Abstract
The physiological effects of epinephrine and norepinephrine are caused by the interaction of these compounds with specific receptor molecules on the external surface of target cells. Since both epinephrine and norepinephrine are found in large quantities in the adrenal gland, these receptors are called adrenergic receptors. Although the existence of these receptor molecules has been suspected for many years, it is only very recently that some information on their molecular and chemical nature has become available.
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References
Aarons, R.D., Nies, A.S., Gal, J., Hegstrand, L.R. and Molinoff, P.B. (1980), J. Clin. Invest., 65, 949–957.
Ahlquist, R.P. (1948), Am. J. Physiol., 153., 586–600.
Aktories, K., Schultz, G. and Jakobs, K.H. (1979), FEBS Lett., 107, 100–104.
Alexander, R.W., Williams, L.T. and Lefkowitz, R.J. (1975a), Proc. Natl. Acad. Sci. USA., 72., 1564–1568.
Alexander, R.W., Davis, J.N. and Lefkowitz, R.J. (1975b), Nature (London), 258, 437–440.
Altman, J. and Anderson, W.J. (1973), J. Comp. Neurol., 149, 123–152.
Anderson, W.B. and Jaworski, C.J. (1979), J. Biol. Chem., 254, 4596–4601.
Ariens, E.J. and Simonis, A.M. (1976), in Beta-Adrenoceptor Blocking Agents (eds. P.R. Saxena and R.P. Forsyth), North-Holland Publishing Co., Amsterdam, pp 3–27.
Armstrong, D.H. and Schild, R.F. (1970), J. Comp. Neurol., 139, 449–456.
Arnold, A. and McAuliff, J.P. (1969), Arch. Int. Pharmacodyn., 179, 381–387.
Arnold, A., McAuliff, J.P., Colella, D.F., O’Connor, W.V. and Brown, Th.G. (1968), Arch. Int. Pharmacodyn., 176, 451–457.
Atlas, D. and Levitzki. A. (1977), Proc. Natl. Acad. Sci. USA., 74, 5290–5294.
Atlas, D. and Melamed, E. (1978), Brain Res., 150, 377–385.
Aurbach, G.D., Fedak, S.A., Woodard, C.J., Palmer, J.S., Hauser, D. and Troxler, F. (1976), Science, 186, 1223–1224.
Axelrod, J., Shein, H.M. and Wurtman, R.J. (1969), Proc. Natl. Acad. Sci. USA., 62, 544–549.
Bakardjieva, A., Calla, H.J. and Helmreich, E.J. (1979), Biochemistry, 18, 3016–3023.
Baker, S.P. and Potter, L.T. (1980a), Br. J. Pharmacol., 68, 65–70.
Baker, S.P. and Potter, L.T. (1980b), Br. J. Pharmacol., 68, 8–10.
Baker, S.P., Boyd, H.M. and Potter, L.T. (1980), Br. J. Pharmacol., 68, 57–63.
Banerjee, S.P., Kung, L.S., Riggi, S.J. and Chanda, S.K. (1977), Nature (London), 268, 455–456.
Banerjee, S.P., Sharma, V.K., Kung, L.S. and Chanda, S.K. (1978), Nature (London), 271, 380–381.
Baraban, J.M. and Aghajanian, G.K. (1980), Neuropharmacology, 19, 355–363.
Barnes, P., Karliner, J., Hamilton, C. and Dollery, C. (1979), Life Sci., 25, 1207–1214.
Barnes, P., Koppel, H., Lewis, P., Hutson, C., Blair, I. and Dollery, C. (1980), Brain Res., 181, 209–213.
Barnett, D.B., Rugg, E.L. and Nahorski, S.R. (1978), Nature (London), 273, 166–168.
Berridge, M.J. and Fain, J.M. (1979), Biochem. J., 178, 59–69.
Berthelsen, S. and Pettinger, W.A. (1977), Life Sci., 21, 595–606.
Bevan, P., Bradshaw, C.M. and Szabadi, E. (1977), Br. J. Pharmacol., 59, 635–641.
Bickerton, R.K. (1963), J. Pharmacol. Exp. Ther., 142, 99–110.
Bilezikian, J.P. and Aurbach, G.D. (1973), J. Biol. Chem., 248, 5575–5583.
Bilezikian, J.P., Spiegel, A.M., Gammon, D.E. and Aurbach, G.D. (1977a), Mol. Pharmacol., 13, 786–795.
Bilezikian, J.P., Spiegel, A.M., Brown, E.M. and Aurbach, G.D. (1977b), Mol. Pharmacol., 13, 775–785.
Bilezikian, J.P., Loeb, J.N. and Gammon, D.E. (1979), J. Clin. Invest., 63, 184–192.
Bird, S.J. and Maguire, M.E. (1978), J. Biol. Chem., 253, 8826–8834.
Black, J.W., Crowther, A.F., Shanks, R.G., Smith, L.H. and Dornhorst, A.C. (1964), Lancet, 1, 1080–1081.
Bloom, F.E., Hoffer, B.J. and Siggins, G.R. (1972), Biol. Psychiat., 4, 157–177.
Blume, A.J. (1978), Proc. Natl. Acad. Sci. USA., 75, 1713–1717.
Boeynaems, J.M. and Dumont, J.E. (1977), Mol. Cell. Endocrinol., 7, 33–47.
Bottari, S., Vauquelin, G., Durieu, O., Kluthchko, C. and Strosberg, A.D. (1979), Biochem. Biophys. Res. Commun., 86, 1311–1318.
Bourne, H.R., Coffino, P. and Tomkins, G.M. (1975), Science, 187, 750–752.
