The Effects of Excipients on Freeze-dried Monoclonal Antibody Formulation Degradation and Sub-Visible Particle Formation during Shaking Meng-Jia JinXin-Zhe GeWei-Jie Fang Original Research Article 30 January 2024 Pages: 321 - 334
Coupling Drug Dissolution with BCS Antony SimitopoulosAthanasios TsekourasPanos Macheras Original Research Article Open access 30 January 2024 Pages: 481 - 491
WANTED DEAD OR ALIVE: New Thinking to Incentivize Drug Development Michael S. Kinch Perspective 30 January 2024 Pages: 199 - 202
Keratinocyte Exosomes for Topical Delivery of Tofacitinib in Treatment of Psoriasis: an In Vitro/ In Vivo Study in Animal Model of Psoriasis Pouya DehghaniJaleh VarshosazMahdi Bodaghi Original Research Article Open access 23 January 2024 Pages: 263 - 279
Correction: Comparative Study of Dermal Pharmacokinetics Between Topical Drugs Using Open Flow Microperfusion in a Pig Model Manfred BodenlenzThean YeohThomas Birngruber Correction Open access 19 January 2024 Pages: 409 - 409
Time-Lapse Macro Imaging with Dissolution Tests for Exploring the Interrelationship Between Disintegration and Dissolution Behaviors of Solid Dosages Yichen YangJiajia GengjiLi Deng Original Research Article 19 January 2024 Pages: 387 - 400
Development of an Accelerated Rotator-based Drug Release Method for the Evaluation of Bupivacaine Multivesicular Liposomes Ziyun XiaMinzhi YuAnna Schwendeman Original Research Article 11 January 2024 Pages: 293 - 303
IVIVC Revised Nikolaos AlimpertisAntony SimitopoulosPanos Macheras Original Research Article 08 January 2024 Pages: 235 - 246
The Osmolality and Hemolysis of High-Concentration Monoclonal Antibody Formulations Meng-Juan PangMeng-Wen WangWei-Jie Fang Original Research Article 03 January 2024 Pages: 281 - 291
Correction: Effect of Buffer Salts on Physical Stability of Lyophilized and Spray-Dried Protein Formulations Containing Bovine Serum Albumin and Trehalose Tarun Tejasvi MutukuriJing LingQi Tony Zhou Correction 29 December 2023 Pages: 405 - 406
Comparative Study of Dermal Pharmacokinetics Between Topical Drugs Using Open Flow Microperfusion in a Pig Model Manfred BodenlenzThean YeohThomas Birngruber Original Research Article Open access 29 December 2023 Pages: 223 - 234
Retraction Note: Dual Blockade of PD-1 and LAG3 Immune Checkpoints Increases Dendritic Cell Vaccine Mediated T Cell Responses in Breast Cancer Model Asal BarshidiVahid KarpishehFarhad Jadidi-Niaragh Retraction Note 26 December 2023 Pages: 407 - 408
An In Silico Platform to Predict Cardiotoxicity Risk of Anti-tumor Drug Combination with hiPSC-CMs Based In Vitro Study Lan SangZhengying ZhouKun Hao Original Research Article Open access 26 December 2023 Pages: 247 - 262
Impact of Formulation and Microneedle Length on Transdermal Metronidazole Permeation through Microneedle-Treated Skin Krishna Kumar PatelNicole K. Brogden Original Research Article 22 December 2023 Pages: 355 - 363
Editorial: Improving Product Quality through Process and Materials Understanding Peter L. D. WildfongRahul V. HawareDavid A. Engers Preface 22 December 2023 Pages: 2759 - 2760
Application of PAT Probes in Aluminum Phosphate Adjuvant Manufacturing Przemyslaw KowalGinny FungMarina Kirkitadze Original Research Article 19 December 2023 Pages: 375 - 385
Exploiting Apical Sodium-Dependent Bile Acid Transporter (ASBT)-Mediated Endocytosis with Multi-Functional Deoxycholic Acid Grafted Alginate Amide Nanoparticles as an Oral Insulin Delivery System Maryam RazmjooeiSeyed Mohammad Hashem HosseiniMohammad Hadi Eskandari Original Research Article 19 December 2023 Pages: 335 - 353
