Current State and Opportunities with Long-acting Injectables: Industry Perspectives from the Innovation and Quality Consortium “Long-Acting Injectables” Working Group Andrea BauerPhilippe BerbenStephanie E. Barrett Review Article 22 February 2023 Pages: 1601 - 1631
A Perspective on Model-Informed IVIVC for Development of Subcutaneous Injectables Clairissa D. CorpsteinTonglei Li Perspective 31 July 2023 Pages: 1633 - 1639
A Retrospective Analysis of Preclinical and Clinical Pharmacokinetics from Administration of Long-Acting Aqueous Suspensions Ashley R. JohnsonJeanine E. BallardAngela M. Wagner Original Research Article 31 January 2023 Pages: 1641 - 1656
Preclinical Considerations for Long-acting Delivery of Tenofovir Alafenamide from Subdermal Implants for HIV Pre-exposure Prophylaxis Manjula GunawardanaMariana Remedios-ChanMarc M. Baum Original Research Article Open access 23 November 2022 Pages: 1657 - 1672
Development and Evaluation of Dissolving Microarray Patches for Co-administered and Repeated Intradermal Delivery of Long-acting Rilpivirine and Cabotegravir Nanosuspensions for Paediatric HIV Antiretroviral Therapy Kurtis MoffattIsmaiel A. TekkoRyan F. Donnelly Original Research Article Open access 12 October 2022 Pages: 1673 - 1696
Modulating Drug Release from Short Poly(ethylene glycol) Block Initiated Poly(L-lactide) Di-block Copolymers Zein AzhariPatricia SmithRuth E. Cameron Original Research Article Open access 26 April 2022 Pages: 1697 - 1707
Osmolality of Excipients for Parenteral Formulation Measured by Freezing Point Depression and Vapor Pressure – A Comparative Analysis Mariana Hugo SilvaSarah P. HudsonRené Holm Original Research Article 22 April 2022 Pages: 1709 - 1722
Unravelling the Hepatic Elimination Mechanisms of Colistin Bing QiMatthias GijsenPieter Annaert Original Research Article 31 May 2023 Pages: 1723 - 1734
Prediction of Omeprazole Pharmacokinetics and its Inhibition on Gastric Acid Secretion in Humans Using Physiologically Based Pharmacokinetic-Pharmacodynamic Model Characterizing CYP2C19 Polymorphisms Shuai LiLei XieLi Liu Original Research Article 24 May 2023 Pages: 1735 - 1750
Clozapine-loaded nanocapsules improve antipsychotic activity in rats: building a sequential PopPK/PD model to discriminate nanocarriers in the preformulation step Ana Cláudia Funguetto-RibeiroTamara Ramos MacielSandra Elisa Haas Original Research Article 22 June 2023 Pages: 1751 - 1763
Physiologically Based Pharmacokinetic Modeling for Multiple Oral Administration Labetalol in Pregnant Women Yudi SongWei WangDefang Ouyang Original Research Article 04 May 2023 Pages: 1765 - 1775
Population Pharmacokinetic Model of Methotrexate in Brazilian Pediatric Patients with Acute Lymphoblastic Leukemia Pricilla de Oliveira HenzAmanda Valle PinhattiTeresa Dalla Costa Original Research Article 08 June 2023 Pages: 1777 - 1787
In vivo Pharmacokinetics/Pharmacodynamics Profiles for Appropriate Doses of Cefditoren pivoxil against S. pneumoniae in Murine Lung-Infection Model Yuki IgarashiNana KojimaKazuaki Matsumoto Original Research Article 30 May 2023 Pages: 1789 - 1797
Antimicrobial Efficacy Evaluations of Metronidazole against Clostridioides difficile Infection using Fecal Pharmacokinetic and Pharmacodynamic Analyses Sho TashiroKazuaki TaguchiKazuaki Matsumoto Original Research Article 24 May 2023 Pages: 1799 - 1806
Development of a New Method to Evaluate the Biodistribution of Antibodies Using Non-Radioactive Metal Labeling and Inductively Coupled Plasma Mass Spectrometry Miho NagayasuYoko TakanoKazuhisa Ozeki Original Research Article 02 June 2023 Pages: 1807 - 1819
Human Serum Albumin-enriched Clopidogrel Bisulfate Nanoparticle Alleviates Cerebral Ischemia–Reperfusion Injury in Rats Yiting LuoYunli XiaLi Deng Original Research Article 08 June 2023 Pages: 1821 - 1833
Thermoresponsive Gel-loaded Oxcarbazepine Nanosystems for Nose- To-Brain Delivery: Enhanced Antiepileptic Activity in Rats Basant A. Abou-TalebSamar O. El-Ganainy Original Research Article Open access 23 June 2023 Pages: 1835 - 1852
Raman Spectroscopic Analysis of Highly-Concentrated Antibodies under the Acid-Treated Conditions Yusui SatoSatoru NagatoishiKouhei Tsumoto Original Research Article Open access 09 May 2023 Pages: 1853 - 1864
Protein Based Amorphous Solid Dispersion: a Case Study Investigating Different Whey Proteins at High Drug Loading Donglei LengBulut BuldukKorbinian Löbmann Original Research Article 26 May 2023 Pages: 1865 - 1872
N-oxidation Regioselectivity and Risk Prediction Using DFT-ALIE Calculations Gabriel A. Valdivia-BerroetaNina C. Gonnella Original Research Article 29 June 2023 Pages: 1873 - 1883