Synthesis and evaluation of anti-inflammatory, analgesic, ulcerogenicity and nitric oxide-releasing studies of novel ibuprofen analogs as nonulcerogenic derivatives Aniket P. SarkateDeepak K. LokwaniKailash G. Bothara Original Research 22 July 2010 Pages: 795 - 808
α-Glucosidase inhibitory and antioxidant properties and antidiabetic activity of Hypericum ascyron L. Wen-Yi KangYan-Li SongLi Zhang Original Research 23 July 2010 Pages: 809 - 816
17-Oximino-5-androsten-3β-yl esters: synthesis, antiproliferative activity, acute toxicity, and effect on serum androgen level Neelima DhingraTilak Raj BhardwajManoj Kumar Original Research 04 August 2010 Pages: 817 - 825
Hansch analysis for the prediction of antimycobacterial activity of ofloxacin derivatives Vikramjeet JudgeRakesh NarangPradeep Kumar Original Research 14 August 2010 Pages: 826 - 837
Synthesis and cytotoxicity of novel chrysin derivatives Kun HuWei WangJie Ren Original Research 15 August 2010 Pages: 838 - 846
Synthesis of pregnenolone–danazol–ethylendiamine conjugate: relationship between descriptors log P, π, R m, and V m and its antibacterial activity in S. aureus and V. cholerae L. Figueroa-ValverdeF. Díaz-cedilloElodia García Cervera Original Research 21 August 2010 Pages: 847 - 853
Synthesis and evaluation of in vitro antitubercular activity and antimicrobial activity of some novel 4H-chromeno[2,3-d]pyrimidine via 2-amino-4-phenyl-4H-chromene-3-carbonitriles Nimesh R. KamdarDhaval D. HaveliwalaSaurabh K. Patel Original Research 24 August 2010 Pages: 854 - 864
Synthesis of some substituted furan-2(5H)-ones and derived quinoxalinones as potential anti-microbial and anti-cancer agents Alaa A. El-TombaryYasser S. Abdel-GhanyFarid S. G. Soliman Original Research 28 August 2010 Pages: 865 - 876
QSAR studies of phthalazinones: novel inhibitors of poly (ADP-ribose) polymerase Prarthana V. RewatkarGanesh R. KokilMayuresh K. Raut Original Research 29 August 2010 Pages: 877 - 886
Conventional and microwave-assisted synthesis of imidazole and guanidine derivatives and their biological evaluation Sham M. SondhiJaiveer SinghA. K. Saxena Original Research 02 September 2010 Pages: 887 - 897
Synthesis, antiplatelet aggregation activity, and molecular modeling study of novel substituted-piperazine analogues Khairia M. YoussefMohamed A. Al-OmarAli S. Al-Tuwaijri Original Research 02 September 2010 Pages: 898 - 911
Synthesis, anti-HSV-1, and cytotoxic activities of some new pyrazole- and isoxazole-based heterocycles Kamal M. DawoodHassan Abdel-GawadFarid A. Badria Original Research 04 September 2010 Pages: 912 - 919
Anti-angiogenic/proliferative behavior of a “4-aryl-4H-chromene” on blood vessel’s endothelial cells: A possible evidence on dual “anti-tumor” activity Kamran MansouriReza KhodarahmiHamidreza Mohammadi Motlagh Original Research 11 September 2010 Pages: 920 - 929
Experimental validation and docking studies of flavone derivatives on aldose reductase involved in diabetic retinopathy, neuropathy, and nephropathy Pagadala Nataraj SekharP. B. Kavi KishorG. Gyananath Original Research 16 September 2010 Pages: 930 - 945
Synthesis and analgesic, anti-inflammatory activities of 3-(3-methoxyphenyl)-2-substituted amino-quinazolin-4(3H)-ones V. AlagarsamyM. GopinathV. Raja Solomon Original Research 16 September 2010 Pages: 946 - 954
Docking and QSAR studies of β-phenylethylidenehydrazine derivatives as a Gamma-aminobutyric acid aminotransferase inhibitor Asghar DavoodMaryam Iman Original Research 17 September 2010 Pages: 955 - 961
