QSAR study on hERG inhibitory effect of kappa opioid receptor antagonists by linear and non-linear methods Eslam PourbasheerAbolghasem BeheshtiParviz Norouzi Original Research 18 December 2012 Pages: 4047 - 4058
Synthesis, docking studies and antioxidant activity of some chalcone and aurone derivatives Tamanna NarsinghaniMukesh C. SharmaSakshi Bhargav Original Research 19 December 2012 Pages: 4059 - 4068
Benzothiazole Schiff-bases as potential imaging agents for β-amyloid plaques in Alzheimer’s disease Changsheng GanLin ZhouHaoshu Wang Original Research 20 December 2012 Pages: 4069 - 4074
Synthesis, characterization, solvatochromic properties, and antimicrobial evaluation of 5-acetyl-2-thioxo-dihydro-pyrimidine-4,6-dione-based chalcones Bhaveshkumar D. DhorajiyaBhimji S. BhakharBharatkumar Z. Dholakiya Original Research 20 December 2012 Pages: 4075 - 4086
Design and synthesis of thienopyridines as novel templates for acetylcholinesterase inhibitors Mohga M. BadranMaha Abdel HakeemRania M. Abdel Salam Original Research 20 December 2012 Pages: 4087 - 4095
Synthesis, biological evaluation and QSAR study of a series of substituted quinazolines as antimicrobial agents Vipul M. BuhaDharmaraj N. RanaNisha K. Shah Original Research 21 December 2012 Pages: 4096 - 4109
Synthesis of 2-[4,5-dimethyl-1-(phenylamino)-1H-imidazol-2-ylthio]-N-(thiazole-2-yl)acetamide derivatives and their anticancer activities Murat DuranŞeref Demirayak Original Research 21 December 2012 Pages: 4110 - 4124
Synthesis and potential antibacterial activity of new rhodanine-3-acetic acid derivatives Jing MiaoChang-Ji ZhengHu-Ri Piao Original Research 21 December 2012 Pages: 4125 - 4132
Activity landscape analysis, CoMFA and CoMSIA studies of pyrazole CB1 antagonists Eduardo Hernández-VázquezOscar Méndez-LucioFrancisco Hernández-Luis Original Research 21 December 2012 Pages: 4133 - 4145
Designing, synthesis, and characterization of some novel coumarin derivatives as probable anticancer drugs Darla Mark ManidharRajesh Kumar KesharwaniKrishna Misra Original Research 24 December 2012 Pages: 4146 - 4157
Synthesis and in vitro antiproliferative activity of novel 12(H)-quino[3,4-b][1,4]benzothiazine derivatives Andrzej ZiębaMałgorzata LatochaAleksander Sochanik Original Research Open access 24 December 2012 Pages: 4158 - 4163
Synthesis and biological evaluation of diamide derivatives of (S)-BINOL and biphenyl as potential anti-inflammatory/anti-arthritic agents Raj RajaduraiRamar PadmanabhanSarkkarai Ananthan Original Research 24 December 2012 Pages: 4164 - 4172
Anti-tyrosinase, antioxidant and antimicrobial activities of hydroxycinnamoylamides Lyubomir GeorgievMaya ChochkovaTsenka Milkova Original Research 24 December 2012 Pages: 4173 - 4182
A 4-(o-methoxyphenyl)-2-aminothiazole: an anti-quorum sensing compound P. G. MoreN. N. KaraleR. H. Patil Original Research 15 November 2012 Pages: 4183 - 4191
Three-dimensional quantitative structure–activity relationship CoMFA/CoMSIA on pyrrolidine-based tartrate diamides as TACE inhibitors Prashant R. MurumkarMayank Kumar SharmaKailash G. Bothara Original Research 03 January 2013 Pages: 4192 - 4201
Synthesis, biopharmaceutical characterization, and antimicrobial study of novel azo dyes of 7-hydroxy-4-methylcoumarin Pravin S. JogiJyotsana MeshramTaibi Ben Hadda Original Research 03 January 2013 Pages: 4202 - 4210
Synthesis, cytotoxic evaluation, and in silico studies of substituted N-alkylbromo-benzothiazoles Rupinder Kaur GillGagandeep SinghA. K. Saxena Original Research 03 January 2013 Pages: 4211 - 4222
