Pyridazin-3(2H)-ones: the versatile pharmacophore of medicinal significance Ranju BansalSridhar Thota Review Article 09 October 2012 Pages: 2539 - 2552
Synthesis of some new 2,6-disubstituted-3(2H)-pyridazinone derivatives and investigation of their analgesic, anti-inflammatory and antimicrobial activities Didem TiryakiMurat SukurogluM. Fethi Sahin Original Research 29 September 2012 Pages: 2553 - 2560
Enhancement of transfection activity in HEK293 cells by lipoplexes containing cholesteryl nitrogen-pivoted aza-crown ethers Alisha SewbalasRafique Ul IslamMario Ariatti Original Research 30 September 2012 Pages: 2561 - 2569
Comparative molecular similarity indices analysis of some 1-substituted imidazole analogs as Candida albicans P450-demethylase inhibitors Nagaraj SelvarajSwastika Ganguly Original Research 02 October 2012 Pages: 2570 - 2577
Synthesis and biological evaluation of 1-(3-chloro-2-oxo-4-phenylazetidin-1-yl)-3-(2-oxo-2-(10H-phenothiazin-10-yl)ethyl)urea derivatives A. RajasekaranK. Sheeja Devi Original Research 04 October 2012 Pages: 2578 - 2588
Design and synthesis of some thieno[2,3-c]pyridazine derivatives of expected anticancer activity Afaf K. El-AnsaryAliaa M. KamalMokhtar AbdHafiz Al-Ghorafi Original Research 04 October 2012 Pages: 2589 - 2601
Antifungal, mosquito deterrent, and larvicidal activity of N-(benzylidene)-3-cyclohexylpropionic acid hydrazide derivatives Nurhayat TabancaDavid E. WedgeMehlika Dilek Altintop Original Research 06 October 2012 Pages: 2602 - 2609
Novel N-aryl(alkaryl)-2-[(3-R-2-oxo-2H-[1,2,4]triazino[2,3-c]quinazoline-6-yl)thio]acetamides: synthesis, cytotoxicity, anticancer activity, COMPARE analysis and docking Sergey I. KovalenkoInna S. NosulenkoAndrey M. Katsev Original Research 07 October 2012 Pages: 2610 - 2632
Synthesis and structure–activity relationship studies on novel 8-amino-3-[2-(4-fluorophenoxy)ethyl]-1,3-diazaspiro[4.5]decane-2,4-dione derivatives as anticonvulsant agents M. MadaiahM. K. PrashanthB. Veeresh Original Research 09 October 2012 Pages: 2633 - 2644
Shuffling multivariate adaptive regression splines as a predictive method for modeling of novel pyridylmethylthio derivatives as VEGFR2 inhibitors M. Asadollahi-BaboliA. Mani-Varnosfaderani Original Research 09 October 2012 Pages: 2645 - 2653
Synthesis of new 3-aryl-4-(3-aryl-4,5-dihydro-1H-pyrazol-5-yl)-1-phenyl-1H-pyrazole derivatives as potential antimicrobial agents Shridhar MalladiArun M. IsloorHoong Kun Fun Original Research 09 October 2012 Pages: 2654 - 2664
Synthesis of some new glutamine linked 2,3-disubstituted quinazolinone derivatives as potent antimicrobial and antioxidant agents M. K. PrashanthH. D. Revanasiddappa Original Research 09 October 2012 Pages: 2665 - 2676
Investigation of retention behavior of anthraquinoids in RP-HPLC on 17 different C18 stationary phases by means of quantitative structure retention relationships Raouf GhavamiZolykha Rasouli Original Research 10 October 2012 Pages: 2677 - 2691
In silico identification of potential drug targets in Clostridium difficile R20291: modeling and virtual screening analysis of a candidate enzyme MurG Vijayalakshmi EzhilarasanOm Prakash SharmaArchana Pan Original Research 10 October 2012 Pages: 2692 - 2705
Screening of flavonoids for antitubercular activity and their structure–activity relationships Akhilesh K. YadavJayprakash ThakurMadan M. Gupta Original Research 11 October 2012 Pages: 2706 - 2716
Efficient entry to diversely functionalized spirooxindoles from isatin and their biological activity Mazaahir KidwaiArti JainPratibha Mehta Luthra Original Research 12 October 2012 Pages: 2717 - 2723
