In silico accounting of novel pyridazine analogues as h-PTP 1B inhibitors: pharmacophore modelling, atom-based 3D QSAR and docking studies Manoj Kumar MahapatraRajnish KumarManoj Kumar Original Research 01 November 2013 Pages: 2701 - 2711
A new trypsin inhibitory phthalic acid ester from Heliotropium strigosum Syed Majid ShahAzhar-ul-Haq Ali ShahUmar Farooq Original Research 01 November 2013 Pages: 2712 - 2714
Synthesis, molecular docking studies, and in vitro screening of barbiturates/thiobarbiturates as antibacterial and cholinesterase inhibitors Saira MumtazRashad HussainA. M. Qureshi Original Research 05 November 2013 Pages: 2715 - 2726
Facile synthesis of novel quinoline derivatives as anticancer agents Sheetal Babu MarganakopRavindra Ramappa KambleGangadhar Yamanappa Meti Original Research 05 November 2013 Pages: 2727 - 2735
Synthesis and antiseizure evaluation of isoindoline-1,3-dione derivatives in mice Alireza AliabadiBabak GholamineTahereh Karimi Original Research 05 November 2013 Pages: 2736 - 2743
Prediction of glucagon receptor antagonist activities of some substituted imidazoles using combined radial basis function neural network and density functional theory Mohsen ShahlaeiZohreh Nazari Original Research 06 November 2013 Pages: 2744 - 2756
Predictive 3D-QSAR and HQSAR model generation of isocitrate lyase (ICL) inhibitors by various alignment methods combined with docking study Nirzari GuptaVivek K. VyasManjunath Ghate Original Research 06 November 2013 Pages: 2757 - 2768
In vitro cytotoxicity, α-glucosidase inhibition, antioxidant, and free radical scavenging activities of Illicium griffithii Hook. f. & Thoms fruits A. VijayakumarB. JeyarajS. Ignacimuthu Original Research 07 November 2013 Pages: 2769 - 2779
Synthesis, anti-inflammatory evaluation, and docking studies of some new thiazole derivatives Pran Kishore DebRajwinder KaurRaghuprasad Mailavaram Original Research 09 November 2013 Pages: 2780 - 2792
Synthesis, anti-inflammatory and analgesic activities of arylidene-2-(3-chloroanilino)nicotinic acid hydrazides Latifeh NavidpourHamed ShafaroodiAbbas Shafiee Original Research 12 November 2013 Pages: 2793 - 2802
Identification of neuraminidase inhibitors by structure-based screening: promising new leads for influenza Soumendranath BhakatFaraz ShaikhRakesh M. Rawal Original Research 12 November 2013 Pages: 2803 - 2809
Synthesis and anticonvulsant evaluation of some new 1,3,4,5-tetrahydro-6-alkoxy-2H-1-benzazepin-2-one derivatives Rong-Bi HanYun-Peng ShaoFeng-Yu Piao Original Research 12 November 2013 Pages: 2810 - 2820
Pancreatic α-amylase inhibition and free radical scavenging activity of substituted pyranochromenone derivatives J. Ashok KumarAshok K. TiwariB. China Raju Original Research 13 November 2013 Pages: 2821 - 2833
Type II diabetes-related enzyme inhibition and molecular modeling study of a novel series of pyrazolone derivatives Shobhitha ShettyBalakrishna KallurayaSandeep B. Telkar Original Research 17 November 2013 Pages: 2834 - 2846
Curcumin as inhibitor of mammalian Cathepsin B, Cathepsin H, acid phosphatase and alkaline phosphatase: a correlation with pharmacological activities Indu RavishNeera Raghav Original Research 17 November 2013 Pages: 2847 - 2855
New azetidine-3-carbonyl-N-methyl-hydrazino derivatives of fluoroquinolones: synthesis and evaluation of antibacterial and anticancer properties G. Govinda RajuluHalehatty S. Bhojya NaikKesavan Poonimangadu Koppolu Original Research 17 November 2013 Pages: 2856 - 2868
Studies on the inhibitory models of pyrazoline derivatives as EGFR kinase inhibitors by 3D-QSAR and molecular docking Peizhen LiYueli TianXiaoyun Zhang Original Research 17 November 2013 Pages: 2869 - 2879