PBPK/PD Modeling of Nifedipine for Precision Medicine in Pregnant Women: Enhancing Clinical Decision-Making for Optimal Drug Therapy Xinyang LiuWei WangDefang Ouyang Original Research Article 04 December 2023 Pages: 63 - 75
Impact of Processing Methods on the Physico-chemical Properties of Posaconazole Amorphous Solid Dispersions Ru HeMatthew S. LammYongjun Li Original Research Article 01 December 2023 Pages: 141 - 151
Professor David E. Smith: A Fearless Scientist and Devoted Mentor Brian ThompsonKim BrouwerMaria M. Posada EditorialNotes 29 November 2023 Pages: 2493 - 2497
General Commentary: A Tribute to Professor Kenneth R. Morris – Scientist, Teacher, Mentor, Friend…and Underappreciated Academic Arborist Peter L. D. Wildfong Tribute 28 November 2023 Pages: 2761 - 2767
Comparative Study of Sorption Phenomena Between Three Medications and Syringes Made of Cyclic Olefin Copolymer or Polypropylene Joëlle ClavesPhilip ChennellValérie Sautou Original Research Article 21 November 2023 Pages: 51 - 62
AgNPs-Modified Polylactic Acid Microneedles: Preparation and In Vivo/In Vitro Antimicrobial Studies Wenqin ZhangXiaozhen CaiJianmin Chen Original Research Article 20 November 2023 Pages: 93 - 104
Elucidating the Impact of Material Properties on Tablet Manufacturability for Binary Paracetamol Blends Lena MareczekCarolin RiehlStephan Reichl Original Research Article 17 November 2023 Pages: 185 - 197
Development of Sustained Release System Based on High Water-Absorbable Gel Formation Using Croscarmellose Sodium, Alkaline Excipients and HPMC (ACSH SR System); Novel Application of Croscarmellose Sodium as a Gel Former Masato GomiNaoya MizutaniKazutaka Higaki Original Research Article 14 November 2023 Pages: 3073 - 3086
LC–MS Approach to Decipher a Light Chain Chromatographic Peak Splitting of a Monoclonal Antibody Yanjun LiuZac VanAernumJennifer S. Chadwick Original Research Article 07 November 2023 Pages: 3087 - 3098
Use of Resonant Acoustic Mixing Technology for Ultra-Low-Dose Blending in a Single-Step Mixing Process Kyle A. FreyHelen BakerDavid A. Engers Original Research Article 07 November 2023 Pages: 165 - 183
Fabrication and Characterization of Dissolving Microneedles for Transdermal Drug Delivery of Apomorphine Hydrochloride in Parkinson’s Disease Daisuke AndoAisa OzawaKen-ichi Izutsu Original Research Article 03 November 2023 Pages: 153 - 163
Pharmaceutical and Immunological Evaluation of Cholera Toxin A1 Subunit as an Adjuvant of Hepatitis B Vaccine Microneedles Jong-Chan KimJung-ah ChoiJung-Hwan Park Original Research Article 01 November 2023 Pages: 3059 - 3071
A Stable Irinotecan Liposome with Enhanced Antitumor Activity in a Range of Tumor Models Zhengxing SuLi LiDong Zhao Original Research Article 01 November 2023 Pages: 3043 - 3058
Integrated Exposure–Response of Dupilumab in Children, Adolescents, and Adults With Atopic Dermatitis Using Categorical and Continuous Efficacy Assessments: A Population Analysis Emily BriggsMohamed A. KamalNidal Huniti Original Research Article Open access 11 December 2023 Pages: 2653 - 2666
Benchmark Glycan Profile of Therapeutic Monoclonal Antibodies Produced by Mammalian Cell Expression Systems Shen LuoBaolin Zhang Original Research Article Open access 01 November 2023 Pages: 29 - 37
A survey of FDA Approved Monoclonal Antibodies and Fc-fusion Proteins for Manufacturing Changes and Comparability Assessment Zhe LiXiulian DuYow-Ming C. Wang Original Research Article 01 November 2023 Pages: 13 - 27
Effect of Food Viscosity on Drug Dissolution Rika HiroseKiyohiko Sugano Original Research Article 26 October 2023 Pages: 105 - 112
