Synthesis and biological evaluation of naphthalene, furan and pyrrole based chalcones as cytotoxic and antimicrobial agents Abhishek BudhirajaKanika KadianK. L. Dhar Original Research 13 July 2011 Pages: 2133 - 2140
Docking study on trametenolic acid B as a α-glucosidase inhibitor Hua-Jun LuoJun-Zhi WangKun Zou Original Research 13 July 2011 Pages: 2141 - 2144
Synthesis, characterization and pharmacological evaluation of (E)-N′-(substituted-benzylidene)isonicotinohydrazide derivatives as potent anticonvulsant agents Manav MalhotraVikramdeep MongaAakash Deep Original Research 15 July 2011 Pages: 2145 - 2152
Atomic and molecular parameters-based comparative QSAR study on tetrahydroimidazodiazepinone derivatives Ahmad Khalid Raza KhanSunil Kumar MishraMohiuddin Ansari Original Research 15 July 2011 Pages: 2153 - 2161
A comparison of crystallographic and DFT optimized geometries on two taxane diterpenoids and docking studies with phospholipase A2 Umesh YadavaHariom GuptaMihir Roychoudhury Original Research 16 July 2011 Pages: 2162 - 2168
Theoretical studies on benzimidazole derivatives as E. coli biotin carboxylase inhibitors Selvaraman NagamaniKarthikeyan MuthusamyGopinath Krishnasamy Original Research 17 July 2011 Pages: 2169 - 2180
Monitoring of cefpirome–antioxidant interaction studies using RP-HPLC M. NawazM. S. ArayneNajma Sultana Original Research 17 July 2011 Pages: 2181 - 2184
Antitumor activities of some new 1,3,2-oxaza- and 1,3,2-diazaphosphorinanes against K562, MDA-MB-231, and HepG2 cells Khodayar GholivandFatemeh GhazianiSina Sarikhani Original Research 20 July 2011 Pages: 2185 - 2195
Rationalization of physicochemical characters and docking of 3-alkoxy-5-phenoxy-N-thiazolyl benzamide analogs toward glucokinase activator activity Arun K. GuptaNeetu SabarwalYogesh P. Agrawal Original Research 19 July 2011 Pages: 2196 - 2207
Synthesis, characterization, and pharmacological evaluation of new GABA analogs as potent anticonvulsant agents Naveen YadavManav MalhotraAakash Deep Original Research 19 July 2011 Pages: 2208 - 2216
Antifungal activity of a novel quercetin derivative bearing a trifluoromethyl group on Candida albicans Tomas C. TempestiM. Gabriela AlvarezEdgardo N. Durantini Original Research 19 July 2011 Pages: 2217 - 2222
Synthesis and biological evaluation of ester derivatives of indomethacin as selective COX-2 inhibitors M. Arockia BabuRakesh ShuklaS. G. Kaskhedikar Original Research 16 July 2011 Pages: 2223 - 2228
Homology modeling and docking study of recent SHV type β-lactamses with traditional and novel inhibitors: an in silico approach to combat problem of multiple drug resistance in various infections Mohd Hassan BaigShazi ShakilAsad U. Khan Original Research 22 July 2011 Pages: 2229 - 2237
Hypoglycemic and insulin mimetic impact of catechin isolated from Cassia fistula: a substantiate in silico approach through docking analysis Daisy PitchaiRajalakshmi Manikkam Original Research 22 July 2011 Pages: 2238 - 2250
Synthesis and biological evaluation of some N4-substituted 5-nitroisatin-3-thiosemicarbazones Humayun PervezNazia ManzoorKhalid M. Khan Original Research 22 July 2011 Pages: 2251 - 2262
Quantitative structure-activity relationship study and directed synthesis of Thieno[2,3-d]pyrimidine-2,4-diones as monocarboxylate transporter 1 inhibitors O. T. DevinyakMikh. V. SlivkaV. G. Lendel Original Research 23 July 2011 Pages: 2263 - 2272
4-Aminoantipyrine-based Schiff-base transition metal complexes as potent anticonvulsant agents Gurunath S. KurdekarM. P. SathishaD. K. Suresh Original Research 24 July 2011 Pages: 2273 - 2279
