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Current status of estrogen receptors

Chapter
Part of the Progress in Drug Research book series (PDR, volume 59)

Summary

Increasing knowledge on structure and function of estrogen receptors is providing information on the mechanism of action of estrogen agonists, as well as antagonists, and in understanding their tissue-selective action. However, there are still many factors associated with estrogen response which are poorly understood. Therefore, the task of designing a tissue-selective estrogen for use as a pharmaceutical in estrogen-dependent disorders remains an uncertain game. This review provides information on the current status of estrogen receptors for a better understanding.

Key words

Estrogen receptors selective estrogen receptor modulators estrogen antagonists hormone receptors. 

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© Springer Basel AG 2002

Authors and Affiliations

  1. 1.Medicinal Chemistry DivisionCentral Drug Research InstituteLucknowIndia

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