Pyrazoles, isoxazoles, and 1,2,3-triazoles as analogs of the natural cytostatic combretastatin A-4: efficient routes of synthesis, tubulin inhibition, and cytotoxicity Roman K. KostinAleksander S. Marshavin OriginalPaper 04 January 2022 Pages: 1061 - 1072
Synthesis of 2H-thiochromene derivatives (microreview) Seyed Sajad SajadikhahMahmoud Nassiri OriginalPaper 06 January 2022 Pages: 1073 - 1075
Synthesis of heterocyclic ring-fused quinones (microreview) Anastasija GaileNelli Batenko OriginalPaper 06 January 2022 Pages: 1076 - 1078
Reactivity of alicyclic 1,5,9-triketones toward five-, six-, and seven-membered rings in acidic medium. Stereochemistry of intramolecular cyclization products Taisia I. AkimovaOlga A. SoldatkinaAlevtina A. Kapustina OriginalPaper 04 January 2022 Pages: 1079 - 1085
Aziridine-2-carboxylic acid derivatives and its open-ring isomers as a novel PDIA1 inhibitors Irena LeiteVictor AndrianovIvars Kalvins OriginalPaper 07 January 2022 Pages: 1086 - 1106
[3+2] Cycloaddition reactions of 1-substituted 3,3,3-trifluoropropenes with diazo compounds and nitrilimines – synthesis of pyrazolines and pyrazoles Yuriy N. МаrkitanovVadim М. ТimoshenkoYuriy G. Shermolovich OriginalPaper 06 January 2022 Pages: 1107 - 1115
Synthetic transformations of sesquiterpene lactones. Controllable synthesis of 11,13-dihydroisoalantolactone azides and 13-(1,2,3-triazolyl)eudesmanolides based on sesquiterpene lactones Sergey S. PatrushevTatyana V. RybalovaElvira E. Shults OriginalPaper 06 January 2022 Pages: 1116 - 1129
Lewis acid catalyzed condensation of 2-aminohetarene N-oxides with N,N-dimethylformamide dimethyl acetal Sergey А. KaralashDmitry M. BystrovLeonid L. Fershtat OriginalPaper 04 January 2022 Pages: 1130 - 1136
Synthesis of methyl(ethyl) pyrazolo[4,3-b]pyridine-6-carboxylates and their conversion to tert-butyl 4,5,6,7-tetrahydropyrazolo-[4,3-b]pyridine-6-carboxylates Georgiy G. YakovenkoLesya N. SaliyevaMykhailo V. Vovk OriginalPaper 06 January 2022 Pages: 1137 - 1145
Synthesis and permethylation of methyl 5-(2-chloropyridin-3-yl)pentanoates Franziska BendrathPeter Langer SHORT COMMUNICATION 06 January 2022 Pages: 1146 - 1148