Solid-Phase Synthesis of 1,3,5-Trisubstituted 1,4-Diazepin-2-one Peptide Mimic

  • Hassan S. Iden
  • William D. Lubell
Conference paper
Part of the Advances in Experimental Medicine and Biology book series (volume 611)


Secondary Amine Dinitrophenyl Hydrazine Reductive Amination Sodium Cyanoborohydride Magnesium Bromide 



The authors acknowledge gratefully financial support from the Natural Sciences and Engineering Research Council of Canada (NSERC) and the Fonds Québécois de la Recherche sur la Nature et les Technologies (FQRNT).


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Copyright information

© Springer Science+Business Media, LLC 2009

Authors and Affiliations

  • Hassan S. Iden
    • 1
  • William D. Lubell
    • 1
  1. 1.Département de chimieUniversité de MontréalMontréalCanada

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