A review on pharmacophoric designs of antiproliferative agents Anil RanaJimi Marin AlexRaj Kumar Review Article 06 August 2014 Pages: 903 - 920
Synthesis, cytotoxic activity, and computational analysis of N10-substituted acridone analogs Rajesh KumarMalkeet Singh BahiaOm Silakari Original Research 29 July 2014 Pages: 921 - 933
3D-QSAR and docking study on 3-benzimidazol-2-ylhydroquinolin-2-one derivatives as VEGFR-2 tyrosine kinase inhibitors Cong-min KangDong-qing LiuYing-tao Lv Original Research 29 July 2014 Pages: 934 - 943
Multistep synthesis of 1-[{(5-alkenyl/hydroxyalkenylsubstituted)-1,3,4-oxadiazol-2-yl}-methyl]-2-methyl-1H-benzimidazole series and in vitro anticancer screening, SAR studies Himani VarshneyAiman AhmadMohammad Owais Original Research 29 July 2014 Pages: 944 - 953
Synthesis and antimicrobial activity of 3-aroyl-4-heteroaryl pyrroles and pyrazoles Shaik Sharafuddin BashaPutta Ramachandra ReddyTartte Vijaya Original Research 29 July 2014 Pages: 954 - 964
Chemical constituents, the stereochemistry of 3-hydroxy furonaphthoquinones from the root bark of Newbouldia laevis Seem (Bignoniaceae), and screening against Onchocerca ochengi parasites Kenneth O. EyongHerve L. KetsemenGabriel N. Folefoc Original Research 29 July 2014 Pages: 965 - 969
Synthesis and antimicrobial activity of pyrazolyl benzoxazoles, benzothiazoles and benzimidazoles Lingaladinne Mallikarjuna ReddyTalapuru Bhanu PrakashVenkatapuram Padmavathi Original Research 29 July 2014 Pages: 970 - 979
Buddlejol, a new α-chymotrypsin inhibitor from Buddleja asiatica Farman Ali KhanNasir Mehmood KhanDerek James Maitland Original Research 29 July 2014 Pages: 980 - 986
QSAR and mechanisms of radical scavenging activity of phenolic and anilinic compounds using structural, electronic, kinetic, and thermodynamic parameters Hussein M. AliIsra H. Ali Original Research 31 July 2014 Pages: 987 - 998
Atom-based QSAR and 3D QSAR using pharmacophore based alignment for discovery of nimesulide-derived SKBR-3 cell line inhibitors Arpita Das Choudhury Original Research 31 July 2014 Pages: 999 - 1012
Synthesis of cis-4-guanidino-l-proline and 1-carbamimidoyl-l-proline derivatives as influenza neuraminidase inhibitors Yuanchao XieDongqing XuWenfang Xu Original Research 01 August 2014 Pages: 1013 - 1017
Synthesis, 3D-QSAR and docking studies of pyrimidine nitrile-pyrazoline: a novel class of hybrid antimalarial agents Akranth MarellaMymoona AkhterMohammad Mumtaz Alam Original Research 01 August 2014 Pages: 1018 - 1037
Structural insights into mode of actions of novel substituted 4- and 6-azaindole-3-carboxamides analogs as renin inhibitors: molecular modeling studies Mukesh C. Sharma Original Research 02 August 2014 Pages: 1038 - 1059
3D-QSAR studies of dipeptidyl peptidase-4 inhibitors using various alignment methods Bhumika D. PatelManjunath D. Ghate Original Research 02 August 2014 Pages: 1060 - 1069
Synthesis of novel 5-methyl pyrazol-3-one derivatives and their in vitro cytotoxic evaluation Pritam N. DubeShweta S. BulePravin R. Dighe Original Research 03 August 2014 Pages: 1070 - 1076
Green synthesis and in silico investigation of dihydro-2H-benzo[1,3]oxazine derivatives as inhibitors of Mycobacterium tuberculosis Rahul D. KambleShrikant V. HeseBhaskar S. Dawane Original Research 06 August 2014 Pages: 1077 - 1088
Estrogenic and Anti-Alzheimer’s studies of Zingiber officinalis as well as Amomum subulatum Roxb.: the success story of dry techniques Ashwani KumarRuchika GoyalParvin Kumar Original Research 06 August 2014 Pages: 1089 - 1097
Mixed 2D–3D-LQTA-QSAR study of a series of Plasmodium falciparum dUTPase inhibitors Rodolfo André de Araújo SantosCarolina Arruda BrazEuzébio Guimarães Barbosa Original Research 06 August 2014 Pages: 1098 - 1111
Bioactive chemical constituents from the root of Clerodendrum phlomidis Akhilesh K. YadavJay Prakash ThakurMadan M. Gupta Original Research 06 August 2014 Pages: 1112 - 1118
Synthesis of N-(3-picolyl)-based 1,3,2λ5-benzoxazaphosphinamides as potential 11β-HSD1 enzyme inhibitors Satheesh Krishna BalamSuresh Kumar KrishnammagariSuresh Reddy Cirandur Original Research 06 August 2014 Pages: 1119 - 1135
Insights into activity enhancement of 4-aminoquinoline-based hybrids using atom-based and field-based QSAR studies K. Kranthi RajSunny ManoharDiwan S. Rawat Original Research 06 August 2014 Pages: 1136 - 1154