Synthesis and in vitro cytotoxicity study of 3-(1H-indol-3-yl)-1,3-diphenylpropan-1-ones Jagadeesh N. MasagalliKittappa M. MahadevanPrashantha Nagaraja Original Research 21 November 2013 Pages: 2880 - 2889
Homology modeling of lanosterol 14α-demethylase of Candida albicans and insights into azole binding Maryam ImanAsghar Davood Original Research 23 November 2013 Pages: 2890 - 2899
Synthesis and antimicrobial screening of some novel chalcones and flavanones substituted with higher alkyl chains Uppuluri Venkata MallavadhaniLaxmidhar SahooUpadyayula Suryanarayana Murty Original Research 24 November 2013 Pages: 2900 - 2908
Synthesis, structure, and in vitro anticancer activity of new polycyclic 1,2-diazines Dorina MantuDan MafteiVasilichia Bejan Original Research 24 November 2013 Pages: 2909 - 2915
Synthesis and antioxidant activity of amido-linked benzoxazolyl/benzothiazolyl/benzimidazolyl-pyrroles and pyrazoles Suram DurgammaAkkarapalli MuralikrishnaAdivireddy Padmaja Original Research 26 November 2013 Pages: 2916 - 2929
Synthesis, molecular docking and antiviral screening of novel N′-substitutedbenzylidene-2-(4-methyl-5,5-dioxido-3-phenylbenzo[e]pyrazolo[4,3-c][1,2]thiazin-1(4H)-yl)acetohydrazides Sana AslamMatloob AhmadRaymond F. Schinazi Original Research 27 November 2013 Pages: 2930 - 2946
Synthesis, characterization, and antibacterial activities of some novel N,N′-disubstituted thiourea, 2-amino thiazole, and imidazole-2-thione derivatives Mehdi KalhorMina SalehifarIraj Nikokar Original Research 27 November 2013 Pages: 2947 - 2954
3D QSAR study of 4H-chromen-1,2,3,4-tetrahydropyrimidine-5-carboxylate derivatives as potential anti-mycobacterial agents Paresh PatelChetan ChinthaVivek K. Vyas Original Research 28 November 2013 Pages: 2955 - 2963
Synthesis of azabicyclo[4.2.0]octa-1,3,5-trien-8-one analogues of 1H-imidazo[4,5-c]quinoline and evaluation of their antimicrobial and anticancer activities Reshma KayarmarG. K. NagarajaT. Arulmoli Original Research 29 November 2013 Pages: 2964 - 2975
Synthesis, characterization of 4,6-disubstituted aminopyrimidines and their sulphonamide derivatives as anti-amoebic agents Shadab Miyan SiddiquiAmir Azam Original Research 30 November 2013 Pages: 2976 - 2984
Vanillin derivatives as the selective small molecule inhibitors of FtsZ Juan SunMing-Hui LiHai-Liang Zhu Original Research 01 December 2013 Pages: 2985 - 2994
Synthesis and biological evaluation of amino acid-linked 1,2,3-bistriazole conjugates as potential antimicrobial agents C. P. KaushikKashmiri LalSunil Kumar Original Research 04 December 2013 Pages: 2995 - 3004
Microwave-assisted synthesis of novel 1,2,3-triazole derivatives and their antimicrobial activity D. AshokD. Mohan GandhiA. Vikas Kumar Original Research 11 December 2013 Pages: 3005 - 3018
New 6-bromoimidazo[1,2-a]pyridine-2-carbohydrazide derivatives: synthesis and anticonvulsant studies Shrikanth UllooraRamakrishna ShabarayaAirody Vasudeva Adhikari Original Research 17 December 2013 Pages: 3019 - 3028
Synthesis and biological evaluation of 1-cyano-2-amino-benzimidazole derivatives as a novel class of antitumor agents Zhang HuLili OuLei Yang Original Research 21 December 2013 Pages: 3029 - 3038
Development of amino acid conjugated sulfonamides as potent antiulcer agent Shakti Prasanna SahooBharat Bhusan Subudhi Original Research 21 December 2013 Pages: 3039 - 3048
Synthesis of 5-arylidine amino-1,3,4-thiadiazol-2-[(N-substituted benzyol)]sulphonamides endowed with potent antioxidants and anticancer activity induces growth inhibition in HEK293, BT474 and NCI-H226 cells Mahavir ChhajedAnil Kumar ShrivastavaVijay Taile Original Research Open access 27 December 2013 Pages: 3049 - 3064
