Synthesis and Pharmacokinetics of a New Liver-Specific Carrier, Glycosylated Carboxymethyl-Dextran, and Its Application to Drug Targeting Makiya NishikawaAkiko KamijoMitsuru Hashida OriginalPaper Pages: 1253 - 1261
The Use of Solution Theories for Predicting Water Vapor Absorption by Amorphous Pharmaceutical Solids: A Test of the Flory–Huggins and Vrentas Models Bruno C. HancockGeorge Zografi OriginalPaper Pages: 1262 - 1267
Peptide Stability in Drug Development. II. Effect of Single Amino Acid Substitution and Glycosylation on Peptide Reactivity in Human Serum Michael F. PowellTracy StewartSonia M. Colon OriginalPaper Pages: 1268 - 1273
Preparation, Characterization, and Pharmaceutical Application of Linear Dextrins. I. Preparation and Characterization of Amylodextrin, Metastable Amylodextrins, and Metastable Amylose Gerrit H. P. Te WierikAnko C. EissensCoenraad F. Lerk OriginalPaper Pages: 1274 - 1279
Preparation, Characterization, and Pharmaceutical Application of Linear Dextrins. II. Complexation and Dispersion of Drugs with Amylodextrin by Freeze-Drying and Kneading Gerrit H. P. Te WierikAnko C. EissensCoenraad F. Lerk OriginalPaper Pages: 1280 - 1284
Evaluation of the Physicochemical Properties and Dissolution Characteristics of Mesalamine: Relevance to Controlled Intestinal Drug Delivery Donna L. FrenchJohn W. Mauger OriginalPaper Pages: 1285 - 1290
In Vivo Skin Penetration of Acitretin in Volunteers Using Three Sampling Techniques Christian SurberKlaus-P. WilhelmHoward I. Maibach OriginalPaper Pages: 1291 - 1294
The Dissolution and Bioavailability of Etodolac from Capsules Exposed to Conditions of High Relative Humidity and Temperatures Mike DeyRobin EneverRichard Weierstall OriginalPaper Pages: 1295 - 1300
Lack of Effect of Ammonium Glycyrrhizinate on the Morphology of Ovine Nasal Mucosa in Vitro Patricia M. ReardonDoris A. WallCaroline H. Gochoco OriginalPaper Pages: 1301 - 1307
Dissolution Modeling: Factors Affecting the Dissolution Rates of Polydisperse Powders Allan T. K. LuMary E. FrisellaKevin C. Johnson OriginalPaper Pages: 1308 - 1314
Convective Solvent Flow Across the Skin During Iontophoresis Aeri KimPhilip G. GreenRichard H. Guy OriginalPaper Pages: 1315 - 1320
A Floating Controlled-Release Drug Delivery System: In Vitro-in Vivo Evaluation Subhash DesaiSanford Bolton OriginalPaper Pages: 1321 - 1325
Topical Penetration of Piroxicam Is Dependent on the Distribution of the Local Cutaneous Vasculature Nancy A. Monteiro-RiviereAlfred O. InmanMichael L. Francoeur OriginalPaper Pages: 1326 - 1331
Rates of Systemic Degradation and Reticuloendothelial System (RES) Uptake of Thermosensitive Liposome Encapsulating Cisplatin in Rats Katsumi IgaYasuaki OgawaHajime Toguchi OriginalPaper Pages: 1332 - 1337
Effect of Age on Distribution of Zidovudine (Azidothymidine) into the Cerebrospinal Fluid of Macaca nemestrina Arturo Lopez-AnayaJashvant D. UnadkatArnold L. Smith OriginalPaper Pages: 1338 - 1340
Effect of Apparent Elimination Half-Life on Nitroglycerin-Induced Hemodynamic Rebound in Experimental Heart Failure John Anthony BauerHo-Leung Fung OriginalPaper Pages: 1341 - 1345
Correlation Between the Plasma Concentration of Mepirodipine and Its Occupancy of Ca2+ Antagonist Receptors in Rats Shizuo YamadaYoumei MatsuokaRyohei Kimura OriginalPaper Pages: 1346 - 1349
Phosphoryloxymethyl Carbamates and Carbonates—Novel Water-Soluble Prodrugs for Amines and Hindered Alcohols Muhammad SafadiReza OliyaiValentino J. Stella OriginalPaper Pages: 1350 - 1355
The Effect of Dihydronicotinate N-Substitution on the Brain-Targeting Efficacy of a Zidovudine Chemical Delivery System Marcus E. BrewsterEmil PopNicholas Bodor OriginalPaper Pages: 1356 - 1362
The Effect of Swelling Characteristics of Superdisintegrants on the Aqueous Coating Solution Penetration into the Tablet Matrix During the Film Coating Process Nazaneen PourkavoosGarnet E. Peck OriginalPaper Pages: 1363 - 1371
Absorption of Recombinant Human Granulocyte Colony-Stimulating Factor (rhG-CSF) from Rat Nasal Mucosa Minoru MachidaKeiko SanoShoji Awazu OriginalPaper Pages: 1372 - 1377
The Influence of Blood Sampling Site in Nasal Drug Delivery Studies in Rats Hing CharSaran KumarCharan R. Behl Note Pages: 1378 - 1380
Single-Puff Particle-Size Analysis of Albuterol Metered-Dose Inhalers (MDIs) by High-Pressure Liquid Chromatography with Electrochemical Detection (HPLC-EC) Moheb M. Nasr Note Pages: 1381 - 1384
Preparation of Small Gelatin and Albumin Microparticles by a Carbon Dioxide Atomization Process Levent ÖnerMichael J. Groves Note Pages: 1385 - 1388
Solid-State Emulsions: The Effects of Maltodextrin on Microcrystalline Aging Scott L. MyersMerrick L. Shively Note Pages: 1389 - 1391