Validation of Anti-Adeno Associated Virus Serotype rh10 (AAVrh.10) Total and Neutralizing Antibody Immunogenicity Assays Elizabeth Butala-FloresThien NguyenAmanda Hays Original Research Article Open access 25 October 2023 Pages: 2383 - 2397
Examination of the Rate and Extent of Drug Released from Commercial Topical Delivery Systems During Wear: An Example with Lidocaine Topical Systems Qing CaiArmita AzarpanahNicole K. Brogden Original Research Article 17 October 2023 Pages: 39 - 50
Discovery of the Next Generation of Non-peptidomimetic Neurolysin Activators with High Blood-Brain Barrier Permeability: a Pharmacokinetics Study in Healthy and Stroke Animals Yong ZhangSejal SharmaThomas J. Abbruscato Original Research Article 13 October 2023 Pages: 2747 - 2758
Hydration Mechanism and Its Effect on the Solubility of Aripiprazole Zhixin ZhengXin HuangHongxun Hao Original Research Article 13 October 2023 Pages: 113 - 127
Mechanistic Static Model based Prediction of Transporter Substrate Drug-Drug Interactions Utilizing Atorvastatin and Rifampicin Pallabi MitraRumanah KasliwalaMitchell E. Taub Original Research Article 11 October 2023 Pages: 3025 - 3042
Cortisol as Biomarker for CYP17-Inhibition is Associated with Therapy Outcome of Abiraterone Acetate Maaike A. C. BruinMa Ida Mohmaed AliAlwin D. R. Huitema Original Research Article 11 October 2023 Pages: 3001 - 3010
A Minimal PBPK Model for Plasma and Cerebrospinal Fluid Pharmacokinetics of Trastuzumab after Intracerebroventricular Administration in Patients with HER2-Positive Brain Metastatic Localizations Alicja PuszkielGuilhem BousquetXavier Declèves Original Research Article 11 October 2023 Pages: 2687 - 2697
Mitigation of Tribocharging in Pharmaceutical Powders using Surface Modified V-Blenders Tanu MehtaRaj MukherjeeBodhisattwa Chaudhuri Original Research Article 11 October 2023 Pages: 2371 - 2381
Industry Perspective – What does Industry Need to Accelerate Drug Product and Process Development? Bikash ChatterjeeRichard SteinerGoldi Kaul Perspective Open access 11 October 2023 Pages: 7 - 11
Assessing Dose-Exposure–Response Relationships of Miltefosine in Adults and Children using Physiologically-Based Pharmacokinetic Modeling Approach Shadrack J. MaduKe WangMingzhong Li Original Research Article Open access 10 October 2023 Pages: 2983 - 3000
Preclinical Pharmacokinetics and Translational Pharmacokinetic/Pharmacodynamic Modeling of M8891, a Potent and Reversible Inhibitor of Methionine Aminopeptidase 2 Floriane LignetManja Friese-HamimFelix Rohdich Original Research Article Open access 05 October 2023 Pages: 3011 - 3023
Application of NMR and Chemometric Analyses to Better Understand the Quality Attributes in pH and Thermally Degraded Monoclonal Antibodies Victor A. BeaumontLucy LiuHai-Young Kim Original Research Article Open access 05 October 2023 Pages: 2457 - 2467
Development and Validation of Discriminatory In-vitro Release Method for Intramammary Drug Product Nada A. HelalMarilyn N. MartinezMohammad T. H. Nutan Original Research Article 03 October 2023 Pages: 129 - 139
Physiological Dynamics in the Upper Gastrointestinal Tract and the Development of Gastrointestinal Absorption Models for the Immediate-Release Oral Dosage Forms in Healthy Adult Human Kai WangGordon L. AmidonDavid E. Smith Review Article 03 October 2023 Pages: 2607 - 2626
Practical Advice on Scientific Design of Freeze-Drying Process: 2023 Update Serguei TchessalovVito MaglioEvgenyi Shalaev Original Research Article Open access 02 October 2023 Pages: 2433 - 2455