Zusammenfassung
Analgetika mit antipyretischer Eigenschaft lassen sich in 3 Gruppen einteilen (Tabelle 1).
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Literatur
Adams S.S. (1960) Analgesics - antipyretics. J Pharm (Lond) 12: 251 - 252
Breddin K (1969) Die Hemmung der Thrombozytenaggregation in vitro and in vivo. Folia Haematol 92: 460 - 469
Breddin K, Scharrer I, Schepping M (1971) Die Hemmung der Plättchenaggregation mit Acetylsalicylsäure. MMW 113: 1284 - 1292
Brune K, Alpermann H (1983) Non-acidic pyrazoles: inhibition of prostaglandin production, carrageenan oedema and yeast fever. Agents Actions 13: 360 - 363
Brune K, Rainsford K.D., Wagner K, Peskar B.A. (1981) Inhibition by anti-inflammatory drugs of prostaglandin production in cultured macrophages. Naunyn-Schmiedebergs Arch Pharmacol 315: 269 - 276
Collins E (1981) Maternal and fetal effects of acetaminophen and salicylates in pregnancy. Obstet Gynecol 58: 57S - 62S
Cranston W.I., Rawlins M.D. (1972) Effects of intracerebral microinjection of sodium salicylate on temperature regulation in the rabbit. J Physiol 222: 257 - 266
Carlsson K.H., Jurna I (1987) The role of descending inhibition in the antinociceptive effects of the pyrazolone derivatives metamizol (dipyrone) and aminophenanzone („Pyramidon). Naunyn-Schmiedebergs Arch Pharmacol 335: 154 - 159
Carlsson K.H., Helmreich J, Jurna I (1987) Activation of inhibition from the periaqueductal grey matter mediates central analgesic effect of metamizol (dipyrone). Pain 27: 373 - 390
Carlsson K.H., Monzel W, Jurna I (1988) Depression by morphine and the non-opioid analgesic agents, metamizol (dipyrone), lysine acetylsalicylate, and paracetamol, of activity in rat thalamus neurones evoked by electrical stimulation of nociceptive afferents. Pain 32: 313 - 326
Ferreira S.H. (1972) Prostaglandins, aspirin-like drugs and analgesia. Nature 240: 200 - 203
Ferreira S.H., Moncada S, Vane JR (1971) Indomethacin and aspirin abolish prostaglandin release from spleen. Nature 231: 237 - 239
Flower R.J. (1974) Drugs which inhibit prostaglandin biosynthesis. Pharmacol Rev 26: 3367
Flower R.J., Blackwell G.J. (1976) The importance of phospholipase A2 in prostaglandin biosynthesis. Biochem Pharmacol 25: 285 - 291
Flower R.J., Vane J.R. (1972) Inhibition of prostaglandin synthetase in brain explains the antipyretic activity of paracetamol (4-acetamidophenol). Nature 240: 410 - 411
Flower R.J., Gryglewski R.J., Herbaczynska-Credo K, Vane R (1972) Effects of anti-inflammatory drugs on prostaglandin biosynthesis. Nature 238: 104 - 106
Gebhart G.F. (1982) Opiate and opioid peptide effects on brain stem neurons: relevance to nociception and antinociceptive pathways. Pain 12: 93 - 140
Gryglewski R.J., Panczenko B, Korbut R, Grodzinska L, Ocetkiewicz A (1975) Corticosteroids inhibit prostaglandin release from perfused mesenteric blood vessels of rabbit and from perfused lungs of sensitized guinea pig. Prostaglandins 10: 343 - 355
Handwerker H.O. (1976) Influences of algogenic substances and prostaglandins on the discharges of myelinated cutaneous nerve fibers identified as nociceptors. Advances in Pain Research and Therapy 1: 41 - 45
Hirata F, Schiffmann E, Venkatsubamanian K, Salomon D, Axelrod J (1980) A phospholipase A2 inhibitory protein in rabbit neutrophils induces by glucocorticoids. Proc Natl Acad Sci USA 77: 2533 - 2536
Hong S.L., Levine L (1976) Inhibition of arachidonic acid release from cells as the biochemical action of anti-inflammatory corticosteroids. Proc Natl Acad Sci USA 73: 1730 - 1734
21a.Jurna I, Brune K (1990) Central effect of the non-steroid anti-inflammatory agents, indometacin, ibuprofen, and diclofenac, determined in C fibre-evoked activity in single neurones of the rat thalamus. Pain 41: 71 - 80