Compounds against inflammation and oxidative insult as potential agents for neurodegenerative disorders Christos M. DoulgkerisIoanna C. SiskouEleni A. Rekka Original Research 28 July 2011 Pages: 2280 - 2291
Synthesis and biological evaluation of novel series of chalcone derivatives as inhibitors of cyclooxygenase and LPS-induced TNF-α with potent antioxidant properties Babasaheb P. BandgarBaliram S. HoteRajesh N. Gacche Original Research 28 July 2011 Pages: 2292 - 2299
Synthesis and evaluation of substituted 5-(3-chloro-2-oxo-4-phenylazetidin-1-ylamino)pyrimidine-2,4,6(1H,3H,5H)-triones against pentylenetetrazole-induced convulsant in mice Karan Deep Singh PuriShailja SoodArunachalam Muthuraman Original Research 29 July 2011 Pages: 2300 - 2306
Ligand-based drug design studies using predictive pharmacophore model generation on 4H-1,2,4-triazoles as AT1 receptor antagonists Sarvesh PaliwalMahima PalRakesh Yadav Original Research 31 July 2011 Pages: 2307 - 2315
Detection of trastuzumab efficacy using 1H MRI ex vivo of breast cancer cells Dorota BartusikBoguslaw Tomanek Original Research 02 August 2011 Pages: 2316 - 2319
Antimicrobial screening of novel synthesized benzimidazole nucleus containing 4-oxo-thiazolidine derivatives N. C. DesaiAmit M. DodiyaAtul H. Makwana Original Research 03 August 2011 Pages: 2320 - 2328
In silico studies on 2,3-dihydro-1,5-benzothiazepines as cholinesterase inhibitors Farzana Latif AnsariSaima KalsoomFarukh Jabeen Original Research 03 August 2011 Pages: 2329 - 2339
Antioxidant and antimicrobial studies of novel N′-(substituted-2-chloroquinolin-3-yl)methylidene-4-hydroxy-2H-1,2-benzothiazine-3-carbohydrazides 1,1-dioxides Matloob AhmadSyed Umar Farooq RizviRuqia Suliman Original Research 03 August 2011 Pages: 2340 - 2348
Synthesis and antitumor evaluation of some novel pyrrolizine derivatives Mona M. HannaNagwa M. AbdelgawadAmany B. Mohammed Original Research 03 August 2011 Pages: 2349 - 2362
Hypoglycemic effect of astaxanthin from shrimp waste in alloxan-induced diabetic mice Juan-juan WangZhi-qiang ChenWen-qing Lu Original Research 04 August 2011 Pages: 2363 - 2367
[1,2,4]Triazolo[4,3-a]quinoxaline: synthesis, antiviral, and antimicrobial activities Morkos A. HenenSerry A. A. El BialyHassan M. Eisa Original Research 06 August 2011 Pages: 2368 - 2378
Light-mediated interaction of methotrexate with transition metal Cu(II) Sandesh ChibberIftekhar HassanImrana Naseem Original Research 06 August 2011 Pages: 2379 - 2387
Synthesis and antimycobacterial activities of some new N-acylhydrazone and thiosemicarbazide derivatives of 6-methyl-4,5-dihydropyridazin-3(2H)-one Oya Unsal TanKeriman OzadaliAyla Balkan Original Research 07 August 2011 Pages: 2388 - 2394
Synthesis of some new thiazolopyrane and thiazolopyranopyrimidine derivatives bearing a sulfonamide moiety for evaluation as anticancer and radiosensitizing agents Dalal A. Abou El EllaMostafa M. GhorabAiten M. Soliman Original Research 09 August 2011 Pages: 2395 - 2407
Metabolic effects of benzylidene thiazolidinedione derivatives in high-fat fed mice Tiago Gomes AraújoBruno Melo CarvalhoVera Lúcia de Menezes Lima Original Research 09 August 2011 Pages: 2408 - 2414
Modeling, docking, simulation, and inhibitory activity of the benzimidazole analogue against β-tubulin protein from Brugia malayi for treating lymphatic filariasis Om Prakash SharmaArchana PanPremendu P. Mathur Original Research 10 August 2011 Pages: 2415 - 2427
