I

  • J. Elks
  • C. R. Ganellin

Keywords

COOH COOH Inosine Pranobex Triiodobenzoic Acid Extra Pharmacopoeia Radioactive Agent 
These keywords were added by machine and not by the authors. This process is experimental and the keywords may be updated as the learning algorithm improves.

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References

  1. Chang, P.K., Biochem. Pharmacol., 1961, 8, 327Google Scholar
  2. Chang, P.K., J. Med. Chem., 1963, 6, 428Google Scholar
  3. Miles, D.W., J. Am. Chem. Soc., 1969, 91, 831Google Scholar
  4. Fritzsche, H., Z. Chem., 1971, 11, 69Google Scholar
  5. Prusoff, W.H., Pharmacol. Ther., 1979, 7, 1Google Scholar
  6. Ghiassy, F., Acta Crystallogr., Sect. B, 1981, 37, 1921Google Scholar
  7. De Clercq, E., Mol. Pharmacol., 1982, 21, 217Google Scholar
  8. Prusoff, W.H., Int. Encyl. Pharmacol. Ther., 1984, 111, 341Google Scholar
  9. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12854.Google Scholar
  10. Gerster, J.F., J. Med. Chem., 1987, 30, 839Google Scholar
  11. Neu, H.C., J. Antimicrob. Chemother., 1987, 19, 175Google Scholar
  12. Goutarel, M., Hely. Chim. Acta, 1956, 39, 742Google Scholar
  13. Bartlett, M.F., J. Am. Chem. Soc., 1958, 80, 126Google Scholar
  14. Biemann, K., Tetrahedron Lett., 1961, 68Google Scholar
  15. Búchi, G., J. Am. Chem. Soc., 1966, 88, 3099Google Scholar
  16. Blbha, K., Collect. Czech. Chem. Commun., 1974, 39, 2258Google Scholar
  17. Rosenmund, P., Chem. Ber., 1975, 108, 1871Google Scholar
  18. Damak, M., Tetrahedron Lett., 1976, 3531Google Scholar
  19. Henwood, J.M., Drugs, 1988, 36, 11Google Scholar
  20. Nagai, H., Jpn. J. Pharmacol., 1983, 33, 1215Google Scholar
  21. Mue, S., Arch. Int. Pharmacodyn. Ther., 1986, 283, 153Google Scholar
  22. Adams, S.S., J. Pharm. Pharmacol., 1968, 20, 305Google Scholar
  23. Pettersen, J.E., Biomed. Mass Spectrom., 1978, 5, 488Google Scholar
  24. Tamura, Y., Chem. Pharm. Bull., 1982, 30, 915Google Scholar
  25. Adams, S.S., Arch. Pharmacodyn. Exp. Ther., 1969, 178, 115.Google Scholar
  26. Adams, S.S., Toxicol. Appl. Pharmacol., 1969, 15, 310Google Scholar
  27. McConnell, J.F., Cryst. Struct. Commun., 1974, 3, 73Google Scholar
  28. Kaiser, D.G., J. Pharm. Sci., 1976, 65, 269Google Scholar
  29. Shiori, T., J. Org. Chem., 1978, 43, 2936Google Scholar
  30. Ghislandi, V., Farmaco, Ed. Sci., 1982, 37, 81Google Scholar
  31. Nicholson, J.S., Chron. Drug Discovery, 1982, 1, 149Google Scholar
  32. Gruber, K., Arzneim.-Forsch., 1983, 33, 1176Google Scholar
  33. Hayashi, T., J. Org. Chem., 1983, 48, 2195Google Scholar
  34. Hiyama, T., Synthesis, 1986, 645Google Scholar
  35. Yamauchi, T., Synthesis, 1986, 1044Google Scholar
  36. Nicoll-Griffith, D.A., J. Chromatogr., 1987, 402, 179Google Scholar
