Discovery and optimization of pseudopeptide leads towards peptidomimetic drugs Jean-Luc Fauchère Section I. Conformation and Design Pages: 115 - 120
New backbone cyclic substance P analogs Gal BitanStephan BehrensChaim Gilon Section I. Conformation and Design Pages: 121 - 124
Bioactive conformations of peptides and mimetics as milestones in drug design: Investigation of NK1 receptor antagonists Solo GoldsteinMichel NeuwelsJean-Pierre Hénichart Section I. Conformation and Design Pages: 125 - 134
New peptidomimetics in the chemistry of fibrinogen receptor antagonists J. GanteH. JuraszykF. Rippmann Section I. Conformation and Design Pages: 135 - 140
Comparative conformational analysis of two endothelin-B antagonists Solo GoldsteinMichel NeuwelsJean-Pierre Hénichart Section I. Conformation and Design Pages: 141 - 146
Design and synthesis of thrombin inhibitors D. Michael JonesButrus AtrashMichael Szelke Section I. Conformation and Design Pages: 147 - 154
Design of superactive and selective integrin receptor antagonists containing the RGD sequence Horst KesslerBeate DiefenbachJochen Wermuth Section I. Conformation and Design Pages: 155 - 160
New conformationally constrained Xxx-Pro bicyclic mimetics Silvana CappellettiMonica PegnaMassimo Pinori Section I. Conformation and Design Pages: 161 - 164
Somatostatin analogues containing o-aminomethylphenylacetic acid as a bridge unit Valerie BrecxAleksandra MisickaGeorge van Binst Section I. Conformation and Design Pages: 165 - 168
Design of new inhibitors specific to the adenosine triphosphate binding site of DNA topoisomerases II Liliane Assairi Section I. Conformation and Design Pages: 169 - 171
Towards nonpeptide agonists: Design of ‘true’ peptidomimetics Gregory V. Nikiforovich Section I. Conformation and Design Pages: 172 - 176
Benzomorphan alkaloids: Natural peptidomimetics of opioid peptide pharmacophores Andrzej W. LipkowskiAleksandra MisickaVictor J. Hruby Section I. Conformation and Design Pages: 177 - 181
Conformation-directed design of cyclic somatostatins containing a βVI-turn mimetic Dirk Tourwé Section I. Conformation and Design Pages: 182 - 186
The polypeptide 310-helix as a template and a spacer Marco CrismaAlberto BiancoJohan Kamphuis Section I. Conformation and Design Pages: 187 - 189
Synthesis of the diastereomers of β-Me-Tyr and β-Me-Phe and their effect on the biological properties of the delta opioid receptor antagonist TIPP Els MannekensDirk TourwéPeter W. Schiller Section II. Synthesis and Libraries Pages: 190 - 192
Synthesis and activity of phosphono desmuramyldipeptide analogs Uroš UrlebStanislav GobecDušan Prelog Section II. Synthesis and Libraries Pages: 193 - 197
Synthesis and evaluation of azaproline peptides as potential inhibitors of dipeptidyl peptidase IV and prolyl oligopeptidase Marianne BorlooKoen AugustynsAchiel Haemers Section II. Synthesis and Libraries Pages: 198 - 202
Amino acids with amphiphilic side chains: Deltorphin analogues with Phe3 replaced by all β-hydroxyphenylalanine diastereoisomers Aleksandra MisickaAndrzej W. LipkowskiVictor J. Hruby Section II. Synthesis and Libraries Pages: 203 - 205
Amino acids derived from ornithine Theo LescrinierChristophe PannecouquePiet Herdewijn Section II. Synthesis and Libraries Pages: 206 - 208
The effect of dibenzofuran substitutions in corticotropin-releasing factor B. RoloffM. BeyermannM. Bienert Section II. Synthesis and Libraries Pages: 209 - 211
Thiolester substrates of dd-peptidases and β-lactamases Christian DamblonPhilippe LedentJean-Marie Frère Section II. Synthesis and Libraries Pages: 212 - 216
Screening of a synthetic peptide library against glycosomal phosphoglycerate kinase of Trypanosoma brucei Isabelle SamsonArthur van AerschotPiet Herdewijn Section II. Synthesis and Libraries Pages: 217 - 219
Screening of phage-displayed peptide libraries with a monoclonal antibody raised against the F protein of the bovine respiratory syncytial virus Pascal MertensJean-Philippe MatheiseJean-Jacques Letesson Section II. Synthesis and Libraries Pages: 220 - 224
5-Hydroxytryptophan as a building block in oligopeptides using Fmoc/tBu SPPS Theo LescrinierRoger BussonPiet Herdewijn Section II. Synthesis and Libraries Pages: 225 - 228
New methods for solid phase peptide synthesis of transitionstate analog inhibitors of HIV-1 protease and DPP-IV Jan PironDirk Tourwé Section II. Synthesis and Libraries Pages: 229 - 232
Recent advances in phosphono- and phosphinopeptide synthesis Patrick JouinJacques CosteLaurent Guillou Section II. Synthesis and Libraries Pages: 233 - 238
Synthesis and conformational analysis of AzAsx-containing oligopeptides Frédéric AndréGuy BoussardAndré Aubry Section II. Synthesis and Libraries Pages: 239 - 242
A convenient method for the stereoselective preparation of 3-hydroxy-2-substituted propionaldehyde derivatives, C-terminal precursors for the synthesis of trans-alkene dipeptide isosteres Philippe RoureNadia WalchshoferJoëlle Paris Section II. Synthesis and Libraries Pages: 243 - 246
Micro- and macromimetics: Condensation of amino acid derivatives with dienophiles Leonid Yu. SklyarovIrina N. SbitnevaNadezhda A. Kopina Section II. Synthesis and Libraries Pages: 247 - 252
Farmer's peptidomimetic approach: A target for synthetic combinatorial libraries Jung LeeRonald E. BarrettPhilippe R. Bovy Section II. Synthesis and Libraries Pages: 253 - 258
Screening of a synthetic pentapeptide library composed of d-amino acids against fructose-1,6-biphosphate aldolase Isabelle SamsonJef RozenskiPiet Herdewijn Section II. Synthesis and Libraries Pages: 259 - 260
Identification of Brucella cell wall antigenic determinants by immunoscreening of a random peptide library expressed at the surface of filamentous phage Bernadette LichtfousePascal MertensJean-Jacques Letesson Section II. Synthesis and Libraries Pages: 261 - 264