Synthesis of tetracyclic aza-/oxa-naphthalen-8-ones and their antimicrobial activity Shubhangi S. SomanTirth H. Thaker Original Research 03 January 2013 Pages: 4223 - 4227
Synthesis and antibacterial activities of para-alkoxy phenyl-β-ketoaldehyde derivatives Jinbing LiuFengyan WuLiangzhong Zhao Original Research 03 January 2013 Pages: 4228 - 4238
Synthesis and pharmacological evaluation of some novel 4-isopropyl thiazole-based sulfonyl derivatives as potent antimicrobial and antitubercular agents G. V. Suresh KumarY. Rajendra PrasadS. M. Chandrashekar Original Research 03 January 2013 Pages: 4239 - 4252
Synthesis, molecular docking study, and anticancer activity of triaryl-1,2,4-oxadiazole Parisa MiralinaghiMona SalimiMohsen Amini Original Research 03 January 2013 Pages: 4253 - 4262
Synthesis and evaluation of thioflavin-T analogs as potential imaging agents for amyloid plaques Soon Jae JungYong Dae ParkKook Hyun Yu Original Research 04 January 2013 Pages: 4263 - 4268
Phytochemical, cytotoxic, hepatoprotective and antioxidant properties of Delonix regia leaves extract Samar S. AzabMohamed Abdel-DaimOmayma A. Eldahshan Original Research 04 January 2013 Pages: 4269 - 4277
Synthesis, anti-inflammatory, and cytotoxicity evaluation of 9,10-dihydroanthracene-9,10-α,β-succinimide and bis-succinimide derivatives Surbhi AryaSandeep KumarSham M. Sondhi Original Research 05 January 2013 Pages: 4278 - 4285
Synthesis and antihyperlipidemic activity of novel condensed 2-fluoromethylpyrimidines Muthu K. KathiravanKapil D. MoreManisha S. Phoujdar Original Research 06 January 2013 Pages: 4286 - 4292
Synthesis of B-ring substituted flavones and evaluation of their antitumor and antioxidant activities Akshada J. JoshiManoj K. GadhwalGirjesh Govil Original Research 06 January 2013 Pages: 4293 - 4299
Synthesis and evaluation of antibacterial activity of water-soluble copper, nickel and zinc tetra (n-carbonylacrylic) aminephthalocyanines P. A. PavaskarS. S. PatilA. V. Salker Original Research 06 January 2013 Pages: 4300 - 4307
Chemico-biological investigation of rhizome essential oil of Zingiber moran—native to Northeast India Archana DasNaresh KasojuLatha Rangan Original Research 06 January 2013 Pages: 4308 - 4315
Synthesis of substituted benzo[d]thiazol-2-ylcarbamates as potential anticonvulsants Ashvini NavaleSmita PawarAmol Kale Original Research 06 January 2013 Pages: 4316 - 4321
Pharmacophore model generation for microtubule-stabilizing anti-mitotic agents (MSAAs) against ovarian cancer Asma AbroSaima KulsoomNaveeda Riaz Original Research 06 January 2013 Pages: 4322 - 4330
QSAR studies of novel potent benzamide derivatives as glucokinase activators Nimisha JainAnand B. MundadaAnupam K. Pathak Original Research 08 January 2013 Pages: 4331 - 4337
One pot synthesis of some novel coumarins containing 5-(substituted-2-hydroxybenzoyl) pyridine as a new class of antimicrobial and antituberculosis agents Varun G. BhilaChirag V. PatelDinkar I. Brahmbhatt Original Research 08 January 2013 Pages: 4338 - 4346
Bioactivity guided isolation of antiinflammatory, analgesic, and antipyretic constituents from the leaves of Pedilanthus tithymaloides (L.) Soma GhoshDebprasad ChattopadhyayAmalesh Samanta Original Research 08 January 2013 Pages: 4347 - 4359
Synthesis of fatty acid Schiff base esters as potential antimicrobial and chemotherapeutic agents Y. MohiniR. B. N. PrasadP. Sujitha Original Research 08 January 2013 Pages: 4360 - 4366