Synthesis, antimicrobial, and antioxidant activity of benzofuran barbitone and benzofuran thiobarbitone derivatives R. KenchappaYadav D. BodkeM. Aruna Sindhe Original Research 27 December 2013 Pages: 3065 - 3081
QSAR study of mGlu5 inhibitors by genetic algorithm-multiple linear regressions Eslam PourbasheerReza AalizadehAlireza Banaei Original Research 27 December 2013 Pages: 3082 - 3091
A comparative molecular dynamics simulation study to assess the exclusion ability of novel GSK3β inhibitors Pradeep HanumanthappaRajanikant G. Krishnamurthy Original Research 28 December 2013 Pages: 3092 - 3095
Structural findings of quinolone carboxylic acids in cytotoxic, antiviral, and anti-HIV-1 integrase activity through validated comparative molecular modeling studies Nilanjan AdhikariAmit Kumar HalderTarun Jha Original Research 29 December 2013 Pages: 3096 - 3127
Microwave-assisted synthesis of some hybrid molecules containing penicillanic acid or cephalosporanic acid moieties and investigation of their biological activities Serap BasogluSerdar UlkerNeslihan Demirbas Original Research Open access 29 December 2013 Pages: 3128 - 3143
Coumarin-containing aminophosphonates bridged with chiral side chain: synthesis and influence of chirality on cytotoxicity and DNA binding Ya-Jun LiMan-Yi YeHeng-Shan Wang Original Research 29 December 2013 Pages: 3144 - 3156
Synthesis, in vitro and in vivo giardicidal activity, and pharmacokinetic profile of a new nitazoxanide analog Adriana Valladares-MéndezEmanuel Hernández-NúñezGabriel Navarrete-Vázquez Original Research 03 January 2014 Pages: 3157 - 3164
Synthesis of progesterone derivatives and evaluation of their efficiency as pneumococcal vaccines Rafat M. MoharebFatma O. Al FaroukKonstantin Karaghiosoff Original Research 03 January 2014 Pages: 3165 - 3177
Synthesis and structure–activity relationship of nuciferine derivatives as potential acetylcholinesterase inhibitors Zhongduo YangZhuwen SongXiaojun Yao Original Research 03 January 2014 Pages: 3178 - 3186
Studies on the synthesis, in vitro antitumor activity of 4H-benzo[h]chromene, 7H-benzo[h]chromene[2,3-d]pyrimidine derivatives and structure–activity relationships of the 2-,3- and 2,3-positions Ahmed M. El-AgrodyAhmed M. FoudaAl-Anood M. Al-Dies Original Research 04 January 2014 Pages: 3187 - 3199
Molecular docking studies on N-hydroxyindole derivatives as potent inhibitors of human lactate dehydrogenase isoform 5 against cancer cell proliferation Manisha Choudhury Original Research 05 January 2014 Pages: 3200 - 3206
Synthesis of 1-benzhydryl piperazine derivatives and evaluation of their ACE inhibition and antimicrobial activities Amlipur SanthoshiSingam Naveen KumarVaidya Jayathirtha Rao Original Research 07 January 2014 Pages: 3207 - 3219
Synthesis, in vitro anticancer activity and in silico study of new disubstituted thiazolidinedione derivatives Moacyr Jesus Barreto de Melo RêgoMarina Rocha Galdino-PittaMaira Galdino da Rocha Pitta Original Research 08 January 2014 Pages: 3220 - 3226
Effect of two series of isoindolines over HDAC8 activity and expression Cynthia R. Trejo MuñozElvia Mera JiménezTeresa Mancilla Percino Original Research 10 January 2014 Pages: 3227 - 3234
Synthesis and pharmacological evaluation of novel thienopyrimidine and triazolothienopyrimidine derivatives Jameel Ahmed S. MullaMohammed Iqbal A. KhaziImtiyaz Ahmed M. Khazi Original Research 12 January 2014 Pages: 3235 - 3243
3D-QSAR study using CoMFA and CoMSIA methods for a series of histone H3 phosphorylation inhibitors Guo-Wu RaoCheng-Hai HuBing-Lan Wang Original Research 04 March 2014 Pages: 3244 - 3254