Scientific Considerations of Pharmaceutical Solid Polymorphism in Abbreviated New Drug Applications Lawrence X. YuM. Scott FurnessAjaz S. Hussain Commentary Pages: 531 - 536
Fluorescent Substrates of Sister-P-Glycoprotein (BSEP) Evaluated as Markers of Active Transport and Inhibition: Evidence for Contingent Unequal Binding Sites Er-jia WangChristopher N. CascianoWilliam W. Johnson OriginalPaper Pages: 537 - 544
16HBE14o- Human Bronchial Epithelial Cell Layers Express P-Glycoprotein, Lung Resistance-Related Protein, and Caveolin-1 Carsten EhrhardtCarsten KneuerClaus-Michael Lehr OriginalPaper Pages: 545 - 551
MDR1 Genotype-Related Duodenal Absorption Rate of Digoxin in Healthy Japanese Subjects Yoshinori MoritaToshiyuki SakaedaKatsuhiko Okumura OriginalPaper Pages: 552 - 556
Induction of Cytochrome P450 2B6 and 3A4 Expression by Phenobarbital and Cyclophosphamide in Cultured Human Liver Slices Hélène MartinJean-Pierre SarsatCarole Lerche-Langrand OriginalPaper Pages: 557 - 568
Mechanistic Studies on Nonviral Gene Delivery to the Intestine Using in Vitro Differentiated Cell Culture Models and an in Vivo Rat Intestinal Loop Sally-Ann CryanCaitriona M. O'Driscoll OriginalPaper Pages: 569 - 575
Vitreous Is a Barrier in Nonviral Gene Transfer by Cationic Lipids and Polymers Leena PitkänenMarika RuponenArto Urtti OriginalPaper Pages: 576 - 583
Influence of Preparation Conditions on Acyclovir-Loaded Poly-d,l-Lactic Acid Nanospheres and Effect of PEG Coating on Ocular Drug Bioavailability Claudia GiannavolaClaudio BucoloMassimo Fresta OriginalPaper Pages: 584 - 590
How Well Can a T-Cell Epitope Replace Its Parent Carrier Protein? A Dose-Response Study James S. CavenaughHsu-Kun WangJames N. Herron OriginalPaper Pages: 591 - 596
Contribution of Ion-Pair Complexation with Bile Salts to the Transport of Organic Cations Across LLC-PK1 Cell Monolayers Im-Sook SongYong-Hae HanChang-Koo Shim OriginalPaper Pages: 597 - 604
Development of a Dog Microdialysis Model for Determining Synovial Fluid Pharmacokinetics of Anti-Arthritis Compounds Exemplified by Methotrexate Mingxin QianWanda WestDavid D. Christ OriginalPaper Pages: 605 - 610
Evaluation of Inhibitory Activity of Casein on Proteases in Rat Intestine Seiji OhtaniKyoko ShirasuToshikiro Kimura OriginalPaper Pages: 611 - 617
Morphine Blood-Brain Barrier Transport Is Influenced by Probenecid Co-Administration Karin TunbladE. Niclas JonssonMargareta Hammarlund-Udenaes OriginalPaper Pages: 618 - 623
Cell Handling, Membrane-Binding Properties and Membrane-Penetration Modeling Approaches of Pivampicillin and Phthalimidomethylampicillin, Two Basic Esters of Ampicillin, in Comparison with Chloroquine and Azithromycin Hugues ChanteuxIsabelle PaternottePaul M. Tulkens OriginalPaper Pages: 624 - 631
Noninvasive Characterization of Regional Variation in Drug Transport into Human Stratum Corneum in Vivo Jui-Chen TsaiChing-Yu LinYing-Hsuan Huang OriginalPaper Pages: 632 - 638
Topical Delivery of 5-Fluorouracil and 6-Mercaptopurine by Their Alkylcarbonyloxymethyl Prodrugs from Water: Vehicle Effects on Design of Prodrugs Kenneth B. SloanScott WasdoRobert Waranis OriginalPaper Pages: 639 - 645
Electroosmotic Pore Transport in Human Skin Olivia D. UittoHenry S. White OriginalPaper Pages: 646 - 652
Pretreatment with a Water-Based Surfactant Formulation Affects Transdermal Iontophoretic Delivery of R-Apomorphine in Vitro Gai Ling LiMeindert DanhofJoke A. Bouwstra OriginalPaper Pages: 653 - 659
Effective Inhibition of Mannitol Crystallization in Frozen Solutions by Sodium Chloride Chitra TelangLian YuRaj Suryanarayanan OriginalPaper Pages: 660 - 667
Stability and Release Performance of a Series of Pegylated Copolymeric Micelles Wen-Jen LinLee-Wei JuangChi-Chang Lin OriginalPaper Pages: 668 - 673
The Stenlying Effect of High Hydrostatic Pressure on Thermally and Hydrolytically Labile Nanosized Carriers Irène BriggerLaurence Armand-LefevrePatrick Couvreur OriginalPaper Pages: 674 - 683
Validation of the Chloramine-T Induced Oxidation of Human Serum Albumin as a Model for Oxidative Damage in Vivo Makoto AnrakuUlrich Kragh-HansenMasaki Otagiri OriginalPaper Pages: 684 - 692
Correlation of rFVIII Inactivation with Aggregation in Solution Wei WangDrew N. Kelner OriginalPaper Pages: 693 - 700
Erratum: A Novel Hepatic-Targeting System for Therapeutic Cytokines That Delivers to the Hepatic Asialoglycoprotein Receptor, But Avoids Receptor-Mediated Endocytosis Pharm. Res. 19:1736-1744 (2002) Erratum Pages: 701 - 701