Synthesis and antitumor screening of new series of pyrimido-[4,5-b]quinolines and [1,2,4]triazolo[2′,3′:3,4]pyrimido[6,5-b]quinolines M. B. El-AshmawyM. A. El-SherbenyN. S. El-Gohary Original Research 17 October 2012 Pages: 2724 - 2736
Antimicrobial activity of thiazolyl benzenesulfonamide-condensed 2,4-thiazolidinediones derivatives Nikhil M. ParekhKrunal V. JuddhawalaBhaskar M. Rawal Original Research 17 October 2012 Pages: 2737 - 2745
Synthesis and anticonvulsant evaluation of 2-(substituted benzylidene/ethylidene)-N-(substituted phenyl)hydrazinecarboxamide analogues Mohamed Jawed AhsanHabibullah KhalilullahJeyabalan Govindasamy Original Research 18 October 2012 Pages: 2746 - 2754
Design, characterization, computational studies, and pharmacological evaluation of substituted-N′-[(1E) substituted-phenylmethylidene]benzohydrazide analogs Suman BalaGoldie UppalD. N. Prasad Original Research 19 October 2012 Pages: 2755 - 2767
Synthesis and theoretic calculations of benzoxazoles and docking studies of their interactions with triosephosphate isomerase César A. Flores SandovalRoberto I. Cuevas HernándezJosé G. Trujillo Ferrara Original Research 20 October 2012 Pages: 2768 - 2777
Quercetin and taxifolin completely break MDM2–p53 association: molecular dynamics simulation study Sharad VermaAmit SinghAbha Mishra Original Research 20 October 2012 Pages: 2778 - 2787
Synthesis and screening of 2-(2-(4-substituted piperazine-1-yl)-5-phenylthiazol-4-yl)-3-aryl quinazolinone derivatives as anticancer agents Ritesh N. SharmaRasik Ravani Original Research 23 October 2012 Pages: 2788 - 2794
Predictive QSAR modeling on tetrahydropyrimidine-2-one derivatives as HIV-1 protease enzyme inhibitors Jimish R. PatelLaxman M. Prajapati Original Research 23 October 2012 Pages: 2795 - 2801
Synthesis antimicrobial and anticancer activity of N′-arylmethylidene-piperazine-1-carbothiohydrazide Umasankar KulandaiveluBoyapati ShireeshaVenkatesan Jayaprakash Original Research 23 October 2012 Pages: 2802 - 2808
The antioxidant effects of the butterfly cluster [(μ-SeCH2)2CH(OH)]Fe2(CO)6 on radical-induced oxidation of DNA Pei-Ze LiZai-Qun Liu Original Research 25 October 2012 Pages: 2809 - 2814
Novel 4(3H)-quinazolinone analogs: synthesis and anticonvulsant activity Adel S. El-AzabSami G. Abdel-HamideHussein I. El-Subbagh Original Research 26 October 2012 Pages: 2815 - 2827
Structure based virtual screening of non-steroidal anti-inflammatory drugs (NSAIDs) against RNA-binding motif 6 (RBM6) involved in human lung cancer Tirumalasetty MunichandrababuBaki Vijaya BhaskarWudayagiri Rajendra Original Research 30 October 2012 Pages: 2828 - 2839
Synthesis and antibacterial activity of some new hydrazones M. RudrapalR. Siva SatyanandamS. Zaheera Original Research 30 October 2012 Pages: 2840 - 2846
Synthesis of licochalcones and inhibition effects on radical-induced oxidation of DNA Jianghua HeJizhen LiZai-Qun Liu Original Research 30 October 2012 Pages: 2847 - 2854
Synthesis and antitumor activity of novel 4-aminoquinoline derivatives Jie RenJuan ZhaoKun Hu Original Research 30 October 2012 Pages: 2855 - 2861
Synthesis, characterization, and antitumor activity of rare earth metal complexes of benzoic acid nitrogen mustard Sufeng ZhouYun FuChangzheng Li Original Research 02 November 2012 Pages: 2862 - 2869
Homology modeling and docking studies of phosphoenolpyruvate carboxykinase in Schistosoma mansoni Ananta SwargiaryAkalesh Kumar VermaKishore Sarma Original Research 02 November 2012 Pages: 2870 - 2878
Synthesis of novel 1,4-naphthoquinone derivatives: antibacterial and antifungal agents Cemil IbisAmac Fatih TuyunVolodymyr Novikov Original Research 02 November 2012 Pages: 2879 - 2888
