Synthesis of pyrrolo[3,2-e][1,4]diazepin-2-ones as potential γ-turn mimetics

  • Philippe Deaudelin
  • William D. Lubell
Conference paper
Part of the Advances in Experimental Medicine and Biology book series (volume 611)


Transcriptase Inhibitor Free Amine Rapid Metabolism Poor Bioavailability Benzyl Ester 
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This work was funded by the Natural Sciences and Engineering Research Council of Canada and the Fonds de Recherches sur la Nature et les Technologies du Québec.


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Copyright information

© Springer Science+Business Media, LLC 2009

Authors and Affiliations

  • Philippe Deaudelin
    • 1
  • William D. Lubell
    • 1
  1. 1.Département de chimieUniversitéde MontréalMontréalCanada

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