Design, synthesis, and anticonvulsant evaluation of some novel 1, 3 benzothiazol-2-yl hydrazones/acetohydrazones Praveen KumarBirendra ShrivastavaJames P. Stables Original Research 10 August 2011 Pages: 2428 - 2442
Simultaneous determination of glipizide and glimepride by Rp-Hplc in dosage formulations and in human serum Najma SultanaM. Saeed ArayneM. Hashim Zuberi Original Research 11 August 2011 Pages: 2443 - 2448
Antihepatotoxic activity of a sterol glucoside from aerial parts of Clerodendrum phlomidis Amita VermaBahar Ahmed Original Research 11 August 2011 Pages: 2449 - 2453
Molecular simulations of bergenin as a new urease inhibitor Mohammad ArfanHazrat AminMuhammad Azam Khan Original Research 12 August 2011 Pages: 2454 - 2457
A novel and eco-friendly procedure for the synthesis of some pyrazolo-thiadiazolo-pyrimidinones and its in vitro anti-bacterial activity Dhananjaya RanganathAbhishek MazumdarMailavaram Raghu Prasad Original Research 13 August 2011 Pages: 2458 - 2464
Synthesis of pyrazole-based 1,5-diaryl compounds as potent anti-inflammatory agents Priyanka ShrivastavaPraveen SinghAshish Kumar Tewari Original Research 13 August 2011 Pages: 2465 - 2475
Bisabolangelone, a gastric H+/K+-ATPase inhibitor: homology modeling and docking study Hua-Jun LuoJun-Zhi WangKun Zou Original Research 13 August 2011 Pages: 2476 - 2479
Aspartate carbamoyltransferase of Plasmodium falciparum as a potential drug target for designing anti-malarial chemotherapeutic agents Amit Kumar BanerjeeNeelima AroraUpadhyayula Surya Narayana Murty Original Research 17 August 2011 Pages: 2480 - 2493
Synthesis and metal ion binding activity of methyl 12-amino-13-nitro-7-oxo dehydrodeisopropylabietate derivatives Kai WangXianxian LiuYingming Pan Original Research 18 August 2011 Pages: 2494 - 2500
Exploring QSAR of antiamoebic agents of isolated natural products by MLR, ANN, and RTO Guillermo Ramírez-GaliciaHeidy Martínez-PachecoOmar Deeb Original Research 29 September 2011 Pages: 2501 - 2516
The imidazolidone analogs as phospholipase D1 inhibitors: analysis of the three-dimensional quantitative structure–activity relationship Srinivas NakkaLalitha Guruprasad Original Research 18 August 2011 Pages: 2517 - 2525
(Naphthalen-1-yloxy)-acetic acid benzylidene/(1-phenyl-ethylidene)-hydrazide derivatives: synthesis, antimicrobial evaluation, and QSAR studies Rakesh NarangBalasubramanian NarasimhanSunil Sharma Original Research 18 August 2011 Pages: 2526 - 2547
Rapid synthesis, characterization, anticancer and antimicrobial activity studies of substituted thiadiazoles and their dinucleating ligand metal complexes Anjali JhaY. L. N. MurthyG. Durga Original Research 18 August 2011 Pages: 2548 - 2556
Computational approaches to enhance activity of taxanes as antimitotic agent Ponnurengam Malliappan SivakumarNaga VigneshMukesh Doble Original Research 20 August 2011 Pages: 2557 - 2570
Theoretical study on some non-selective beta-adrenergic antagonists and correlation to their biologically active configurations Ahmad Reza BekhradniaMohammad Ali Ebrahimzadeh Original Research 20 August 2011 Pages: 2571 - 2578
A search of novel antimicrobial based on benzimidazole and 2-pyridone heterocycles N. C. DesaiAmit M. DodiyaNiraj R. Shihory Original Research 23 August 2011 Pages: 2579 - 2586
Synthesis and anticonvulsant activity of 8-alkoxy-5,6-dihydro-4H-benzo[f][1,2,4]triazolo[4,3-a]azepine derivatives Wen-Bin ZhangRong-Bi HanFeng-Yu Piao Original Research 27 August 2011 Pages: 2587 - 2594