Synthesis, biological activities, and pharmacokinetics studies of a mutual prodrug of aceclofenac and paracetamol Asif HusainPriyanka AhujaM. S. Zaman Current Trends 24 August 2013 Pages: 1077 - 1083
Synthesis and antioxidant activity of pyrazolyl-oxazolines/thiazolines and isoxazolyl-oxazolines/thiazolines Adivireddy PadmajaChittoor RajasekharVenkatapuram Padmavathi Original Research 24 August 2013 Pages: 1084 - 1098
Antiproliferative effects of novel urea derivatives against human prostate and lung cancer cells; and their inhibition of β-glucuronidase activity Shahnaz PerveenSana MustafaWolfgang Voelter Original Research 27 August 2013 Pages: 1099 - 1113
Prospective atom-based 3D-QSAR model prediction, pharmacophore generation, and molecular docking study of carbamate derivatives as dual inhibitors of AChE and MAO-B for Alzheimer’s disease Vikas KumarNidhi ChadhaAnil K. Mishra Original Research 25 August 2013 Pages: 1114 - 1122
Synthesis, characterization, biological activity, and 3D-QSAR studies on some novel class of pyrrole derivatives as antitubercular agents Shrinivas D. JoshiUttam A. MoreAravind M. Badiger Original Research 25 August 2013 Pages: 1123 - 1147
Quantitative structure–property relationship study on the intercalation of anticancer drugs with ct-DNA Shahin AhmadiMohammad Reza KhazaeiAzize Abdolmaleki Original Research 28 August 2013 Pages: 1148 - 1161
Docking and receptor-based QSAR approaches for modeling of CETP inhibitors M. Asadollahi-Baboli Original Research 27 August 2013 Pages: 1162 - 1169
Oligoamides of 2-amino-5-alkylthiazole 4-carboxylic acids: anti-trypanosomal compounds Stuart LangAbedawn I. KhalafColin J. Suckling Original Research 28 August 2013 Pages: 1170 - 1179
Synthesis of pyranochromene and pyranopyrimidine derivatives from substituted natural coumarin isolated from Ammi majus L. and their biological evaluation N. H. OufY. A. SelimA. S. Badr El-din Original Research 25 August 2013 Pages: 1180 - 1188
Homology modeling, binding site identification, and docking study of human β-arrestin: an adaptor protein involved in apoptosis Chetan ChinthaNirzari GuptaVivek K. Vyas Original Research 28 August 2013 Pages: 1189 - 1201
Biotransformation of artemisinin derivatives by Glycyrrhiza glabra, Lavandula officinalis, and Panax quinquefolium Rashmi GaurSuman PatelRajendra Singh Bhakuni Original Research 24 August 2013 Pages: 1202 - 1206
Regioselective synthesis and antibacterial evaluation of novel bis-pyrimidine derivatives via a three-component reaction Nosrat O. MahmoodiSajede ShojaMehdi Rassa Original Research 28 August 2013 Pages: 1207 - 1213
Synthesis, in vitro antiplasmodial and antiproliferative activities of a series of quinoline–ferrocene hybrids David D. N’DaPeter J. Smith Original Research 28 August 2013 Pages: 1214 - 1224
Cytotoxic activity assessment and c-Src tyrosine kinase docking simulation of thieno[2,3-b] pyridine-based derivatives Ali Reza NikkhooRamin MiriAmir Ahmad Salarian Original Research 29 August 2013 Pages: 1225 - 1233
Rapid in silico selection of an MCHR1 antagonists’ focused library from multi-million compounds’ repositories: biological evaluation Beáta FlachnerTünde TömöriGyörgy Dormán Original Research 30 August 2013 Pages: 1234 - 1247
Novel derivatives of 5-amino-1-cyclopropyl-7-[(3R,5S)3,5-dimethylpiperazine-1-yl]-6,8-difluoro-4-oxo-quinoline-3-carboxylic acid: their synthesis, antimicrobial, antifungal, and urease inhibitory studies M. Saeed ArayneNajma SultanaAjmal Khan Original Research 30 August 2013 Pages: 1248 - 1256
Synthesis and cytotoxic evaluation of novel 2,3-di-O-alkyl derivatives of l-ascorbic acid Santosh R. KoteRatnakar MishraShankar R. Thopate Original Research 30 August 2013 Pages: 1257 - 1266