Bowman, W.C. and Nott, M.W. (1969), Pharmacol. Rev., 21, 27–72.
Brittain, R.T., Farmer, J.B., Jack, D., Marin, L.E. and Simpson, W.T. (1968), Nature (London), 219, 862–863.
Brown, E.M., Aurbach, G.D., Hauser, D. and Troxler, F. (1976a), J. Biol. Chem., 251, 1232–1238.
Brown, E.M., Fedak, S.M., Woodard, C.J., Aurbach, G.D. and Rodbard, D. (1976b), J. Biol. Chem., 251, 1239–1246.
Brown, M., Hurwitz, S.H. and Aurbach, G.D. (1978), Endocrinology, 103, 893–899.
Burges, R.A. and Blackburn, K.J. (1972), Nature (London) New Biol., 235, 249–250.
Burns, J.J., Colville, K.I., Lindsay, L.A. and Salvador, R.A. (1964), J. Pharmacol. Exp. Ther., 144, 163–171.
Burns, T.W., Langley, P.E. and Robison, G.A. (1971), Ann. N.Y. Acad. Sci., 185, 115–128.
Bylund, D.B. and Snyder, S.H. (1976), Mol. Pharmacol.12, 568–580.
Cambridge, D., Davey, M.J. and Massingham, R. (1977), Br. J. Pharmacol., 59, 514P.
Cannon, W.B. and Rosenblueth, A. (1937), Autonomic Neuroeffector Systems, Macmillan, New York.
Carlsson, E. and Hedberg, A. (1977), Acta Physiol. Scand. Suppl.,44, 47.
Carlsson, E., Ablad, B., Brandstrom, A. and Carlsson, B. (1972), Life Sci., 11, 953–958.
Carlsson, E., Dahlof, C-G., Hedberg, A., Persson, H. and Tangstrand, B. (1977), Naunyn-Schmiedeberg’s Arch. Pharmacol., 300, 101–105.
Caron, M.G. and Lefkowitz, R.J. (1976), J. Biol. Chem., 251, 2374–2384.
Caron, M.G., Srinivasan, Y., Pitha, J., Kociolek, K. and Lefkowitz, R.J. (1979), J. Biol. Chem., 254, 2923–2927.
Cassel, D. and Pfeuffer, T. (1978), Proc. Natl. Acad. Sci. USA, 75, 2669–2673.
Cassel, D. and Selinger, Z. (1976), Biochim, Biophys. Acta, 452, 538–551.
Cassel, D. and Selinger, Z. (1977a), J. Cyclic Nucleotide Res., 3, 11–22.
Cassel, D. and Selinger, Z. (1977b), Proc. Natl. Acad. Sci. U.S.A., 74, 3307–3311.
Cassel, D. and Selinger, Z. (1978), Proc. Natl. Acad. Sci. U.S.A., 75, 4155–4159.
Catt, K.J., Harwood, J.P., Aguilera, G. and Dufau, M.L. (1979), Nature (London), 280, 109–116.
Cedarbaum, J.M. and Aghajanian, G.K. (1977), Eur. J. Pharmacol., 44, 375–385.
Chan, T.M. and Exton, J.H. (1977), J. Biol. Chem., 252, 8645–8651.
Chang, R.S.L., Tran, V.T. and Snyder, S.H. (1980), Brain Res., 190, 95–110.
Charness, M.E., Bylund, D.R., Beckman, B.S., Hollenberg, M.D. and Snyder, S.H. (1976), Life Sci., 19, 243–250.
Chasin, M., Mamrak, F. and Sulser, F. (1974), J. Neurochem., 22, 1031–1038.
Chen, F.M., Yamamura, H.I. and Roeske, W.R. (1979), Eur. J. Pharmacol., 58, 255–264.
Chuang, D-M., and Costa, E. (1979), Proc. Natl. Acad. Sci. U.S.A., 76, 3024–3028.
Ciaraldi, T. and Marinetti, G.V. (1977), Biochem. Biophys. Res. Commun., 74, 984–990.
Coleman, A.J., Paterson, D.S. and Somerville, A.R. (1979), Biochem. Pharmacol., 28, 1003–1010.
Coyle, J.T. and Schwarcz, R. (1976), Nature (London), 263, 244–246.
Creese, I., Usdin, T.B. and Snyder, S.H. (1979), Mol. Pharmacol., 16, 69–76.
Cuatrecasas, P. (1971), Proc. Natl. Acad. Sci. U.S.A., 68, 1264–1266.
Cuatrecasas, P. (1974), Annu. Rev. Biochem., 43, 169–214.
Cuatrecasas, P., Tell, G.P., Sica, V., Parikh, I. and Chang, K-J. (1974), Nature (London), 247, 92–97.
Cubeddu, L.X., Barnes, E., Langer, S.Z. and Weiner, N. (1974), J. Pharmacol. Exp. Ther., 190, 431–450.
Dahlof, C., Ljung, B. and Ablad, B. (1978), Eur. J. Pharmacol., 50, 75–78.
Dale, H.H. (1907), J. Physiol. (London), 34, 163–206.
Davis, J.N. and Lefkowitz, R.J. (1976), Brain Res., 113, 214–218.
Davis, J.N., Strittmatter, W., Hoyler, E. and Lefkowitz, R.J. (1977), Brain Res., 132, 327–336.
Davis, J.N., Arnett, C.D., Hoyler, E., Stalvey, L.P., Daly, J.W. and Skolnick, P. (1978), Brain Res., 159, 125–135.
Deguchi, T. and Axelrod, J. (1972), Proc. Natl. Acad. Sci. U.S.A., 69, 2208–2211.
