New Insights on Solid-State Changes in the Levothyroxine Sodium Pentahydrate during Dehydration and its Relationship to Chemical Instability Harsh S. ShahKaushalendra ChaturvediKenneth Morris Research Article 02 January 2019 Article: 39
A Novel Simulation-Based Approach for Comparing the Population Against Average Bioequivalence Statistical Test for the Evaluation of Nasal Spray Products on Spray Pattern and Droplet Size Distribution Parameters Jernej GrmašVesna Lužar-StifflerRade Injac Research Article 02 January 2019 Article: 38
A Combined Utilization of Plasdone-S630 and HPMCAS-HF in Ziprasidone Hydrochloride Solid Dispersion by Hot-Melt Extrusion to Enhance the Oral Bioavailability and No Food Effect Xu XueGuoguang ChenLili Ren Research Article 02 January 2019 Article: 37
Mechanical Properties of Topical Anti-Psoriatic Medicines: Implications for Patient Satisfaction with Treatment A. TeixeiraV. VasconcelosI. F. Almeida Research Article 02 January 2019 Article: 36
Development of Valsartan Floating Matrix Tablets Using Low Density Polypropylene Foam Powder: In vitro and In vivo Evaluation Mohamed RahamathullaS. SaisivamH. V. Gangadharappa Research Article 02 January 2019 Article: 35
On the Stability of Nano-formulations Prepared by Direct Synthesis: Simulated Ostwald Ripening of a Typical Nanocrystal Distribution Post-nucleation Peter J. SkrdlaHusheng Yang Brief/Technical Note 02 January 2019 Article: 34
Topical Delivery of Artemisone, Clofazimine and Decoquinate Encapsulated in Vesicles and Their In vitro Efficacy Against Mycobacterium tuberculosis Lindi van ZylJoe M. ViljoenJeanetta du Plessis Research Article 02 January 2019 Article: 33
A Novel Phytantriol-Based Lyotropic Liquid Crystalline Gel for Efficient Ophthalmic Delivery of Pilocarpine Nitrate Xingqi WangYong ZhangXiaoqin Chu Research Article 02 January 2019 Article: 32
Determination of Mycoplasma hyopneumoniae-Specific IgG, IgG1, and IgG2a Titers in BALB/c Mice Induced by Mineral Oil-Based Oil-in-Water Emulsion Adjuvants Prepared Using a Self-Emulsifying Drug Delivery System Rakesh BastolaJo-Eun SeoSangkil Lee Research Article 02 January 2019 Article: 31
5β-Cholanic Acid/Glycol Chitosan Self-Assembled Nanoparticles (5β-CHA/GC-NPs) for Enhancing the Absorption of FDs and Insulin by Rat Intestinal Membranes Chengyun YanJiwei GuYing Liao Research Article 02 January 2019 Article: 30
Systematic Evaluation of a Diclofenac-Loaded Carboxymethyl Cellulose-Based Wound Dressing and Its Release Performance with Changing pH and Temperature Tina MaverLidija GradišnikUroš Maver Research Article 02 January 2019 Article: 29
In Situ Cocrystallization of Dapsone and Caffeine during Fluidized Bed Granulation Processing Valerio TodaroZelalem Ayenew WorkuAnne Marie Healy Research Article 02 January 2019 Article: 28
Influence of Dissolution Vessel Geometry and Dissolution Medium on In Vitro Dissolution Behaviour of Triamterene-Coated Model Stents in Different Test Setups Katharina PruessmannMonika WentzlaffAnne Seidlitz Research Article 02 January 2019 Article: 27
Lipid Nanoemulsions of Rebamipide: Formulation, Characterization, and In Vivo Evaluation of Pharmacokinetic and Pharmacodynamic Effects Arjun NaralaSwathi GudaKishan Veerabrahma Research Article 02 January 2019 Article: 26
Manufacturing of Multi-drug Formulations with Customised Dose by Solvent Impregnation of Mesoporous Silica Tablets Marek ŠoltysSarah AkhlasováFrantišek Štěpánek Research Article 02 January 2019 Article: 25
Predicting the Effects of Different Triazole Antifungal Agents on the Pharmacokinetics of Tamoxifen Lu ChenLiqin ZhuNan Wang Research Article 02 January 2019 Article: 24
Tunable Properties of Poly-DL-Lactide-Monomethoxypolyethylene Glycol Porous Microparticles for Sustained Release of Polyethylenimine-DNA Polyplexes Treniece L. TerryBrittany E. GivensAliasger K. Salem Research Article 02 January 2019 Article: 23
Agranulocytosis-Protective Olanzapine-Loaded Nanostructured Lipid Carriers Engineered for CNS Delivery: Optimization and Hematological Toxicity Studies Dnyandev G. GadhaveAmol A. TagalpallewarChandrakant R. Kokare Research Article 02 January 2019 Article: 22