Synthesis of hydrophobic N-acylated isonicotinic acid hydrazide derivatives as potential enoyl–acyl carrier protein reductase (InhA) inhibitors H. S. Naveen KumarThaigarajan ParumasivamAmirin Sadikun Original Research 30 August 2013 Pages: 1267 - 1277
Synthesis and antiproliferative activities of some pyrazole-sulfonamide derivatives Samet MertAyşe Şahin YağlıoğluRahmi Kasımoğulları Original Research 30 August 2013 Pages: 1278 - 1289
Synthesis and evaluation of novel benzimidazole derivatives as antimicrobial agents Deepkumar JoshiKalpesh Parikh Original Research 30 August 2013 Pages: 1290 - 1299
Comparative molecular docking studies of novel 3, 5-disubstituted thiazolidinedione analogs as HIV-1-RT inhibitors Radhe Shyam BahareSwastika Ganguly Original Research 30 August 2013 Pages: 1300 - 1308
Synthesis of novel pyrazolobenzothiazine 5,5-dioxide derivatives as potent anti-HIV-1 agents Matloob AhmadSana AslamRaymond F. Schinazi Original Research 01 September 2013 Pages: 1309 - 1319
Synthesis of some benzoxazinyl pyrazolone arylidenes as potent antimicrobials and antioxidants George SoniaKnolin K. ThachilRavi Thengungal Kochupappy Original Research 01 September 2013 Pages: 1320 - 1326
Interactions of G-quadruplex DNA binding site with berberine derivatives and construct a structure-based QSAR using docking descriptors Malihe EbrahimiTaghi Khayamian Original Research 01 September 2013 Pages: 1327 - 1339
Synthesis and antitumor activity evaluation of 2-arylisoquinoline-1,3(2H,4H)-diones in vitro and in vivo Bo-Rui KangJuan WangSan-Qi Zhang Original Research 01 September 2013 Pages: 1340 - 1349
Synthesis and in vitro antimicrobial evaluation of novel fluorine-containing 3-benzofuran-2-yl-5-phenyl-4,5-dihydro-1H-pyrazoles and 3-benzofuran-2-yl-5-phenyl-4,5-dihydro-isoxazoles Tejpal Singh ChundawatNutan SharmaSunita Bhagat Original Research 01 September 2013 Pages: 1350 - 1359
New 4-thiazolidinones from 5-ethyl pyridine-2-ethanol: their antibacterial, antifungal, and antitubercular activity Navin B. PatelHemant R. PatelDhanji Rajani Original Research 01 September 2013 Pages: 1360 - 1370
Synthesis and antibacterial evaluation of 3,3′-diindolylmethane derivatives Sutapa RoyRahul GajbhiyeParasuraman Jaisankar Original Research 01 September 2013 Pages: 1371 - 1377
Synthesis and leishmanicidal activity of cinnamic acid esters: structure–activity relationship Elver OteroSara M. RobledoWilson Cardona Original Research 01 September 2013 Pages: 1378 - 1386
Synthesis and biological evaluation of pyrrole-2-carboxamide derivatives: oroidin analogues Balaram S. TakaleNeha V. DesaiVikas N. Telvekar Original Research 01 September 2013 Pages: 1387 - 1396
Exploring QSAR studies on 4-substituted quinazoline derivatives as antimalarial compounds for the development of predictive models Mitali MishraVikash Kumar MishraSushil K. Kashaw Original Research 01 September 2013 Pages: 1397 - 1405
Novel cyclotides from Hedyotis biflora inhibit proliferation and migration of pancreatic cancer cell in vitro and in vivo Xiangmin DingDousheng BaiJianjun Qian Original Research 01 September 2013 Pages: 1406 - 1413
A combined approach based on 3D pharmacophore and docking for identification of new aurora A kinase inhibitors Akshada J. JoshiManoj K. GadhwalUrmila J. Joshi Original Research 01 September 2013 Pages: 1414 - 1436
Synthesis and antitumor activity evaluation of anilinoquinoline derivatives by the effect on the expression of polo-like kinase Huang-Kai PengI-Ling LinShyh-Chyun Yang Original Research 01 September 2013 Pages: 1437 - 1446