Synthesis of novel imidazo[2,1-b][1,3,4]thiadiazoles appended to sydnone as anticancer agents Gireesh TegginamathRavindra R. KambleGangadhar Y. Meti Original Research 09 January 2013 Pages: 4367 - 4375
Pyridine-2,5-dicarboxylate complexes with 2,2′-bipyridine and Co(II), Zn(II), Cu(II): syntheses, characterization, antimicrobial, and cytotoxic effects Alper Tolga ColakFerdag ColakRuhi Uyar Original Research 09 January 2013 Pages: 4376 - 4383
QSAR analysis of some 1-(3,3-diphenylpropyl)-piperidinyl amides and ureas as CCR5 inhibitors using genetic algorithm-least square support vector machine Mohsen ShahlaeiAfshin Fassihi Original Research 10 January 2013 Pages: 4384 - 4400
Ligand-based drug design for human endothelin converting enzyme-1 inhibitors Karunakar TanneeruItishri SahuLalitha Guruprasad Original Research 10 January 2013 Pages: 4401 - 4409
Exploring the crucial structural elements required for tricyclic quinoline analogs as protein kinase CK2 inhibitors by a combined computational analysis Yue ZhouNa ZhangRugang Zhong Original Research 10 January 2013 Pages: 4410 - 4422
Modeling of CCR5 antagonists as anti HIV agents using combined genetic algorithm and adaptive neuro-fuzzy inference system (GA–ANFIS) Mohsen ShahlaeiAlireza Pourhossein Original Research 10 January 2013 Pages: 4423 - 4436
Synthesis, characterization, and SAR studies of new (1H-indol-3-yl)alkyl-3-(1H-indol-3-yl)propanamide derivatives as possible antimicrobial and antitubercular agents Ranjith Pakkath KaruvalamRajeesh PakkathNalilu Suchetha Kumari Original Research 10 January 2013 Pages: 4437 - 4454
Antimicrobial activity of Schiff bases of coumarin-incorporated 1,3,4-oxadiazole derivatives: an in vitro evaluation Mashooq Ahmad BhatMohamed A. Al-OmarNadeem Siddiqui Original Research 10 January 2013 Pages: 4455 - 4458
Synthesis and antimicrobial activity of novel bis-azaphenothiazines Khushbu KushwahaRajeev SakhujaSubhash C. Jain Original Research 10 January 2013 Pages: 4459 - 4467
3D-QSAR and pharmacophore model study on aryl diphenolic azoles as estrogen receptor-β ligands Hua-Jun LuoKun ZouWei-Qiao Deng Original Research 11 January 2013 Pages: 4468 - 4480
Structure–activity relationship investigation of methoxy substitution on anticancer pyrimido[4,5-c]quinolin-1(2H)-ones Kamel MetwallyAshraf KhalilKhalid El Sayed Original Research 12 January 2013 Pages: 4481 - 4491
In vitro antiproliferative activity of 11-aminoalkylamino-substituted 5H-indolo[2,3-b]quinolines; improving activity of neocryptolepines by installation of ester substituent Wen-Jie LuMarta ŚwitalskaTsutomu Inokuchi Original Research 12 January 2013 Pages: 4492 - 4504
Computational studies on structurally diverse dipeptidyl peptidase IV inhibitors: an approach for new antidiabetic drug development Bhumika PatelManjunath Ghate Original Research 12 January 2013 Pages: 4505 - 4521
Synthesis, characterization, and in vitro anti-Mycobacterium tuberculosis activity of terpene Schiff bases Mashooq A. BhatMohamed A. Al-Omar Original Research 12 January 2013 Pages: 4522 - 4528
Molecular modeling of the Candida albicans Vps4 and a virtual screening study for novel inhibitors Hengye ChenHaoyuan YuDong Yang Original Research 12 January 2013 Pages: 4529 - 4536
Simulated screening of flavonoids as probable anti-Helicobacter pylori drug Kashi Prakash-Gupta RajeshHanumanthappa ManjunathaBasavapattana Rudresh Bharath Original Research 13 January 2013 Pages: 4537 - 4546