A Mechanistic Approach To Model the Compression Cycle of Different Toolings Based on Compression Roller Interactions Rohit P. DugarRobert SedlockRutesh H. Dave Research Article 02 January 2019 Article: 21
Cryogenic Fabrication of Dry Powders to Enhance the Solubility of a Promising Anticancer Drug, SHetA2, for Oral Administration Mariam IbrahimManolya Kukut HatipogluLucila Garcia-Contreras Research Article 02 January 2019 Article: 20
Exploring the Nano Spray-Drying Technology as an Innovative Manufacturing Method for Solid Lipid Nanoparticle Dry Powders Krystyna GlaubittMaurizio RicciStefano Giovagnoli Research Article 02 January 2019 Article: 19
Mucoadhesive Polymeric Films to Enhance Barbaloin Penetration Into Buccal Mucosa: a Novel Approach to Chemoprevention Giulia Di PrimaAlice ConigliaroViviana De Caro Research Article 02 January 2019 Article: 18
Surface-Activated Fibre-Like SBA-15 as Drug Carriers for Bone Diseases Magdalena ProkopowiczJacek ŻeglinskiGavin Walker Research Article Open access 20 December 2018 Article: 17
Critical In Vitro Characterization Methods of Lipid-Based Formulations for Oral Delivery: a Comprehensive Review Nitin Kumar SwarnakarNatarajan VenkatesanGuru Betageri Review Article 19 December 2018 Article: 16
Active Targeting of Drugs and Bioactive Molecules via Oral Administration by Ligand-Conjugated Lipidic Nanocarriers: Recent Advances A. B. ShreyaSushil Yadaorao RautSrinivas Mutalik Review Article 18 December 2018 Article: 15
Use of Risk Assessment and Plackett–Burman Design for Developing Resveratrol Spray-Dried Emulsions: a Quality-by-Design Approach Pontip BenjasirimongkolSuchada PiriyaprasarthPornsak Sriamornsak Research Article 18 December 2018 Article: 14
Folic Acid-Functionalized Gold Nanorods for Controlled Paclitaxel Delivery: In Vitro Evaluation and Cell Studies Ligeri PapaioannouAthina AngelopoulouKonstantinos Avgoustakis Research Article 17 December 2018 Article: 13
The Influence of Cellulosic Polymer’s Variables on Dissolution/Solubility of Amorphous Felodipine and Crystallization Inhibition from a Supersaturated State Nian-Qiu ShiYing JinXian-Rong Qi Research Article 17 December 2018 Article: 12
Recent Advances in Formulation Strategies for Efficient Delivery of Vitamin D Rahul GuptaChittaranjan BeheraPrem N. Gupta Review Article 17 December 2018 Article: 11
Solubility Prediction of Drugs in Binary Solvent Mixtures at Various Temperatures Using a Minimum Number of Experimental Data Points Sina DadmandFarzin KamariAbolghasem Jouyban Research Article 17 December 2018 Article: 10
In vitro SPF and Photostability Assays of Emulsion Containing Nanoparticles with Vegetable Extracts Rich in Flavonoids Letícia Caramori CefaliJanaína Artem AtaideEliana Barbosa Souto Research Article 17 December 2018 Article: 9
Solid-State Characterization of Three Polymorphs of an Orally Available Analog of Diethylenetriaminepentaacetic Acid Carla Coste SanchezArjun KalraMichael Jay Research Article 17 December 2018 Article: 8
Novel Dissolution Method for Oral Film Preparations with Modified Release Properties Isabell SpeerMaren PreisJörg Breitkreutz Research Article 17 December 2018 Article: 7
Moisture Monitoring in Fluid-Bed Granulation by Multi-Resonance Microwave Sensor: Applicability on Crystal-Water Containing Donepezil Granules Johanna PetersWolfgang TauteJörg Breitkreutz Research Article 17 December 2018 Article: 6
Brain Microdialysis Study of Vancomycin in the Cerebrospinal Fluid After Intracerebroventricular Administration in Mice Yusuke MiuraYuki FuchigamiShigeru Kawakami Brief/Technical Note 17 December 2018 Article: 5
Stability, Cytotoxicity, and Retinal Pigment Epithelial Cell Binding of Hyaluronic Acid-Coated PLGA Nanoparticles Encapsulating Lutein Chuda ChittasuphoPenpitcha PosritongPakaporn Ariyawong Research Article 17 December 2018 Article: 4
Inhibition of Co-Crystallization of Olmesartan Medoxomil and Hydrochlorothiazide for Enhanced Dissolution Rate in Their Fixed Dose Combination Magdy M. AbdelquaderEbtessam A. EssaGamal M. El Maghraby Research Article 17 December 2018 Article: 3
Raman Spectroscopy for Process Analytical Technologies of Pharmaceutical Secondary Manufacturing Brigitta NagyAttila FarkasGyörgy Marosi Review Article 17 December 2018 Article: 1