2D, 3D-QSAR, and pharmacophore studies on thiazolidine-4-carboxylic acid derivatives as neuraminidase inhibitors in H3N2 influenza virus Neni FrimayantiVannajan Sanghiran LeeNoorsaadah Abd. Rahman Original Research 01 September 2013 Pages: 1447 - 1453
p-Toluenesulfonic acid-catalyzed solvent-free synthesis and biological evaluation of new 1-(4′,6′-dimethylpyrimidin-2′-yl)-5-amino-4H-3-arylpyrazole derivatives Ranjana AggarwalAnshul BansalJitender Sharma Original Research 01 September 2013 Pages: 1454 - 1464
Synthesis, cytotoxic evaluation, and molecular docking study of 4,5-diaryl-thiazole-2-thione analogs of combretastatin A-4 as microtubule-binding agents Marjan SalehiSeyed Nasser OstadMohsen Amini Original Research 01 September 2013 Pages: 1465 - 1473
Synthesis and characterization of novel benzimidazole bearing pyrazoline derivatives as potential antimicrobial agents N. C. DesaiD. D. PandyaPriyanka Desai Original Research 01 September 2013 Pages: 1474 - 1487
Amberlite IRA 402(OH)-mediated synthesis and evaluation of fused tricyclic quinolinium salts as potent non-detergent type microbicidal spermicides Maitreyee BanerjeeShrabanti KumarNirup B. Mondal Original Research 01 September 2013 Pages: 1488 - 1500
Design, synthesis, and antiviral activity of new 1H-1,2,3-triazole nucleoside ribavirin analogs Maria de Lourdes G. FerreiraLuiz C. S. PinheiroNúbia Boechat Original Research 01 September 2013 Pages: 1501 - 1511
Hologram quantative structure–activity relationship studies on 1-(5-carboxyindol-1-yl)propan-2-one inhibitors of human cytosolic phospholipase A2α Xiang-Lin YangYuan ZhouXin-Ling Liu Original Research 01 September 2013 Pages: 1512 - 1518
Synthesis and structure evaluation of new complex butylarylpiperazin-1-yl derivatives Daniel SzulczykAnna BielenicaMarta Struga Original Research Open access 03 September 2013 Pages: 1519 - 1536
Synthesis, antibacterial screening, and POM analyses of novel bis-isoxazolyl/pyrazolyl-1,3-diols Harjeet JunejaDhanashri PanchbhaiTaibi Ben Hadda Original Research 03 September 2013 Pages: 1537 - 1547
Computer-assisted design of dual-target anti-HIV-1 compounds Maria C. GuimarãesDaniel G. SilvaMatheus P. Freitas Original Research 03 September 2013 Pages: 1548 - 1558
Design, synthesis, and antimicrobial activity of some novel homodrimane sesquiterpenoids with diazine skeleton Kaleria KuchkovaAculina AricuIonel I. Mangalagiu Original Research 04 September 2013 Pages: 1559 - 1568
Eco-friendly synthesis and antimicrobial activities of substituted-5-(1H-indol-3-yl)methylene)-2,2-dimethyl-1,3-dioxane-4,6-dione derivatives G. ThirupathiM. VenkatanarayanaY. Bharathi Kumari Original Research 04 September 2013 Pages: 1569 - 1580
Theoretical studies, synthesis, and biological activity of 1-[(4-methylphenyl)sulfonyl]-5-oxo-2,3,4,5-tetrahydro-1H-1-benzazepine-4-carbonitrile (C9) as a non-peptide antagonist of the arginine vasopressin V1a and V2 receptors M. Citlalli Contreras-RomoJosé Correa-BasurtoAndrés Quintanar-Stephano Original Research 04 September 2013 Pages: 1581 - 1590
Synthesis and pharmacological evaluation of pyrazolopyrimidopyrimidine derivatives: anti-inflammatory agents with gastroprotective effect in rats Amine KarouiFatma AlloucheFakher Chabchoub Original Research Open access 04 September 2013 Pages: 1591 - 1598
Synthesis and cytotoxic activity of novel hybrid compounds between 2-alkylbenzofuran and imidazole Wei-Chao WanWen ChenXiao-Dong Yang Original Research 04 September 2013 Pages: 1599 - 1611
Synthesis, antimicrobial, and cytotoxicity studies of novel sulfur-linked quinoline–coumarin bisheterocycles Nidhin PaulShanmugam Muthusubramanian Original Research 04 September 2013 Pages: 1612 - 1621