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A combination of ligand SAR and receptor site-directed mutagenesis reveals requirements for antagonist activity at the melanocortin-3 receptor

  • Bettina Proneth
  • Federico P. Portillo
  • Carrie Haskell-Luevano
Part of the Advances in Experimental Medicine and Biology book series (volume 611)

Keywords

Para Position Antagonist Activity Melanocortin Receptor Potent Antagonist Rational Drug Design 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

Notes

Acknowledgments

The work was funded by the NIH RO1DK57080 grant.

References

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Copyright information

© Springer Science+Business Media, LLC 2009

Authors and Affiliations

  • Bettina Proneth
    • 1
  • Federico P. Portillo
    • 1
  • Carrie Haskell-Luevano
    • 1
  1. 1.Department of Medicinal ChemistryUniversity of FloridaGainesvilleUSA

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