Levy M (1985) Pharmkokinetik von Metamizolmetaboliten. In: Brune K, Lanz R (Hrsg) 100 Jahre Pyrazolone. Urban & Schwarzenberg, München Wien Baltimore, S 163 - 166
Lim R.K.S. (1970) Pain. Annu Rev Physiol 32: 269 - 288
Meredith T.J., Prescott L.F., Vale J.A. (1986) Why do patients still die from paracetamol poisoning? Br Med J 293: 345 - 346
Okuyama S, Aihara H. (1984) The mode of action of analgesic drugs in adjuvant arthritic rats as an experimental model of chronic inflammatory pain: possible central analgesic action of acidic nonsteroidal antiinflammatory drugs. Jap J Pharmacol 35: 95 - 103
Rainsford K.D. (1978) Stucture-activity relationships of non-steroid anti-inflammatory drugs. 1. Gastric ulcerogenic activity. Agents Actions 8: 587 - 605
Roth J (1985) Pharmakokinetik and Metabolisierung der Pyrazolinone. In: Brune K, Lanz R (Hrsg) 100 Jahre Pyrazolone. Urban & Schwarzenberg, München Wien Baltimore S 167 - 180
Roth G.J., Stanford N, Majerus P.W. (1975) Acetylation of prostaglandin synthetase by aspirin. Proc Nat Acad Sci USA 72: 3073 - 3076
Schroth H.J., Steinsträßer A, Berberich R, Kloss G (1985) Motilität der ableitenden Harnwege. Änderung der Ausscheidungsphase im Nierensequenzszintigram unter der Wirkung von Metamizol - ein Parameter zur Beurteilung. MMW 127: 227 - 228
Schaible H.G., Schmidt R.F. (1985) Entladungsverhalten von Rezeptoren mit feinen Afferenzen aus normalen and entzündeten Gelenken: Einfluß von Analgetika and Prostaglandinen. In: Brune K, Lanz R (Hrsg) 100 Jahre Pyrazolone Urban & Schwarzenberg, München Wien Baltimore, S 87 - 99
Seegers A.J.M., Jager L.P., Van Noordwijk J (1979) Effects of phenacetin, paracetamol and caffeine on the erosive activity of acetylsalicylic acid in the rat stomach: dose response relationship, time course of erosion development and effects on acid secretion. J Pharm Pharmacol 31: 840 - 848
Shapiro S (1984) Agranulocytoses and pyrazolone. Lancet 1: 451
Shen T.Y. (1979) Prostaglandin synthetase inhibitors I. In: Vane JR, Ferreira SH (eds) Anti-Inflammatory Drugs. Springer, Berlin Heidelberg New York (Handbook of Experimental Pharmacology, vol 50 /11: 305 - 347 )
Shyu K.W., Lin M.T. (1985) Hypothalamic monoaminergic mechanisms of aspirin-induced analgesia in monkeys. J Neural Transm 62: 285 - 293
Szczeklik A (1984) Anti-inflammatory drugs and asthma. Int Med 4: 6 - 9
Szczeklik A, Gryglewski R.J., Czerniawska-Mysik G, Pieton R (1977) Asthma attacks in aspirine-sensitive patients by diclofenac and naproxen. Br Med J 2: 231 - 232
Tammisto T, Tigerstedt I (1980) Mild analgesics in postoperative pain. Br J Clin Pharmacol 10: 347S - 350S
Vane J.R. (1971) Inhibition of prostaglandin synthesis as a mechanism of action for aspirin-like drugs. Nature 231: 232 - 235
Kolfschoten A, Zandberg P, Jager L.P., Noordwijk J (1982) The influence of paracetamol on the erosive activity of indometacin on the rat stomach. Agents Actions 12: 247 - 253
Weithmann K.U., Alpermann H.G. (1985) Biochemical and pharmacological effects of dipyrone and its metabolites in model systems related to arachidonic acid cascade. Arzneim Forsch 35: 947 - 952
Winder C.V., Wax J, Burr V, Been M, Rosiere C.E. (1958) A study of pharmacological influences on ultraviolet erythema in guinea pigs. Arch Int Pharmacodyn Ther 116: 261 - 292
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Jurna, I. (1990). Analgetika mit antipyretischer Wirkung: Klinische Pharmakologie. In: Lehmann, K.A. (eds) Der postoperative Schmerz. Springer, Berlin, Heidelberg. https://doi.org/10.1007/978-3-662-06539-6_7
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