CURRENT TRENDS IN DRUG DISCOVERY RESEARCH Stephen J. CutlerAnil Saxena OriginalPaper Pages: 563 - 564
PHENYLPYRUVIC ACID DERIVATIVES AS ENZYME INHIBITORS: THERAPEUTIC POTENTIAL ON MACROPHAGE MIGRATION INHIBITORY FACTOR Alain J.M. CarpyPetrus P. HaasbroeckDouglas W. Oliver OriginalPaper Pages: 565 - 577
ADVANCES IN VIRTUAL HIGH THROUGHPUT SCREENING (v-HTS) Marco PintoreJacques R. Chretien OriginalPaper Pages: 578 - 589
3D QSAR STUDIES OF INHIBITORS OF CHOLESTEROL ESTER TRANSFER PROTEIN (CETP) BY CoMFA, CoMSIA AND GFA METHODOLOGIES Mandar A. KelkarDeepa V. PednekarKrishnacharya G. Akamanchi OriginalPaper Pages: 590 - 604
3D QSAR STUDIES OF INHIBITORS OF EPIDERMAL GROWTH FACTOR RECEPTOR [EGFR] USING CoMFA AND GFA METHODOLOGIES Deepa V. PednekarMandar A. KelkarKrishnacharya G. Akamanchi OriginalPaper Pages: 605 - 618
STUDIES ON NOVEL NON-IMIDAZOLE HUMAN H4 RECEPTOR ANTAGONISTS USING GFA AND FREE-WILSON ANALYSIS Surekha R. PimpleMandar A. KelkarKrishnacharya G. Akamanchi OriginalPaper Pages: 619 - 630
SYNTHESIS, ANOREXIGENIC ACTIVITY AND QSAR OF SUBSTITUTED ARYLOXYPROPANOLAMINES Shipra SrivastavaKalpana BhandariAnil K. Saxena OriginalPaper Pages: 631 - 642
CHEMICAL GENOMICS FOR FASTAND INTEGRATED TARGET IDENTIFICATION AND LEAD OPTIMIZATION Ferenc DarvasGyörgy DormánLászló Ürge OriginalPaper Pages: 643 - 659
A FACILE SYNTHESIS OF 2-BENZYLOXY/2-(4-ISOPROPYLBENZYLOXY)-2-METHYL-3-(4-SUBSTITUTED PHENYL)PROPANOIC ACID BASED INSULIN SNESITIZING AGENTS: RSR13-15 AND PKR13-15 Raman K. VermaRubina SinglaV.T. Punniyakoti OriginalPaper Pages: 660 - 676
CoMFA, ADVANCE CoMFA AND CoMSIA STUDIES ON THE OXADIAZOLE SUBSTITUTED α-ISOPROPOXY PHENYLPROPIONIC ACIDS FOR PPARα AGONISTIC ACTIVITY Gyanendra PandeySushil K. KashawAmil K. Saxena OriginalPaper Pages: 677 - 686
GLUTATHIONE SYNTHESIS IN FILARIAL WORMS: AN ATTRACTIVE TARGET FOR THE DESIGN AND SYNTHESIS OF NEW ANTIFILARIALS Kavita AroraR.C. MishraRolf D. Walter OriginalPaper Pages: 687 - 706
INHIBITORS OF FILARIAL GAMMA-GLUTAMYL CYCLE ENZYMES AS POSSIBLE MACROFILARICIDAL AGENTS Sapna GuptaKavita AroraRolf D. Walter OriginalPaper Pages: 707 - 723
MODULATION OF FILARIAL GLUTATHIONE-S-TRANSFERASE(S) ACTIVITY: A POSSIBILITY TOWARDS THE SYNTHESIS OF NEW CLASSES OF ANTIFILARIAL AGENTS Rumana AhmadR.C. MishraRolf D. Walter OriginalPaper Pages: 724 - 745
CoMFA AND CoMSIA STUDIES ON A SET OF BENZYL PIPERAZINES, PIPERADINES, PYRAZINOPYRIDOINDOLES, PYRAZINOISOQUINOLINES AND SEMI RIGID ANALOGS OF DIPHENHYDRAMINE Stuti GaurPhilip PrathipatiAnil. K. Saxena OriginalPaper Pages: 746 - 757
A CONVENIENT ROUTE FOR THE SYNTHESIS OF CIS-1-SUBSTITUTED 1,2,3,4,4a,5,11,11a-OCTAHYDRO-6H-PYRIDO[3,2-b]CARBAZOLES AND 4-SUBSTITUTED 1,2,3,4,4a,5,6,11c-OCTAHYDRO-7H-PYRIDO[2,3-c] CARBAZOLES AS POTENT DOPAMINE AGONISTS Keshav K. AwasthisRuchika ChakrabartyAnil K. Saxena OriginalPaper Pages: 758 - 769
QSAR AND MOLECULAR MODELING STUDIES IN IMIDAZOPYRIDINETHIAZOLIDINE-2,4-DIONES: PPARγ AGONISTS Amit KapoorSushil K. KashawAnil K. Saxena OriginalPaper Pages: 770 - 780
NEW QUASSINOIDS FROM AILANTHUS EXCELSA Anuj PandeyBipin Chandra JoshiAnakshi Khare OriginalPaper Pages: 781 - 789
PRODUCTION OF ANTIBACTERIAL AND ANTIFUNGAL METABOLITES BY STREPTOMYCES VIOLACEUSNIGER AND MEDIA OPTIMIZATION STUDIES FOR THE MAXIMUM METABOLITE PRODUCTION C.K.M. TripathiVandana PraveenVinod Bihari OriginalPaper Pages: 790 - 799
3D-QSAR STUDIES ON SUBSTITUTED DIHYDROPYRIDINES FOR THEIR α1A-ADRENERGIC RECEPTOR BINDING AFFINITY Neeraj ShakyaZeeshan FatimaAnil K. Saxena OriginalPaper Pages: 812 - 823