Volume 16, Issue 1

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February 2012

Special issue : Dedicated to Prof. Árpád Furka on his 80th birthday

Issue Editor:

György Dormán

20 articles in this issue

Combinatorial chemistry has matured in the last three decades: dedicated to Professor Árpád Furka on the occasion of his 80th birthday
Gábor Dibó
Full-Length Paper 06 January 2012 Pages: 1 - 3
Parallel microwave chemistry in silicon carbide microtiter platforms: a review
C. Oliver Kappe
Markus Damm
Short Review 30 November 2011 Pages: 5 - 25
The generation of purinome-targeted libraries as a means to diversify ATP-mimetic chemical classes for lead finding
Eduard R. Felder
Alessandra Badari
Barbara Salom
Full-Length Paper 15 February 2012 Pages: 27 - 51
Ultrasound-assisted click chemistry in continuous flow
Noah P. Tu
Jill E. Hochlowski
Stevan W. Djuric
Short Communication 17 September 2011 Pages: 53 - 58
Combining 2D and 3D in silico methods for rapid selection of potential PDE5 inhibitors from multimillion compounds’ repositories: biological evaluation
Tünde Tömöri
István Hajdú
György Dormán
Full-Length Paper 27 September 2011 Pages: 59 - 72
Facile, novel two-step syntheses of benzimidazoles, bis-benzimidazoles, and bis-benzimidazole-dihydroquinoxalines
Zhigang Xu
Arthur Y. Shaw
Christopher Hulme
Full-Length Papers 12 January 2012 Pages: 73 - 79
Parallel synthesis of 1,2,4-triazole derivatives using microwave and continuous-flow techniques
Tamás Szommer
András Lukács
János Gerencsér
Full-Length Paper 26 January 2012 Pages: 81 - 90
α-Azido ketones. Part 7: synthesis of 1,4-disubstituted triazoles by the “click” reaction of various terminal acetylenes with phenacyl azides or α-azidobenzo(hetera)cyclanones
Krisztina Kónya
Szabolcs Fekete
Tamás Patonay
Full-Length Paper 04 February 2012 Pages: 91 - 102
Effect of core epitope modification on the antibody recognition of a MUC2 mucin peptide
Katalin Uray
Ferenc Hudecz
Full-Length Paper 04 March 2012 Pages: 103 - 112
Multicomponent synthesis of acylated short peptoids with antifungal activity against plant pathogens
Matías D. Galetti
Adriana M. Cirigliano
Javier A. Ramírez
Full-Length Paper 16 September 2011 Pages: 113 - 119
Magnetic nanoparticles catalyzed synthesis of diverse N-Heterocycles
Mazaahir Kidwai
Arti Jain
Saurav Bhardwaj
Full-Length Paper 06 November 2011 Pages: 121 - 128
VCl₃ catalyzed imine-based multicomponent reactions for the facile access of functionalized tetrahydropyridines and β-amino carbonyls
Suman Pal
Lokman Hakim Choudhury
Tasneem Parvin
Full-Length Paper 01 November 2011 Pages: 129 - 143
Three-component reactions of isocyanides, dialkyl acetylenedicarboxylates, and trans-cinnamoyl chlorides for the synthesis of highly functionalized 2-vinyl furans
Abbas Ali Esmaeili
Mahdieh Zangouei
Ali Reza Fakhari
Full-Length Paper 16 December 2011 Pages: 145 - 150
Spiro[pyrrolidine-2,3′-oxindole] derivatives synthesized by novel regionselective 1,3-dipolar cycloadditions
Gang Chen
Jing Yang
Xiaojiang Hao
Full-Length Paper 02 December 2011 Pages: 151 - 156
First cascade Mitsunobu reactions for the synthesis of 2-benzoxazole-N-phenyl and 2-benzimidazole-N-phenyl derivatives
Yu Yan
Qifei Zhong
Gang Liu
Full-Length Paper 30 November 2011 Pages: 157 - 162
Synthesis of polyfunctionalized acrylates via one-pot reactions of arylamines, methyl propiolate, aromatic aldehydes, and active methylene compounds
Yan Sun
Jing Sun
Chao-Guo Yan
Full-Length Paper 30 November 2011 Pages: 163 - 171
Synthesis of novel 4H-pyrimido[1,6-a]pyrimidines via a one-pot three-component condensation
Jinbao Xiang
Hanghang Li
Xu Bai
Full-Length Paper 04 December 2011 Pages: 173 - 181
In silico design of multi-target inhibitors for C–C chemokine receptors using substructural descriptors
Alejandro Speck-Planche
Valeria V. Kleandrova
Full-Length Paper 22 October 2011 Pages: 183 - 191
Identification of novel potential HIF-prolyl hydroxylase inhibitors by in silico screening
Mahesh Kumar Teli
G. K. Rajanikant
Full-Length Paper 01 November 2011 Pages: 193 - 202
4D-LQTA-QSAR and docking study on potent gram-negative specific LpxC inhibitors: a comparison to CoMFA modeling
Jahan B. Ghasemi
Reihaneh Safavi-Sohi
Euzébio G. Barbosa
Full-Length Paper 30 November 2011 Pages: 203 - 213

Volume 16, Issue 1

Combinatorial chemistry has matured in the last three decades: dedicated to Professor Árpád Furka on the occasion of his 80th birthday

Parallel microwave chemistry in silicon carbide microtiter platforms: a review

The generation of purinome-targeted libraries as a means to diversify ATP-mimetic chemical classes for lead finding

Ultrasound-assisted click chemistry in continuous flow

Combining 2D and 3D in silico methods for rapid selection of potential PDE5 inhibitors from multimillion compounds’ repositories: biological evaluation

Facile, novel two-step syntheses of benzimidazoles, bis-benzimidazoles, and bis-benzimidazole-dihydroquinoxalines

Parallel synthesis of 1,2,4-triazole derivatives using microwave and continuous-flow techniques

α-Azido ketones. Part 7: synthesis of 1,4-disubstituted triazoles by the “click” reaction of various terminal acetylenes with phenacyl azides or α-azidobenzo(hetera)cyclanones

Effect of core epitope modification on the antibody recognition of a MUC2 mucin peptide

Multicomponent synthesis of acylated short peptoids with antifungal activity against plant pathogens

Magnetic nanoparticles catalyzed synthesis of diverse N-Heterocycles

VCl₃ catalyzed imine-based multicomponent reactions for the facile access of functionalized tetrahydropyridines and β-amino carbonyls

Three-component reactions of isocyanides, dialkyl acetylenedicarboxylates, and trans-cinnamoyl chlorides for the synthesis of highly functionalized 2-vinyl furans

Spiro[pyrrolidine-2,3′-oxindole] derivatives synthesized by novel regionselective 1,3-dipolar cycloadditions

First cascade Mitsunobu reactions for the synthesis of 2-benzoxazole-N-phenyl and 2-benzimidazole-N-phenyl derivatives

Synthesis of polyfunctionalized acrylates via one-pot reactions of arylamines, methyl propiolate, aromatic aldehydes, and active methylene compounds

Synthesis of novel 4H-pyrimido[1,6-a]pyrimidines via a one-pot three-component condensation

In silico design of multi-target inhibitors for C–C chemokine receptors using substructural descriptors

Identification of novel potential HIF-prolyl hydroxylase inhibitors by in silico screening

4D-LQTA-QSAR and docking study on potent gram-negative specific LpxC inhibitors: a comparison to CoMFA modeling

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