Privileged heterocyclic scaffolds in chemical biology and drug discovery: synthesis and bioactivity News 27 April 2017 Pages: 239 - 239
N-(Hetero)aryl-2-imidazolines: an emerging privileged motif for contemporary drug design Mikhail Krasavin REVIEWS 26 April 2017 Pages: 240 - 255
Preparation and biological properties of 2-thio-containing pyrimidines and their condensed analogs Oleksii Yu. VoskoboynikOleksandra S. KolomoetsSergiy I. Kovalenko OriginalPaper 27 April 2017 Pages: 256 - 272
Heterocycles as classical and nonclassical ring B isosters in combretastatin A-4 Nikolay A. ZefirovOlga N. Zefirova OriginalPaper 24 April 2017 Pages: 273 - 280
1,5-Diarylpyrroles as potent antitubercular and anti-inflammatory agents Giulia VendittiGiovanna PoceMariangela Biava OriginalPaper 27 April 2017 Pages: 281 - 291
2-(Azolyl)anilines: methods of synthesis, cyclocondensations, and biological properties Oleksii M. AntypenkoSergiy V. KholodnyakSergiy I. Kovalenko OriginalPaper 25 April 2017 Pages: 292 - 309
3,4-Dihydroquinoxalin-2-ones: recent advances in synthesis and bioactivities (microreview) Tone KristoffersenJørn H. Hansen HETEROCYCLES IN FOCUS 26 April 2017 Pages: 310 - 312
Synthesis of indolizinium salts (microreview) Anna IvanovaPavel Arsenyan HETEROCYCLES IN FOCUS 24 April 2017 Pages: 313 - 315
Exploring the influence of the substituent at position 4 in a series of 3,4-dihydropyrimidin-2(1H)-one A2B adenosine receptor antagonists Abel CrespoAbdelaziz El MaatouguiEddy Sotelo OriginalPaper 26 April 2017 Pages: 316 - 321
Functionalization of four-membered cyclic sulfoximines by a convenient lithiation/trapping sequence Arianna TotaFlavio FanelliLeonardo Degennaro OriginalPaper 27 April 2017 Pages: 322 - 328
2-Arylazetidines as ligands for nicotinic acetylcholine receptors Leonardo DegennaroMarina ZenzolaGiovanni Lentini OriginalPaper 26 April 2017 Pages: 329 - 334
Synthesis and structure of dihydroberberine nitroaryl derivatives – potential ligands for G-quadruplexes Oleg N. BurovSergey V. KurbatovIgor E. Mikhailov OriginalPaper 26 April 2017 Pages: 335 - 340
Investigation on the synthesis of new 3-[4-(arylalkoxy)phenylethyl]-2-thioxo-1,3-thiazolidin-4-ones and their biological evaluation against cancer cells Camille Déliko DagoChristelle N’ta AmbeuJean-Pierre Bazureau OriginalPaper 27 April 2017 Pages: 341 - 349
Synthesis of phenylpyridine derivatives and their biological evaluation toward dipeptidyl peptidase-4 Yan ZhuXiangguo MengWeicheng Zhou OriginalPaper 26 April 2017 Pages: 350 - 356
Physicochemical properties and antimicrobial activity of new spirocyclic thieno[2,3-d]pyrimidin-4(3H)-one derivatives Modesto de CandiaClaudia AltamuraCosimo D. Altomare OriginalPaper 27 April 2017 Pages: 357 - 363
Synthesis of new heterocyclic dehydroabietylamine derivatives and their biological activity Kseniya S. KovalevaOlga I. YarovayaNariman F. Salakhutdinov OriginalPaper 27 April 2017 Pages: 364 - 370
Synthesis and biological activity of heterocyclic borneol derivatives Anastasiya S. SokolovaOlga I. YarovayaNariman F. Salakhutdinov OriginalPaper 24 April 2017 Pages: 371 - 377
(5S,7R)-5-Aryl-7-methyl-4,5,6,7-tetrahydro-[1, 2, 4]triazolo[1,5-a]pyrimidin-7-ols as products of three-component condensation Sergey A. KomykhovAndrey A. BondarenkoSergey M. Desenko SHORT COMMUNICATION 22 April 2017 Pages: 378 - 380