHDA model of Parkinson’s disease J. B. Senthil KumarRita KumariPratibha Mehta Luthra Original Research 01 February 2016 Pages: 596 - 608
Pharmacophore and docking-based hierarchical virtual screening for the designing of aldose reductase inhibitors: synthesis and biological evaluation Bhawna VyasManjinder SinghBaldev Singh Original Research 03 February 2016 Pages: 609 - 626
Synthesis and biological evaluation of novel resveratrol-oxadiazole hybrid heterocycles as potential antiproliferative agents M. S. R. MurtyRaju PenthalaN. Jain Original Research 04 February 2016 Pages: 627 - 643
Synthesis, characterization and antimicrobial activity of 4-((1-benzyl/phenyl-1H-1,2,3-triazol-4-yl)methoxy)benzaldehyde analogues Kashmiri LalPinki YadavAshwani Kumar Original Research 08 February 2016 Pages: 644 - 652
Structural characterization of human CRTh2: a combined homology modeling, molecular docking and 3D-QSAR-based in silico approach Sathya BabuSanthosh Kumar NagarajanThirumurthy Madhavan Original Research 09 February 2016 Pages: 653 - 671
Design and development of pyrrole carbaldehyde: an effective pharmacophore for enoyl-ACP reductase Shrinivas D. JoshiDevendra KumarTejraj M. Aminabhavi Original Research 09 February 2016 Pages: 672 - 689
Alkyl phenols, alkenyl cyclohexenones and other phytochemical constituents from Lannea rivae (chiov) Sacleux (Anacardiaceae) and their bioactivity Dorothy A. OkothHoseah M. AkalaNeil A. Koorbanally Original Research 13 February 2016 Pages: 690 - 703
Soluble epoxide hydrolase inhibitory activity by rhizomes of Kaempferia parviflora Wall. ex Baker Nguyen Phuong ThaoBui Thi Thuy LuyenYoung Ho Kim Original Research 16 February 2016 Pages: 704 - 711
Synthesis, biological valuation, and QSAR studies of novel pyrazole bearing pyridyl oxadiazole analogues as potential antimicrobial agents N. C. DesaiG. M. KotadiyaP. C. Jha Original Research 16 February 2016 Pages: 712 - 727
The novel coumarin[3,2-c]thiophene and its hydroxamic acid and ureido derivatives: synthesis and cytostatic activity evaluations Karlo WittineIvana RatkajMladen Mintas Original Research 17 February 2016 Pages: 728 - 737
Synthesis and in vitro cytotoxic evaluation of new triazole derivatives based on artemisinin via click chemistry Le Huy BinhNguyen Thi Thuy VanTran Khac Vu Original Research 17 February 2016 Pages: 738 - 750
2-Amino-2,3-dihydro-1H-2λ5-[1,3,2]diazaphospholo[4,5-b]pyridin-2-one-based urea and thiourea derivatives: synthesis, molecular docking study and evaluation of anti-inflammatory and antimicrobial activities Subba Rao DevineniMadhava GollaUsha Rani Asupathri Original Research 17 February 2016 Pages: 751 - 768
Synthesis, crystal structure, biological evaluation, electronic aspects of hydrogen bonds, and QSAR studies of some new N-(substituted phenylurea) diazaphosphore derivatives as anticancer agents Niloufar DorostiBahram DelfanAli Asghar Ebrahimi Valmoozi Original Research 18 February 2016 Pages: 769 - 789
Synthesis, biological evaluation and molecular docking of novel coumarin incorporated triazoles as antitubercular, antioxidant and antimicrobial agents Mubarak H. ShaikhDnyaneshwar D. SubhedarSandip S. Shinde Original Research 19 February 2016 Pages: 790 - 804
Antidiabetic potential and enzyme kinetics of benzothiazole derivatives and their non-bonded interactions with α-glucosidase and α-amylase Ninad V. PuranikHemalata M. PuntambekarPratibha Srivastava Original Research 19 February 2016 Pages: 805 - 816
Erratum to: Synthesis, antimicrobial activity and docking studies of new N-ethyl-3-indolyl heterocycles Wael A. El-SayedHebat-Allah S. AbbasTomasz Magdziarz Erratum 28 January 2016 Pages: 817 - 817