QSAR analysis of 2-benzoxazolyl hydrazone derivatives for anticancer activity and its possible target prediction N. S. Hari Narayana MoorthyNuno S. CerqueiraPedro A. Fernandes Original Research 02 December 2010 Pages: 133 - 144
QSAR analysis of B-ring-modified diaryl ether derivatives as a InhA inhibitors Abhishek K. JainRavichandran VeerasamyR. K. Agrawal Original Research 03 December 2010 Pages: 145 - 151
Discovery of a novel histone deacetylase 8 inhibitor by virtual screening Lei ZhangMinyong LiWenfang Xu Original Research 03 December 2010 Pages: 152 - 156
Predictions and correlations of structure activity relationship of some aminoantipyrine derivatives on the basis of theoretical and experimental ground Parvez AliJyotsna MeshramTaibi Ben Hadda Original Research 07 December 2010 Pages: 157 - 164
Pharmacophore modeling of some novel indole β-diketo acid and coumarin-based derivatives as HIV integrase inhibitors Shailesh V. JainLalit V. SonawaneSanjaykumar B. Bari Original Research 07 December 2010 Pages: 165 - 173
Synthesis, in vitro cytotoxicity, and anti-microbial studies of 1,4-bis(4-substituted-5-mercapto-1,2,4-triazol-3-yl)butanes Madhusudan PurohitYergeri C. Mayur Original Research 08 December 2010 Pages: 174 - 184
An efficient one-pot cyclization of quinoline thiosemicarbazones to quinolines derivatized with 1,3,4-thiadiazole as anticancer and anti-tubercular agents Sheetal B. MarganakopRavindra R. KambleMahadevappa Y. Kariduraganvar Original Research 08 December 2010 Pages: 185 - 191
Design and synthesis of some thiazolotriazolyl esters as anti-inflammatory and analgesic agents Birsen TozkoparanS. Peri AytaçGöknur Aktay Original Research 12 December 2010 Pages: 192 - 201
3D-QSAR of amino-substituted pyrido[3,2B]pyrazinones as PDE-5 inhibitors Omprakash TanwarRikta SahaMymoona Akhtar Original Research 15 December 2010 Pages: 202 - 211
Synthesis and biological activity studies of new hybrid molecules containing tryptamine moiety Hakan BektasAhmet DemirbasSengul Alpay Karaoglu Original Research 15 December 2010 Pages: 212 - 223
Radiolabeling of EGCG with 131I and biodistribution in rats Feriha ToksozIlknur DemirFatma Yurt Lambrecht Original Research 16 December 2010 Pages: 224 - 228
In vitro evaluation of the antibacterial and antifungal activity of some new pyrazolyl-quinazolin-4(3H)-one derivatives Navin B. PatelJaymin C. PatelGaman G. Barat Original Research 16 December 2010 Pages: 229 - 238
Restoration of p53–DNA interaction loss upon R273H mutation by CP-31398: an ultra accelerated quantum chemical molecular dynamics approach Shah Md. Abdur RaufKamlesh Kumar SahuAkira Miyamoto Original Research 25 December 2010 Pages: 239 - 244
3D-QSAR study of multi-target-directed AchE inhibitors based on autodocking Na ChenChunkai LiuHuabei Zhang Original Research 25 December 2010 Pages: 245 - 256
Synthesis and biological evaluation of a novel class as antileishmanial agent M. N. S. SaudiM. M. A. El-SemaryN. M. Baddour Original Research 25 December 2010 Pages: 257 - 267