3-Indol carboxaldehyde, an imidazole synthesized from naphthoquinone β-lapachone downregulates Candida albicans biofilm José Alexandre da Rocha CurveloAnna Lea Silva BarretoRosangela Maria de Araújo Soares Original Research 06 August 2014 Pages: 1155 - 1161
Design, synthesis, characterization, antioxidant and in vitro cytotoxic activities of novel coumarin thiazole derivatives Sreekanth ThotaKavitha NadipellyRajeshwar Yerra Original Research 07 August 2014 Pages: 1162 - 1169
2-Aminobenzimidazole conjugates of NSAIDS: novel compounds with immunomodulatory, anti-inflammatory and antioxidant actions Yogita BansalOm Silakari Original Research 08 August 2014 Pages: 1170 - 1179
Synthesis of triazole- and tetrazole-xyloside analogues as potent hyaluronidase inhibitors Yuki KatoMasayuki NinomiyaMamoru Koketsu Original Research 08 August 2014 Pages: 1180 - 1188
The polyion complex nano-prodrug of doxorubicin (DOX) with poly(lactic acid-co-malic acid)-block-polyethylene glycol: preparation and drug controlled release Yanan ZhangCaihua NiWang Li Original Research 08 August 2014 Pages: 1189 - 1195
Metronidazole derivatives as a new class of antiparasitic agents: synthesis, prediction of biological activity, and molecular properties Dua’ Y. AlawadiHaythem A. SaadehMohammad S. Mubarak Original Research 09 August 2014 Pages: 1196 - 1209
Synthesis of some 3(2H)-pyridazinone and 1(2H)-phthalazinone derivatives incorporating aminothiazole moiety and investigation of their antioxidant, acetylcholinesterase, and butyrylcholinesterase inhibitory activities Cem YamalıH. Ozan GülcanDeniz S. Doğruer Original Research 09 August 2014 Pages: 1210 - 1217
Synthesis of some novel purine derivatives incorporating tetrazole ring and investigation of their antimicrobial activity and DNA interactions Selin Kinali-DemirciÖnder İdilAli Dişli Original Research 10 August 2014 Pages: 1218 - 1225
Design, synthesis, in vitro and in silico anti-cancer activity of 4H-chromenes with C4-active methine groups A. ParthibanM. KumaravelH. Surya Prakash Rao Original Research 12 August 2014 Pages: 1226 - 1240
Effect of information leakage and method of splitting (rational and random) on external predictive ability and behavior of different statistical parameters of QSAR model Vijay H. MasandDevidas T. MahajanAhmed M. Alfeefy Original Research 12 August 2014 Pages: 1241 - 1264
Sodium-glucose-linked transporter 2 inhibitors from Sophora flavescens Jing YangXinzhou YangPing Zhao Original Research 12 August 2014 Pages: 1265 - 1271
Molecular modeling studies on substituted aminopyrimidines derivatives as potential antimalarial compounds Mukesh C. SharmaSmita SharmaK. S. Bhadoriya Original Research 13 August 2014 Pages: 1272 - 1288
Simultaneous determination of seven active ingredients in rat plasma by UPLC-MS/MS and application in pharmacokinetic studies after oral administration of scutellaria-coptis herb couple Le-yue DuJian-ming GuoMin Zhao Original Research 13 August 2014 Pages: 1289 - 1297
Rational design, synthesis and evaluation of novel-substituted 1,2,3-triazolylmethyl carbazoles as potent inhibitors of Mycobacterium tuberculosis Goverdhan SurineniPerumal YogeeswariSrinivas Kantevari Original Research 14 August 2014 Pages: 1298 - 1309
Synthesis crystal structure of 2-methoxybenzoylhydrazones and evaluation of their α-glucosidase and urease inhibition potential Muhammad TahaNor Hadiani IsmailM. Iqbal Choudhary Original Research 14 August 2014 Pages: 1310 - 1324
Erratum to: Synthesis crystal structure of 2-methoxybenzoylhydrazones and evaluation of their α-glucosidase and urease inhibition potential Muhammad TahaNor Hadiani IsmailM. Iqbal Choudhary Erratum 16 September 2014 Pages: 1325 - 1325
Cytotoxic flavone glycosides from Solanum elaeagnifolium Mohamed M. RadwanAhmed BadawySafwat A. Ahmed Original Research 14 August 2014 Pages: 1326 - 1330
Molecular docking and biological evaluation of hydroxy-substituted (Z)-3-benzylideneindolin-2-one chalcones for the lead identification as tyrosinase inhibitors Sharad Kumar SutharVaibhav AggarwalManu Sharma Original Research 15 August 2014 Pages: 1331 - 1341
Synthesis, in vitro anthelmintic, and molecular docking studies of novel 5-nitro benzoxazole derivatives R. V. SatyendraK. A. VishnumurthyA. Shruthi Original Research 17 August 2014 Pages: 1342 - 1350
Syntheses of arylcinnamic acids, using Alum-Cs2CO3 as precursors of new 2-heterostyrylbenzimidazoles and their antimicrobial evaluation T. Ashok KumarP. N. Kishore BabuB. Rama Devi Original Research 17 August 2014 Pages: 1351 - 1364