1. Novel triazoles of 3-acetylbetulin and betulone as anticancer agents

   • Ewa Bębenek
   • Monika Kadela-Tomanek
   • Stanisław Boryczka

   Review Article Open access 17 July 2018 Pages: 2051 - 2061

   

2. Docking study and antiosteoporosis effects of a dibenzylbutane lignan isolated from Litsea cubeba targeting Cathepsin K and MEK1

   • Wei Peng
   • Hui Shen
   • Ting Han

   Original Research 14 July 2018 Pages: 2062 - 2070

   

3. Synthesis of NSAIDs–Se derivatives as potent anticancer agents

   • lei Liu
   • Shaolei Li
   • Xianran He

   Original Research 12 July 2018 Pages: 2071 - 2078

4. Naturally bioactive compounds from Hemimycale aff arabica: antimicrobial, antiglycation, cytotoxicity, and molecular docking studies

   • Mohamed Shaaban
   • Amal Zaki Hassan
   • Ahmed B. Abdelwahab

   Original Research 17 July 2018 Pages: 2079 - 2088

   

5. Development of 7-methylimidazo[1,5-a]pyrazin-8(7H)-one derivatives as a novel chemical series of BRD4 inhibitors

   • Xueting Liu
   • Zhenwei Wu
   • Jinpei Zhou

   Original Research 19 July 2018 Pages: 2089 - 2099

   

6. Development of hydroxamic acid derivatives as anticancer agent with the application of 3D-QSAR, docking and molecular dynamics simulations studies

   • Preeti Patel
   • Harish Rajak

   Original Research 04 August 2018 Pages: 2100 - 2115

   

7. Cytotoxicities of novel hydrazone compounds with pyrrolidine moiety: inhibition of mitochondrial respiration may be a possible mechanism of action for the cytotoxicity of new hydrazones

   • Kaan Kucukoglu
   • Mustafa Gul
   • Bernard Geny

   Original Research 21 July 2018 Pages: 2116 - 2124

   

8. Thiazoles with cyclopropyl fragment as antifungal, anticonvulsant, and anti-Toxoplasma gondii agents: synthesis, toxicity evaluation, and molecular docking study

   • Krzysztof Z. Łączkowski
   • Natalia Konklewska
   • Agata Paneth

   Original Research Open access 21 July 2018 Pages: 2125 - 2140

   

9. Synthesis and biological evaluation of coumarin clubbed thiazines scaffolds as antimicrobial and antioxidant

   • Nilesh B. Chauhan
   • Navin B. Patel
   • Bhupendra M. Mistry

   Original Research 17 July 2018 Pages: 2141 - 2149

   

10. Evaluation of the effect of 2-(2,4-dihydroxyphenyl)-4H-benzofuro[3,2-d][1,3]thiazin-4-one on colon cells and its anticancer potential

    • Arkadiusz Czerwonka
    • Marta K. Lemieszek
    • Wojciech Rzeski

    Original Research Open access 25 July 2018 Pages: 2150 - 2159

    

11. Revisiting the molecular mechanism of acquired resistance to reversible tyrosine kinase inhibitors caused by EGFR gatekeeper T790M mutation in non-small-cell lung cancer

    • Yan Zhao
    • Yingjie Jiao
    • Xudong Liu

    Original Research 28 July 2018 Pages: 2160 - 2170

    

12. Synthesis, anticonvulsant activity, and molecular modeling studies of novel 1-phenyl/1-(4-chlorophenyl)-2-(1H-triazol-1-yl)ethanol ester derivatives

    • İnci Selin Doğan
    • Zeynep Özdemir
    • Selma Saraç

    Original Research 02 August 2018 Pages: 2171 - 2186

    

13. Isoindolines/isoindoline-1,3-diones as AChE inhibitors against Alzheimer’s disease, evaluated by an improved ultra-micro assay

    • Erik Andrade-Jorge
    • Luis A. Sánchez-Labastida
    • José G. Trujillo-Ferrara

    Original Research 30 July 2018 Pages: 2187 - 2198

    

14. Convenient one-pot synthesis of resin acid Mannich bases as novel anticancer and antifungal agents

    • Elena V. Tret’yakova
    • Gul’sasyak F. Zakirova
    • Lyudmila V. Parfenova

    Original Research 02 August 2018 Pages: 2199 - 2213

    

15. Computational molecular modelling of N-cinnamoyl and hydroxycinnamoyl amides as potential α-glucosidase inhibitors

    • José R. Mora
    • Edgar A. Márquez
    • Luis Calle

    Original Research 06 August 2018 Pages: 2214 - 2223

    

16. In vitro leishmanicidal activity of lactone 1,4-dihydroquinoline derivatives against Leishmania (Leishmania) amazonensis

    • Ana Paula da Rocha Pissurno
    • Fernanda Amorim Santos
    • Rosangela da Silva de Laurentiz

    Original Research 07 August 2018 Pages: 2224 - 2229