Deguchi, T. and Axelrod, J. (1973), Proc. Natl. Acad. Sci. U.S.A., 70, 2411–2414.
DeHaen, C. (1976), J. Theoret. Biol., 58, 383–400.
DeLean, A., Stadel, J.M. and Lefkowitz, R.J. (1980), J. Biol. Chem.255, 7108–7117.
DeVellis, J. and Brooker, G. (1974), Science, 186, 1221–1223.
Dibner, M.D. and Molinoff, P.B. (1979), J. Pharmacol. Exp. Ther., 210, 433–439.
Dillier, N., Laszlo, J., Muller, B., Koella, W.P. and Olpe, H.-R. (1978), Brain Res., 154, 61–74.
Dolphin, A., Adrien, J., Hamon, M. and Bockaert, J. (1979), Mol. Pharmacol., 15, 1–15.
Dungan, K.W., Cho, Y.W., Gomoll, A.W., Aviado, D.M. and Lish, P.M. (1968), J. Pharmacol. Exp. Ther., 164, 290–301.
Dunlop, D. and Shanks, R.G. (1968), Br. J. Pharmacol., 32, 201–218.
Dunnick, J.K., Marinetti, G.V. (1971), Biochim, Biophys. Acta, 249, 122–134.
Edvinsson, L. and Owman, C. (1974), Circ. Res., 35, 835–849.
Exton, J.H. (1979), J. Cyclic Nucleotide Res., 5, 277–287.
Fain, J.N. and Garcia-Sainz, J.A. (1980), Life Sci., 26, 1183–1194.
Furchgott, R.F. (1972), Handb. Exp. Pharmacol., 33, 283–335.
Gibson, R.E., Rzeszotarski, W.J., Komai, T., Reba, R.C. and Eckelman, W.C. (1979), J. Pharmacol. Exp. Ther., 209, 153–161.
Gill, D.M. (1975), Proc. Natl. Acad. Sci. U.S.A., 72. 2064–2068
Gill, D.M. and Meren, R. (1978), Proc. Natl. Acad. Sci. U.S.A., 75, 3050–3054.
Glaubiger, G. and Lefkowitz, R.J. (1977), Biochem. Biophys. Res. Commun., 78, 720–725.
Glaubiger, G., Tsai, B.S., Lefkowitz, R.J., Weiss, B. and Johnson, E.M., Jr. (1978), Nature (London) 273, 240–242.
Govier, W.C. (1968), J. Pharmacol. Exp. Ther.,159, 82–90.
Greenberg, D.A. and Snyder, S.H. (1978), Mol. Pharmacol., 14, 38–49.
Greenberg, D.A., U’Prichard, D.C. and Snyder, S.H. (1976), Life Sci., 19, 69–76.
Greenberg, L.H. and Weiss, B. (1978), Science, 201, 61–63.
Greenglass, P. and Bremner, R. (1979), Eur. J. Pharmacol., 55, 323–326.
Gross, G., Brodde, O.-E. and Schumann, H.-J. (1980), Eur. J. Pharmacol., 61, 191–194.
Guellaen, G., Yates-Aggerbeck, M., Vauquelin, G., Strosberg, D. and Hanoune, J. (1978), J. Biol. Chem., 253, 1114–1120.
Haga, R., Ross, E.M., Anderson, H.J. and Gilman, A.G. (1977a), Proc. Natl. Acad. Sci. U.S.A., 74, 2016–2020.
Haga, R., Haga, K. and Gilman, A.G. (1977b), J. Biol. Chem., 252, 5778–5782.
Hancock, A.A., DeLean, A.L. and Lefkowitz, R.J. (1979), Mol. Pharmacol., 16, 1–9.
Hanski, E., Rimon, G. and Levitzki, A. (1979), Biochemistry, 18, 846–853.
Harden, T.K., Wolfe, B.B. and Molinoff, P.B. (1976), Mol. Pharmacol., 12, 1–15.
Harden, T.K., Wolfe, B.B., Sporn, J.R., Perkins, J.P. and Molinoff, P.B. (1977a), Brain Res., 125, 99–108.
Harden, T.K., Wolfe, B.B., Sporn, J.R., Poulos, B.K. and Molinoff, P.B. (1977b), J. Pharmacol. Exp. Ther., 203, 132–143.
Harden, T.K., Su, Y-F. and Perkins, J.P. (1979), J. Cyclic Nucleotide Res., 5, 99–106.
Harik, S.I., Sharma, V.K., Wetherbee, J.R., Warren, R.H. and Banerjee, S.P. (1980), Eur. J. Pharmacol., 61, 207–208.
Hedberg, A. (1980), Private communication.
Hedberg, A., Minneman, K.P. and Molinoff, P.B. (1980), J. Pharmacol. Exp. Ther., 213, 503–508.
Hegstrand, L.R., Minneman, K.P. and Molinoff, P.B. (1979), J. Pharmacol. Exp. Ther., 210., 215–221.
Heidenreich, K.H., Weiland, G.A. and Molinoff, P.B. (1980), J. Cyclic Nucleotide Res., 6,217–230.
Heidmann, T. and Changeux, J.-P. (1978), Annu. Rev. Biochem., 47, 317–357.
Hendley, E. (1978), Soc. Neurosci. Abstr., 4, 494.
Herbst, T.J., Raichle, M.E. and Ferrendelli, J.A. (1979), Science., 204, 330–332.
Hess, A. (1979), Brain Res., 160, 533–538.
Hirata, F. and Axelrod, J. (1980), Science., 209, 1082–1090.
Hirata, F., Strittmatter, W.J. and Axelrod, J. (1979), Proc. Natl. Acad. Sci. U.S.A., 76, 368–372.
Hoffer, B.J., Siggins, G.R. and Bloom, F.E. (1971), Brain Res., 25, 523–534.
Hoffman, B. and Lefkowitz, R.J. (1980), Biochem. Pharmacol., 29, 1537–1541.
Hokfelt, T., Fuxe, K., Goldstein, M. and Johansson, O. (1974), Brain Res., 66, 235–251.
Hokin, L.E. and Sherwin, A.L. (1957), J. Physiol. (London), 135, 18–29.
Howlett, A.C., Van Arsdale, P.M. and Gilman, A.G. (1978), Mol. Pharmacol., 14, 531–539.
Howlett, A.C., Sternweis, P.C., Macik, B.A., Van Arsdale, P.M. and Gilman, A.G. (1979), J. Biol. Chem., 254, 2287–2295.
Ignarro, L.J. and Titus, E. (1968), J. Pharmacol. Exp. Ther., 160, 72–80.
Innes, I.R. (1962), Br. J. Pharmacol. Chemother., 19, 120–128.
Insel, P.A., Maguire, M.E., Gilman, A.G., Bourne, H.R., Coffino, P. and Melmon, K.L. (1976), Mol. Pharmacol., 12, 1062–1069.
Iversen, L.L. (1967), The Uptake and Storage of Noradrenaline in Sympathetic Nerves, Cambridge University Press, Cambridge.
Jacobs, S. and Cuatrecasas, P. (1976), Biochem. Biophys. Acta, 433, 482–495.
Johnson, G.L., Wolfe, B.B., Harden, T.K., Molinoff, P.B. and Perkins, J.P. (1978a), J. Biol. Chem., 253, 1472–1480.
Johnson, G.L., Kaslow, H.R. and Bourne, H.R. (1978b), J. Biol. Chem., 253, 7120–7123.
Johnson, G.L., Kaslow, H.R., Farfel, Z. and Bourne, H.R. (1980), Adv. Cyclic Nucleotide Res., 13,1–37.
Jones, L.M. and Michell, R.H. (1974), Biochem. J., 142, 583–590.
Kalisker, A., Rutledge, C.O. and Perkins, J.P. (1973), Mol. Pharmacol., 9, 619–629.
Kauzmann, W. (1959), Adv. Protein Chem., 14, 1–63.
Kebabian, J.W., Zatz, M., Romero, J.A. and Axelrod, J. (1975), Proc. Natl. Acad. Sci. U.S.A., 72, 3735–3739.
Kent, R.S., DeLean, A. and Lefkowitz, R.J. (1980), Mol. Pharmacol., 17, 14–23.
Kirk, C.J., Verrinder, T.R. and Hems, D.A. (1977), FEBS Lett., 83, 267–271.
Klainer, L.M., Chi, Y-M., Freidberg, S.L., Rall, T.W. and Sutherland, E.W. (1962), J. Biol. Chem., 237, 1239–1243.
Klein, D.C., Berg, G.R. and Weller, J.L. (1970), Science, 168, 979–980.
Kleinstein, J. and Glossman, H. (1978), Naunyn Schmiedebergs Arch. Pharmacol.305, 191–200.
Klotz, I.M. and Urguhart, J.M. (1949), J. Am. Chem. Soc., 71, 847–851.
Kneer, N.M., Wagner, M.J. and Lardy, H.A. (1979), J. Biol. Chem., 254, 12160–12168.
Krawietz, W., Weinsteiger, M., Pruchniewski, M. and Erdmann, E. (1979), Biochem. Pharmacol., 2999–3007.
Kuffler, S.W. (1943), J. Neurophys., 6, 99–110.
Lad, P.M., Nielsen, T.B., Preston, M.S. and Rodbell, M. (1980), J. Biol. Chem., 255, 988–995.
Lands, A.M., Arnold, A., McAuliff, J.P., Luduena, F.P. and Brown T.T. (1967a), Nature (London), 214, 597–598.
Lands, A.M., Luduena, F.P. and Buzzo, H.J. (1967b), Life Sci., 6, 2241–2249.
Langer, S.Z. (1974), Biochem. Pharmacol., 23, 1793–1800.
Langer, S.Z. (1977), Br. J. Pharmacol., 60, 481–497.
Lauzon, G.J., Kulshrestha, S., Starr, L. and Bar, H. (1976), J. Cyclic Nucleotide Res., 2, 99–114.
Lefkowitz, R.J. (1974), Biochem. Biophys. Res. Commun., 58, 1110–1118.
Lefkowitz, R.J. (1975), Biochem. Pharmacol., 24, 583–590.
Lefkowitz, R.J. and Haber, E. (1971), Proc. Natl. Acad. Sci. U.S.A., 68, 1773–1777.
Lefkowitz, R.J. and Hamp, M. (1977), Nature (London), 268, 453–454.
Lefkowitz, R.J. and Williams, L.T. (1977), Proc. Natl. Acad. Sci. U.S.A., 74, 515–519.
Lefkowitz, R.J., Haber, E. and O’Hara, D. (1972), Proc. Natl. Acad. Sci. U.S.A 69, 2828–2832.
Lefkowitz, R.J., Mukherjee, C., Coverstone, M. and Caron, M.G. (1974), Biochem. Biophys. Res. Commun., 60., 703–709.
Lefkowitz, R.J ., Mullikin, D. and Caron, M.G. (1976), J. Biol. Chem., 251, 4684–4692.
Levitzki, A., Atlas, D. and Steer, M.L. (1974), Proc. Natl. Acad. Sci. U.S.A., 71, 2773–2776.
Levitzki, A., Sevilia, N., Atlas, D. and Steer, M.L. (1975), J. Mol. Biol., 97, 35–53.
Levy, B. (1966), J. Pharmacol. Exp. Ther., 151, 413–422.
Limbird, L.E. and Lefkowitz, R.J. (1976), J. Biol. Chem., 251, 5007–5014.
Limbird, L.E. and Lefkowitz, R.J. (1977), J. Biol. Chem., 252, 799–802.
Limbird, L.E. and Lefkowitz, R.J. (1978), Proc. Natl. Acad. Sci. U.S.A.75, 228–232.
Limbird, L.E., De Meyts, P. and Lefkowitz, R.J. (1975), Biochem. Biophys. Res. Commun., 64, 1160–1168.
Limbird, L.E., Hickey, A.R. and Lefkowitz, R.J. (1979), J. Biol. Chem., 254, 2677–2683.
Limbird, L.E., Gill, D.M. and Lefkowitz, R.J. (1980), Proc. Natl. Acad. Sci. U.S.A., 77, 775–779.
Lin, M.C., Nicosia, S., Lad, P.M. and Rodbell, M. (1977), J. Biol. Chem., 252, 2790–2792.
Maggi, A., Schmidt, M.J., Ghetti, B. and Enna, S.J. (1979), Life Sci., 24, 367–374.
Maggi, A., U’Prichard, D.C. and Enna, S.J. (1980), Science, 207, 645–647.
Maguire, M.E., Goldman, P.H. and Gilman, A.G. (1974), Mol. Pharmacol., 10, 563–581.
Maguire, M.E., Wiklund, R.A., Anderson, H.J. and Gilman, A.G. (1976a), J. Biol. Chem., 251, 1221–1231.
Maguire, M.E., Van Arsdale, P.M. and Gilman, A.G. (1976b), Mol. Pharmacol., 12, 335–339.
Maguire, M.E., Ross, E.M. and Gilman, A.G. (1977), Adv. Cyclic Nucleotide Res., 8, 1–83.
Malbon, C.C. and Cabelli, R.J. (1978), Biochim. Biophys. Acta, 544, 93–101.
Malbon, C.C., Moreno, F.J., Cabelli, R.J. and Fain, J.N. (1978), J. Biol. Chem., 253, 671–678.
Mallorga, P., Tallman, J.F., Henneberry, R.C., Hirata, F., Strittmatter, W.J. and Axelrod, J. (1980), Proc. Natl. Acad. Sci. U.S.A., 77, 3341–3345.
Mayer, S.E. (1978), Beta Adrenergic Blockade: A New Era in Cardiovascular Medicine (ed. E. Braunwald), Excerpta Medica, Amsterdam, pp 25–37.
Mayer, S.E. (1980), in The Pharmacological Basis of Therapeutics (eds. A.G. Gilman, L.S. Goodman and A. Gilman), MacMillan, New York, pp 56–90.
Mayer, S.E. and Moran, N.C. (1960), J. Pharmacol. Exp. Ther., 129, 271–281.
McGeer, E.G. and McGeer, P.L. (1976), Nature (London), 263, 517–519.
Miach, P.J., Dausse, J.-P. and Meyer, P. (1978), Nature (London), 274, 492–494.
Miach, P.J., Dausse, J-P, Cardot, A. and Meyer, P. (1980), Naunyn Schmiedeberg’s Arch. Pharmacol., 313, 23–26.
Michell, R.H. (1975), Biochim. Biophys. Acta, 415, 81–147.
Mickey, J., Tate, R. and Lefkowitz, R.J. (1975), J. Biol. Chem., 250, 5727–5729.
Mickey, J., Tate, R., Mullikin, D. and Lefkowitz, R.J. (1976), Mol. Pharmacol., 12, 409–419.
Minneman, K.P. (1977), Mol. Pharmacol., 13, 735–744.
Minneman, K.P. and Iversen, L.L. (1976), Science, 192, 803–805.
Minneman, K.P. and Molinoff, P.B. (1980), Biochem. Pharmacol., 29, 1317–1323.
Minneman, K.P., Quik, M. and Emson, P.C. (1978), Brain Res., 151, 507–521.
Minneman, K.P., Hegstrand, L.R. and Molinoff, P.B. (1979a), Mol. Pharmacol., 16, 21–33.
Minneman, K.P., Hegstrand, L.R. and Molinoff, P.B. (1979b), Mol. Pharmacol., 16, 34–46.
Minneman, K.P., Hedberg, A. and Molinoff, P.B. (1979c), J. Pharmacol. Exp. Ther., 211, 502–508.
Minneman, K.P., Dibner, M.D., Wolfe, B.B. and Molinoff, P.B. (1979d), Science, 204, 866–868.
Minneman, K.P., Weiland, G.A. and Molinoff, P.B. (1980a), Mol. Pharmacol., 17, 1–7.
Minneman, K.P., Pittman, R.N., Yeh, H., Woodward, D.J. and Molinoff, P.B. (1980b), Brain Res., in press.
Minneman, K.P., Pittman, R.N. and Molinoff, P.B. (1981), Annu. Rev. Neurosci., 4, 419–461.
Mobley, P.L. and Sulser, F. (1980), Nature (London), 286, 608–609.
Moises, H.C., Woodward, D.J., Hoffer, B.J. and Freedman, R. (1979), Exp. Neurol., 64, 493–515.
Molinoff, P.B. and Axelrod, J. (1971), Annu. Rev. Biochem., 40, 465–500.
Moran, N.C. (1975), Handb. Physiol.-Endocrinol. Sect. 7, 6, 447–472.
Moran, N.C. and Perkins, M.E. (1958), J. Pharmacol. Exp. Ther., 124, 223–237.
Mukherjee, C. and Lefkowitz, R.J. (1977), Mol. Pharmacol., 13, 291–303.
Mukherjee, C., Caron, M.G., Coverstone, M. and Lefkowitz, R.J. (1975), J. Biol. Chem., 250, 4869–4876.
Murad, F. (1973), Biochim. Biophys. Acta, 304, 181–187.
Nahorski, S.R. (1976), Nature (London), 259, 488–489.
Nahorski, S.R. (1977), Mol. Pharmacol., 13, 679–689.
Nahorski, S.R. (1978), Eur. J. Pharmacol., 51, 199–209.
Nahorski, S.R., Barnett, D.B., Howlett, D.R. and Rugg, E.L. (1979a), Naunyn Schmiedeberg’s Arch. Pharmacol., 207, 227–233.
Nahorski, S.R., Howlett, D.R. and Redgrave, P. (1979b), Eur. J. Pharmacol., 60, 249–252.
Nathanson, J.A. (1977), Physiol. Rev., 57, 157–256.
Nathanson, J.A. (1980), Life Sci., 26, 1793–1799.
Nathanson, J.A. and Glaser, G.H. (1979), Nature (London), 278, 567–569.
Nickerson, M. (1949), Pharmacol. Rev., 1, 27–101.
Nickerson, M. and Goodman, L.S. (1947), J. Pharmacol. Exp. Ther., 89, 167–185.
Nickols, G.A. and Brooker, G. (1979), J. Cyclic Nucleotide Res., 5, 435–477.
Nordeen, S.K. and Young, D.A. (1978), J. Biol. Chem., 253, 1234–1239.
O’Donnell, S.R. and Wanstall, J.C. (1979), Naunyn Schmiedeberg’s Arch. Pharmacol., 308, 183–190.
Olpe, H.R. and Schellenberg, A. (1980), Eur. J. Pharmacol., 63, 7–13.
Palacios, J.M. and Kuhar, M.J. (1980), Science, 208, 1378–1380.
Palmer, G.C. (1972), Neuropharmacology, 11, 145–149.
Partington, C.R., Edwards, M.W. and Daly, J.W. (1980), Proc. Natl. Acad. Sci. U.S.A., 77, 3024–3028.
Peroutka, S.J., Greenberg, D.A., U’Prichard, D.C. and Snyder, S.H. (1978), Mol. Pharmacol., 14, 403–412.
Peroutka, S.J., Moskowitz, M.A., Reinhard, J.F., Jr. and Snyder, S.H. (1980), Science, 208, 610–612.
Petrack, B. and Czernik, A.J. (1976), Mol. Pharmacol., 12, 203–207.
Pfeuffer, T. (1977), J. Biol. Chem., 252, 7224–7234.
Pfeuffer, T. and Helmreich, E.J.M. (1975), J. Biol. Chem., 250, 867–876.
Pike, L.J. and Lefkowitz, R.J. (1978), Mol. Pharmacol., 14, 370–375.
Pittman, R.N., Minneman, K.P. and Molinoff, P.B. (1980a), Brain Res., 188, 357–368.
Pittman, R.N., Minneman, K.P. and Molinoff, P.B. (1980b), J. Neurochem., 35, 273–275.
Pollet, R.J., Standaert, M.L. and Haase, B.A. (1980), Proc. Natl. Acad. Sci. U.S.A., 77, 4340–4344.
Potter, L.T. (1967), J. Pharmacol. Exp. Ther., 155, 91–100.
Powell, C.E. and Slater, I.H. (1958), J. Pharmacol. Exp. Ther., 122, 480–488.
Reisine, T.D., U’Prichard, D.C., Wiech, N.L., Ursillo, R.C. and Yamamura, H.I. (1980), Brain Res., 188, 587–592.
Roberts, J.M., Insel, P.A., Goldfien, R.D. and Goldfien, A. (1977), Nature (London), 270, 624–625.
Robison, G.A., Butcher, R.W. and Sutherland, E.W. (1971), Cyclic AMP, Academic Press, New York, Chapter 6.
Rodbell, M., Krans, H.M., Pohl, S.L. and Birnbaumer, L. (1971a), J. Biol. Chem., 246, 1861–1871.
Rodbell, M., Krans, H.M.J., Pohl, S.L. and Birnbaumer, L. (1971b), J. Biol. Chem., 246, 1872–1876.
Rodbell, M., Birnbaumer, L., Pohl, S.L. and Krans, H.M.J. (1971c), J. Biol. Chem., 246, 1877–1882.
Rogers, J., Silver, M.A., Shoemaker, W.J. and Bloom, F.E. (1979), Soc. Neurosci. Abstr., 5, 10.
Romero, J.A. and Axelrod, J. (1974), Science, 184, 1091–1092.
Romero, J.A., Zatz, M., Kebabian, J.W. and Axelrod, J. (1975), Nature (London), 258, 435–436.
Rosenberger, L.B., Roeske, W.R. and Yamamura, H.R. (1979), Eur. J. Pharmacol., 58, 255–257.
Rosenberger, L.B., Yamamura, H.I. and Roeske, W.R. (1980), Eur. J. Pharmacol., in press.
Ross, E.M. and Gilman, A.G. (1977), Proc. Natl. Acad. Sci. U.S.A..74, 3715–3719.
Ross, E.M. and Gilman, A.G. (1980), Annu. Rev. Biochem., 49, 533–564.
Ross, E.M., Maguire, M.E., Sturgill, T.W., Biltonen, R.L. and Gilman, A.G. (1977), J. Biol. Chem., 252, 5761–5775.
Ross, E.M., Howlett, A.C., Ferguson, K.M. and Gilman, A.G. (1978), J. Biol. Chem., 253, 6401–6412.
Rouot, B.R. and Snyder, S.H. (1979), Life Sci., 25, 759–774.
Rouot, B.M., U’Prichard, D.C. and Snyder, S.H. (1980), J. Neurochem., 34, 374–384.
Rugg, E.L., Barnett, D.B. and Nahorski, S.R. (1978), Mol. Pharmacol., 14, 996–1005.
Russell, M.P. and Moran, N.C. (1980), Circ. Res., 46, 344–352.
Sabol, S.L., and Nirenberg, M. (1979), J. Biol. Chem., 254, 1913–1920.
Salzman, E.W. and Neri, L.L. (1969), Nature (London), 224, 609–610.
Scatchard, G. (1949), Ann. N.Y. Acad. Sci., 51, 600–672.
Schramm, M. (1976), J. Cyclic Nucleotide Res., 2, 347–358.
Schramm, M. and Rodbell, M. (1975), J. Biol. Chem., 250, 2232–2237.
Schramm, M., Feinstein, H., Naim, E., Lang, M. and Lasser, M. (1972), Proc. Natl. Acad. Sci. U.S.A., 69, 523–527.
Schramm, M., Orley, J., Eimerl, S. and Korner, M. (1977), Nature (London), 268, 310–313.
Schultz, J. (1976), Nature (London), 261, 417–418.
Schumann, H.J., Endoh, M. and Wagner, J. (1974), Naunyn Schmiedeberg’s Arch. Pharmacol., 284, 133–148.
Schwarcz, R. and Coyle, J.T. (1976), Brain Res., 127, 235–249.
Segal, M. and Bloom, F.E. (1974), Brain Res., 72, 99–114.
Sercombe, R., Aubineau, P., Edvinsson, L., Mamo, H., Owman, C. and Seylaz, J. (1977), Pflügers Arch., 368, 241–244.
Sharma, V.K. and Banerjee, S.P. (1978), J. Biol. Chem., 253, 5277–5279.
Shear, M., Insel, P., Melmon, K.L. and Coffino, P. (1976), J. Biol. Chem., 251, 7572–7576.
Shein, H.M. and Wurtman, R.J. (1969), Science, 166, 519–520.
Siggins, G.R., Hoffer, B.J. and Bloom, F.E. (1969), Science, 165, 1018–1020.
Singer, S.J. and Campbell, D.H. (1955), J. Am. Chem. Soc., 4851–4855.
Skolnick, P., Stalvey, L.P., Daly, J.W., Hoyler, E. and Davis, J.N. (1978), Eur. J. Pharmacol., 47, 201–210.
Smith, C.B. (1963), J. Pharmacol. Exp. Ther., 142, 163–170.
Sporn, J.R. and Molinoff, P.B. (1976), J. Cyclic Nucleotide Res., 2, 149–161.
Sporn, J.R., Harden, T.K., Wolfe, B.B. and Molinoff, P.B. (1976), Science, 194, 624–626.
Sporn, J.R., Wolfe, B.B., Harden, T.K. and Molinoff, P.B. (1977), Mol. Pharmacol., 13, 1170–1180.
Starke, K., Montel, H., Gayk, W. and Merker, R. (1974), Naunyn Schmiedeberg’s Arch. Pharmacol., 285, 133–150.
Starke, K., Borowski, E. and Endo, T. (1975), Eur. J. Pharmacol., 34, 385–388.
Sternweis, P.C. and Gilman, A.G. (1979), J. Biol. Chem., 254, 3333–3340.
Stone, T.W. (1976), Naunyn Schmiedeberg’s Arch. Pharmacol., 278, 333–340.
Strada, S.J. and Weiss, B. (1974), Arch. Biochem. Biophys., 160, 197–204.
Strickland, S., Palmer, G. and Massey, V. (1975), J. Biol. Chem., 250, 4048–4052.
Strittmatter, W.J., Davis, J.N. and Lefkowitz, R.J. (1977), J. Biol. Chem., 252, 5472–5477.
Strittmatter, W.J., Hirata, F. and Axelrod, J. (1979), Science, 204, 1205–1207.
Su, Y-F., Cubeddu, L. and Perkins, J.P. (1976), J. Cyclic Nucleotide Res., 2, 257–270.
Su, Y-F., Harden, T.K. and Perkins, J.P. (1979), J. Biol. Chem., 254, 38–41.
Sutherland, E.W. and Rall, T.W. (1960), Pharmacol. Rev., 12, 265–299.
Taylor, A. and Wilson, R. (1970), Experientia., 26, 267–269.
Terasaki, W.L. and Brooker, G. (1978), J. Biol. Chem., 253, 5418–5425.
Terasaki, W.L., Brooker, G., DeVellis, J., Inglish, D., Hsu, C-Y., and Moylan, R.D. (1978), Adv. Cyclic Nucleotide Res., 9, 33–52.
Trendelenburg, U. (1963), Pharmacol. Rev., 15, 225–276.
Tsai, B.S. and Lefkowitz, R.J. (1978a), Mol. Pharmacol., 14, 61–68.
Tsai, B.S. and Lefkowitz, R.J. (1978b), Mol. Pharmacol., 14, 540–548.
Tse, J., Wrenn, R.W. and Kuo, J.F. (1980), Endocrinology, 107, 6–16.
Tuttle, R.R. and Mills, J. (1975), Circ. Res., 36, 185–196.
U’Prichard, D.C. and Snyder, S.H. (1977), J. Biol. Chem., 252, 6450–6453.
U’Prichard, D.C. and Snyder, S.H. (1978a), J. Biol. Chem., 253, 3444–3452.
U’Prichard, D.C. and Snyder, S.H. (1978b), Eur. J. Pharmacol., 51, 145–155.
U’Prichard, D.C. and Snyder, S.H. (1979), Life Sci., 24, 79–88.
U’Prichard, D.C., Greenberg, D.A. and Snyder, S.H. (1977), Mol. Pharmacol., 13, 454–473.
U’Prichard, D.C., Bylund, D.B. and Snyder, S.H. (1978), J. Biol. Chem., 253, 5090–5102.
U’Prichard, D.C., Bechtel, W.D., Rouot, B.M. and Snyder, S.H. (1979), Mol. Pharmacol., 16, 47–60.
U’Prichard, D.C., Reisine, T.D., Mason, S.T., Fibiger, H.C. and Yamamura, H.I. (1980), Brain Res., 187, 143–154.
Vatner, D. and Lefkowitz, R.J. (1974), Mol. Pharmacol., 10, 450–456.
Vauquelin, G., Lacombe, M.L., Guellaen, G., Strosberg, A.D. and Hanoune, J. (1976), Biochem. Pharmacol., 25, 2605–2608.
Vauquelin, G., Geynet, P., Hanoune, J. and Strosberg, A.D. (1977), Proc. Natl. Acad. Sci. U.S.A., 74, 3710–3714.
Vauquelin, G., Bottari, S. and Strosberg, A.D. (1980a), Mol. Pharmacol., 17, 163–171.
Vauquelin, G., Bottari, S., Andre, C., Jacobsson, B. and Strosberg, A.D. (1980b), Proc. Natl. Acad. Sci. U.S.A., 77, 3801–3805.
Vetulani, J., Stawarz, R.J., Dingell, J.V. and Sulser, F. (1976a), Naunyn Schmiedeberg’s Arch. Pharmacol., 293, 109–114.
Vetulani, J., Stawarz, R.J. and Sulser, F. (1976b), J. Neurochem., 27, 661–666.
von Euler, U.S. (1956), Noradrenaline: Chemistry, Physiology, Pharmacology and Clinical Aspects, Thomas, Springfield, Illinois.
Watanabe, A.M., McConnaughey, M.M., Strawbridge, R.A., Fleming, J.W., Jones, L.R. and Besch, H.R., Jr. (1978), J. Biol. Chem., 253, 4833–4836.
Weiland, G.A., Minneman, K.P. and Molinoff, P.B. (1979), Nature (London), 281, 114–117.
Weiland, G.A., Minneman, K.P. and Molinoff, P.B. (1980), Mol. Pharmacol.18, 341–347.
Weiss, B. and Costa, E. (1968), J. Pharmacol Exp. Ther., 161, 310–319.
Weiss, B. and Costa, E. (1969), J. Pharmacol. Exp. Ther., 168, 146–152.
Weiss, B., Greenberg, L. and Cantor, E. (1979), Fed. Proc. Fed. Am. Soc. Exp. Biol., 38, 1915–1921.
Wikberg, J.E.S. (1978), Nature (London), 273, 164–166.
Williams, L.T. and Lefkowitz, R.J. (1977), J. Biol. Chem., 252, 7207–7213.
Williams, L.T., Mullikin, D. and Lefkowitz, R.J. (1976a), J. Biol. Chem., 251, 6915–6923.
Williams, L.T., Jarett, L. and Lefkowitz, R.J. (1976b), J. Biol. Chem., 251, 3096–3104.
Williams, L.T., Lefkowitz, R.J., Watanabe, A.M., Hathaway, D.R. and Besch, H.R., Jr. (1977), J. Biol. Chem., 252,2787–2789.
Williams, L.T., Mullikin, D. and Lefkowitz, R.J. (1978), J. Biol. Chem.253, 2984–2989.
Wolfe, B.B., (1980), Private communication.
Wolfe, B.B., Zirrolli, J.A., and Molinoff, P.B. (1974), Mol. Pharmacol., 10, 582–596.
Wolfe, B.B., Harden, T.K. and Molinoff, P.B. (1976), Proc. Natl. Acad. Sci. U.S.A., 73, 1343–1347.
Wolfe, B.B., Harden, T.K. and Molinoff, P.B. (1977), Annu. Rev. Pharmacol. Toxicol., 17, 575–604.
Wolfe, B.B., Harden, T.K., Sporn, J.R. and Molinoff, P.B. (1978), J. Pharmacol. Exp. Ther., 207, 446–457.
Wolff, J. and Cook, G.H. (1973), J. Biol. Chem., 248, 350–355.
Woodcock, E.A. and Johnston, C.I. (1980), Nature (London), 286, 159–160.
Woodward, D.J., Hoffer, B.J. and Altman, J. (1974), J. Neurobiol., 5, 283–304.
Yamashita, K., Yamashita, S. and Ogata, E. (1977), Life Sci., 21, 607–612.
Young, W.S., III and Kuhar, M.J. (1980), Proc. Natl. Acad. Sci. U.S.A., 77, 1696–1700.
Zahniser, N.R., Minneman, K.P. and Molinoff, P.B. (1979), Brain Res., 178, 589–595.
Zatz, M. (1978), Life Sci.21, 1267–1276.
Zatz, M., Romero, J.A. and Axelrod, J. (1976), Biochem. Pharmacol., 25, 903–906.
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Minneman, K.P. (1981). Adrenergic Receptor Molecules. In: Yamamura, H.I., Enna, S.J. (eds) Neurotransmitter Receptors. Receptors and Recognition, vol 10. Springer, Dordrecht. https://doi.org/10.1007/978-94-009-5928-6_5
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