Synthesis, spectral, and antimicrobial evaluation of some new 8-membered phosphorus heterocyclic compounds Arigala Uma Ravi SankarSanapalli Subba ReddyChamarthi Naga Raju Original Research 17 September 2010 Pages: 962 - 967
Antioxidant activity and inhibition effect on the growth of human colon carcinoma (HT-29) cells of esculetin from Cortex Fraxini Kai WangYe ZhangYingming Pan Original Research 25 September 2010 Pages: 968 - 974
Synthesis and biological activity of novel 1H-1,4-diazepines containing benzene sulfonyl piperazine moiety Shalini SaingarRajesh KumarYogesh Chandra Joshi Original Research 25 September 2010 Pages: 975 - 980
Synthesis, spectral, theoretical, and antimicrobial screening of some heterocyclic oximes Jayaraman JayabharathiAnnamalai ManimekalaiManoharan Padmavathy Original Research 26 September 2010 Pages: 981 - 995
Synthesis and evaluation of 7-substituted-3,4-dihydrobenzo[f][1,4]oxazepin-5(2H)-ones as anticonvulsant and hypnotic agents Xian-Qing DengMing-Xia SongZhe-Shan Quan Original Research 26 September 2010 Pages: 996 - 1004
Ligand-based in silico 3D-QSAR study of PPAR-γ agonists Lalit Vijay SonawaneSanjaykumar Baburao Bari Original Research 29 September 2010 Pages: 1005 - 1014
Design, synthesis and preliminary evaluation of some novel [1,4]diazepino [5,6-b]pyrrolizine and 6-(2-oxopyrrolidino)-1H-pyrrolizine derivatives as anticonvulsant agents Safinaz E. AbbasFadi Mohsen AwadallahBassem A. Shehata Original Research 29 September 2010 Pages: 1015 - 1023
Synthesis, characterization and in vitro cytotoxic properties of some new Schiff and Mannich bases in Hep G2 cells Dhanya SunilArun M. IsloorK. Satyamoorthy Original Research 29 September 2010 Pages: 1024 - 1032
Synthesis and antimicrobial activity of new pyridine derivatives-I Navin B. PatelSuresh N. AgravatFaiyazalam M. Shaikh Original Research 30 September 2010 Pages: 1033 - 1041
EGFR tyrosine kinase targeted compounds: synthesis, docking study, and in vitro antitumor activity of some new quinazoline and benzo[d]isothiazole derivatives Kamelia M. AminHanan H. GeorgeyFadi M. Awadallah Original Research 02 October 2010 Pages: 1042 - 1053
Synthesis and in vitro microbial activities of amides of pyridoquinolone Navin B. PatelSarvil D. PatelHiren I. Chauhan Original Research 02 October 2010 Pages: 1054 - 1067
Synthesis of novel porphyrin-based lipids and their antibacterial activity Amarnath VelidandiKranthi Kumar GadidasuV. Srilakshmi Patri Original Research 06 October 2010 Pages: 1068 - 1073
Synthesis, characterization, antioxidant, and anticancer studies of 6-[3-(4-chlorophenyl)-1H-pyrazol-4-yl]-3-[(2-naphthyloxy)methyl][1,2,4]triazolo[3,4-b][1,3,4]thiadiazole in HepG2 cell lines Dhanya SunilArun M. IsloorA. S. Bharath Prasad Original Research 06 October 2010 Pages: 1074 - 1080
Synthesis and antibacterial evaluation of 6-azapyrimidines with α-methylene-γ-(4-substituted phenyl)-γ-butyrolactone pharmacophores Po-Jui HuangKuan-Han Lee Original Research 06 October 2010 Pages: 1081 - 1090
Synthesis and characterization of some heterocyclic schiff bases: potential anticonvulsant agents Shailendra PandeyR. S. Srivastava Original Research 06 October 2010 Pages: 1091 - 1101
Evaluation of biological activity of new hemiesters of 17-hydroxy-16,17-secoestra-1,3,5(10)-triene-16-nitrile Suzana S. Jovanović-ŠantaSilvana AndrićJulijana A. Petrović Original Research 06 October 2010 Pages: 1102 - 1110
Normalizing effects of Costus speciosus rhizome crude extracts and its fractions on diabetic complications in STZ-induced diabetic rats J. ElizaM. RajalakshmiP. Daisy Original Research 06 October 2010 Pages: 1111 - 1118