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Biological Activity in the Quinazolone Series

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Progress in Drug Research / Fortschritte der Arzneimittelforschung / Progrès des recherches pharmaceutiques

Abstract

It is a happy coincidence that the year 1969 in which this review is being written, marks the centenary of the synthesis by Griess [1] of the first derivative of quinazoline, though the name of the hypothetical basic compound, unknown at that time, was given as ‘quinazoline’ only in 1887 by Weddige [2] and quinazoline itself was synthesised in 1903 by Gabriel [3]. Paul and Busch [4] suggested the following numbering which is still in use today (I).

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  1. Research Division, Alembic Chemical Works Co. Ltd., Baroda-3, India

    A. H. Amin, D. R. Mehta & S. S. Samarth

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    Ernst Jucker

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Amin, A.H., Mehta, D.R., Samarth, S.S. (1970). Biological Activity in the Quinazolone Series. In: Jucker, E. (eds) Progress in Drug Research / Fortschritte der Arzneimittelforschung / Progrès des recherches pharmaceutiques. Progress in Drug Research / Fortschritte der Arzneimittelforschung / Progrès des Recherches Pharmaceutiques, vol 14. Birkhäuser Basel. https://doi.org/10.1007/978-3-0348-7075-7_5

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