  37. Piccolo, O., J. Org. Chem., 1987, 52, 10Google Scholar
  38. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 2867Google Scholar
  39. Wernicke, E.A., Chem. Ztg., 1936, 60, 85Google Scholar
  40. Gugenheim, P.G., J. Soc. Chem. Ind. (London), 1950, 69, 107Google Scholar
  41. Wernicke, E.A., Arzneim-Forsch., 1953, 3, 187Google Scholar
  42. Koch, J., Arch. Pharm. (Weinheim, Ger.), 1985, 318, 198Google Scholar
  43. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1615.Google Scholar
  44. Sax, N.I., Dangerous Properties of Industrial Materials, 6th Ed., Van Nostrand-Reinhold, 1984, 1604.Google Scholar
  45. Chiti, W., Farmaco, Ed. Sci., 1960, 15, 809Google Scholar
  46. Marmo, E., Arzneim.-Forsch., 1970, 20, 277Google Scholar
  47. Kelly, T.R., Tetrahedron Lett., 1978, 4457Google Scholar
  48. Broadhurst, M.J., J. Chem. Soc., Perkin Trans. 1, 1982, 2249Google Scholar
  49. Rao, A.V.R., J. Chem. Soc., Chem. Commun., 1984, 453Google Scholar
  50. Ganzina, F., Invest. New Drugs, 1986, 4, 85Google Scholar
  51. Weiss, R.B., Cancer Chemother. Pharmacol., 1986, 18, 185Google Scholar
  52. Zini, G., Cancer Chemother. Pharmacol., 1986, 16, 107Google Scholar
  53. Okamoto, K., Chem. Pharm. Bull., 1982, 30, 2797.Google Scholar
  54. Naguoka, A., Jpn. J. Pharmacol., 1984, 36, 291.Google Scholar
  55. Atfani, M., C.R. Acad. Sci. Ser. 2, 1986, 302, 171Google Scholar
  56. Ferry, N., Biochem. Pharmacol., 1986, 35, 1511Google Scholar
  57. Carron, M., Arzneim.-Forsch., 1971, 21, 1992Google Scholar
  58. Schulten, H.-R., Biomed. Mass Spectrom., 1974, 1, 223Google Scholar
  59. Perales, A., Acta Crystallogr., Sect. B, 1977, 33, 1935Google Scholar
  60. Takamizawa, A., Chem. Pharm. Bull., 1977, 25, 2900Google Scholar
  61. Kinas, R.W., Bull. Acad. Pol. Sci. Ser. Sci. Chim., 1978, 26, 39Google Scholar
  62. Ludeman, S.M., J. Org. Chem., 1979, 44, 1163Google Scholar
  63. Pankiewicz, K., J. Am. Chem. Soc., 1979, 101, 7712Google Scholar
  64. Wroblewski, A.E., Inorg. Chem., 1980, 19, 3713Google Scholar
  65. Su, C.N., J. Am. Chem. Soc., 1982, 104, 7343Google Scholar
  66. Misiura, K., J. Med. Chem., 1983, 26, 674Google Scholar
  67. Brade, W.P., Med. Actual., 1984, 20, 491Google Scholar
  68. Buess, M.L., Org. Magn. Reson., 1984, 22, 67Google Scholar
  69. Brade, W.P., Cancer Treat. Rev., 1985, 12, 1Google Scholar
  70. Kleinrok, Z., Arch. Immunol. Ther. Exp., 1986, 34, 293Google Scholar
  71. Berdel, W.E., Cancer Res., 1983, 43, 5538Google Scholar
  72. Leder, G.H., Lipids, 1987, 22, 958Google Scholar
  73. Herrmann, D.B., Lipids, 1988, 23, 76Google Scholar
  74. Krause, W., Eur. J. Clin. Pharmacol., 1986, 30, 61Google Scholar
  75. Schenker, K.V., Hely. Chim. Acta, 1986, 69, 1718Google Scholar
  76. Schillinger, E., New Cardiovasc. Drugs, 1986, 209Google Scholar
  77. Kampe, K.D., