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Selective Anodic Fluorination of Heterocycles. Potential Application towards Pharmaceuticals

  • Toshio Fuchigami

Abstract

Various heterocyclic compounds having potentially biological activities were regioselectively monofluorinated by electrochemical fluorination using various supporting fluoride salts. Indirect anodic fluorodesulfurization of β-lactams using triarylamine mediators was also successful.

Keywords

Heterocyclic Compound High Current Efficiency Fluoride Salt Platinum Anode Benzylic Carbon 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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Copyright information

© Springer Japan 1998

Authors and Affiliations

  • Toshio Fuchigami
    • 1
  1. 1.Department of Electronic ChemistryTokyo Institute of TechnologyNagatsuta, Yokohama 226Japan

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