Prodrugs of Peptides. 6. Bioreversible Derivatives of Thyrotropin-Releasing Hormone (TRH) with Increased Lipophilicity and Resistance to Cleavage by the TRH-Specific Serum Enzyme Hans BundgaardJudi Møss OriginalPaper Pages: 885 - 892
Diffusion in Porous Materials Above the Percolation Threshold Jayne E. HastedtJames L. Wright OriginalPaper Pages: 893 - 901
Caco-2 Cell Monolayers as a Model for Drug Transport Across the Intestinal Mucosa Allen R. HilgersRobert A. ConradiPhilip S. Burton OriginalPaper Pages: 902 - 910
Determination of Solute–Polymer Interaction Properties and Their Application to Parenteral Product Container Compatibility Evaluations Richard A. KenleyDennis R. Jenke OriginalPaper Pages: 911 - 918
Synthesis and Calcium Channel Antagonist Activity of 3-Arylmethyl 5-Isopropyl l,4-Dihydro-2,6-dimethyl-4-(pyridyl)-3,5-pyridinedicarboxylates Murthy R. AkulaWandikayi C. MatoweEdward E. Knaus OriginalPaper Pages: 919 - 922
Structure Elucidation and Thermospray High-Performance Liquid Chromatography/Mass Spectroscopy (HPLC/MS) of the Microbial and Mammalian Metabolites of the Antimalarial Arteether Charles D. HuffordIk-Soo LeeJohn K. Baker OriginalPaper Pages: 923 - 927
Influence of Average Molecular Weights of Poly(DL-Lactic Acid-Co-Glycolic Acid) Copolymers 50/50 on Phase Separation and in Vitro Drug Release from Microspheres Jean-Marc RuizJean-Pierre BusnelJean-Pierre Benoît OriginalPaper Pages: 928 - 934
Physicochemical Factors Associated with Binding and Retention of Compounds in Ocular Melanin of Rats: Correlations Using Data from Whole-Body Autoradiography and Molecular Modeling for Multiple Linear Regression Analyses Patricia A. ZaneShirley D. BrindleSpencer L. Tripp OriginalPaper Pages: 935 - 941
Melting Point, Boiling Point, and Symmetry Robert AbramowitzSamuel H. Yalkowsky OriginalPaper Pages: 942 - 947
Enhanced Delivery of Zidovudine Through Rat and Human Skin via Ester Prodrugs Toshinobu SekiTakeo KawaguchiKazuhiko Juni OriginalPaper Pages: 948 - 952
Comparison of Single-Dose and Steady-State Nadolol Plasma Concentrations Julie J. KrukemyerHarisios BoudoulasJohn J. Lima OriginalPaper Pages: 953 - 956
Solubilization of Liposomes by Weak Electrolyte Drugs. I. Propranolol James A. RogersGurupadappa V. BetageriYoung W. Choi OriginalPaper Pages: 957 - 961
Particle Size and Content Uniformity Samuel H. YalkowskySanford Bolton OriginalPaper Pages: 962 - 966
Influence of Solute Degradation on the Accumulation of Solutes Migrating into Solution from Polymeric Parenteral Containers Lawrence A. CruzMai P. JenkeDennis R. Jenke OriginalPaper Pages: 967 - 972
In Vitro and in Vivo Testing and Correlation for Oral Controlled/Modified-Release Dosage Forms Jerome P. SkellyGordon L. AmidonAvraham Yacobi Legacy Pages: 975 - 982