1. Preface to this special issue on chemical biology and drug discovery

   • Ho Jeong Kwon

   Preface 26 August 2015 Pages: 1561 - 1562

2. Chemical biology approach for the development of hypoxia inducible factor (HIF) inhibitor LW6 as a potential anticancer agent

   • Ravi Naik
   • Seunghyeon Han
   • Kyeong Lee

   Review 27 August 2015 Pages: 1563 - 1574

   

3. Identification of a thienopyrimidine derivatives target by a kinome and chemical biology approach

   • Chulho Lee
   • Jee Sun Yang
   • Gyoonhee Han

   Review 18 July 2015 Pages: 1575 - 1581

   

4. Organelle-specific Hsp90 inhibitors

   • Young Ho Seo

   Review 22 July 2015 Pages: 1582 - 1590

   

5. Considerations of the chemical biology of microbial natural products provide an effective drug discovery strategy

   • Hyukjae Choi
   • Dong-Chan Oh

   Review 01 August 2015 Pages: 1591 - 1605

   

6. Developing Streptomyces venezuelae as a cell factory for the production of small molecules used in drug discovery

   • Eun Ji Kim
   • Inho Yang
   • Yeo Joon Yoon

   Review 28 July 2015 Pages: 1606 - 1616

   

7. Existing drugs and their application in drug discovery targeting cancer stem cells

   • Junfang Lv
   • Joong Sup Shim

   Review 09 July 2015 Pages: 1617 - 1626

   

8. Target deconvolution of bioactive small molecules: the heart of chemical biology and drug discovery

   • Hye Jin Jung
   • Ho Jeong Kwon

   Review 04 June 2015 Pages: 1627 - 1641

   

9. Application of chemical biology in target identification and drug discovery

   • Yue Zhu
   • Ting Xiao
   • Ming-Wei Wang

   Review 05 August 2015 Pages: 1642 - 1650

   

10. Chemical biology of compounds obtained from screening using disease models

    • Estu Tashiro
    • Masaya Imoto

    Review 17 July 2015 Pages: 1651 - 1660

    

11. Affinity purification in target identification: the specificity challenge

    • Wenlu Zheng
    • Gang Li
    • Xiaoyu Li

    Review 08 August 2015 Pages: 1661 - 1685

    

12. Role of computer-aided drug design in modern drug discovery

    • Stephani Joy Y. Macalino
    • Vijayakumar Gosu
    • Sun Choi

    Review 25 July 2015 Pages: 1686 - 1701

    

13. Next-generation antimicrobials: from chemical biology to first-in-class drugs

    • Michelle Lay Teng Ang
    • Paul Murima
    • Kevin Pethe

    Review Open access 11 August 2015 Pages: 1702 - 1717

14. Drug compound characterization by mass spectrometry imaging in cancer tissue

    • Ho Jeong Kwon
    • Yonghyo Kim
    • György Marko-Varga

    Review 23 July 2015 Pages: 1718 - 1727

    

15. Antiangiogenic activity of herboxidiene via downregulation of vascular endothelial growth factor receptor-2 and hypoxia-inducible factor-1α

    • Hye Jin Jung
    • Yonghyo Kim
    • Ho Jeong Kwon

    Research Article 21 July 2015 Pages: 1728 - 1735