Prediction of the binding modes between macrolactin N and peptide deformylase from Staphylococcus aureus by molecular docking and molecular dynamics simulations Jian GaoYuanhua ChengMingjuan Ji Original Research 02 November 2012 Pages: 2889 - 2901
Neurological activities of lapachol and its furano derivatives from Kigelia africana Kenneth O. EyongHarquin S. FoyetVeronica Nastasa Original Research 03 November 2012 Pages: 2902 - 2911
Synthesis and in vitro antimicrobial evaluation of novel 2-amino-6-(phenylthio)-4-(2-(phenylthio)quinolin-3-yl)pyridine-3,5-dicarbonitriles Mehul B. KananiManish P. Patel Original Research 03 November 2012 Pages: 2912 - 2920
Synthesis and biological evaluation of some Schiff bases of 4-amino-5-(4-methylsulfonyl)benzyl-2,4-dihydro-3H-[1,2,4]-triazole-3-thione V. SumangalaBoja PoojaryShalini Shenoy Original Research 03 November 2012 Pages: 2921 - 2928
A possible correlation between antioxidant and antidiabetic potentials of oxovanadium(IV) complexes A. SheelaN. C. SaradaR. Vijayaraghavan Original Research 04 November 2012 Pages: 2929 - 2937
Isolation, characterization, antibacterial, antihelminthic, and in silico studies of polyprenol from Kirganelia reticulata Baill S. D. ShruthiS. Padmalatha RaiY. L. Ramachandra Original Research 04 November 2012 Pages: 2938 - 2945
Antiproliferative activity of pentadeca-(8E, 13Z) dien-11-yn-2-one and (E)-1,8-pentadecadiene from Echinacea pallida (Nutt.) Nutt. roots Ayse Sahin YaglıogluBayram AkdulumSaban Tekin Original Research 04 November 2012 Pages: 2946 - 2953
Microwave-induced CAN promoted atom-economic synthesis of 1H-benzo[b]xanthene and 4H-benzo[g]chromene derivatives of N-allyl quinolone and their antimicrobial activity Hardik H. JardoshManish P. Patel Original Research 04 November 2012 Pages: 2954 - 2963
Synthesis and antimicrobial activities of highly functionalised novel β-lactam and thiazolidine-grafted tetrahydrobenzothiophenes Mariappan BabuKasi PitchumaniPenugonda Ramesh Original Research 07 November 2012 Pages: 2964 - 2974
Design, synthesis and in vitro antimicrobial activity of novel phenylbenzamido-aminothiazole-based azasterol mimics Rama Krishna YadlapalliO. P. ChourasiaRamu Sridhar Perali Original Research 07 November 2012 Pages: 2975 - 2983
Green approach towards the facile synthesis of dihydropyrano(c)chromene and pyrano[2,3-d]pyrimidine derivatives and their biological evaluation Pradeep K. PaliwalSrinivasa Rao JettiShubha Jain Original Research 09 November 2012 Pages: 2984 - 2990
QSAR and docking studies of novel β-carboline derivatives as anticancer Ravindra Kumar ChourasiyaA. Raghuram RaoRam Kishore Agrawal Original Research 09 November 2012 Pages: 2991 - 3001
A study on the reactions of alkyl 4,6-bis(4-fluorophenyl)-2-oxocyclohex-3-ene-1-carboxylate and in vitro antioxidant activity of derivatives Seranthimata SamshuddinBadiadka NarayanaLeelavathi Narayana Madhu Original Research 09 November 2012 Pages: 3002 - 3011
A 2D image-based method for modeling some c-Src tyrosine kinase inhibitors Mohsen ShahlaeiAlireza Pourhossein Original Research 09 November 2012 Pages: 3012 - 3025
Synthesis and analgesic activity of new heterocyclic compounds derived from monoterpenoids Oksana MikhalchenkoIrina Il’inaNariman Salakhutdinov Original Research 09 November 2012 Pages: 3026 - 3034
Microwave-assisted synthesis of pyrido[1,2-a]benzimidazole derivatives of β-aryloxyquinoline and their antimicrobial and antituberculosis activities Chetan B. SanganiHardik H. JardoshRanjan G. Patel Original Research 09 November 2012 Pages: 3035 - 3047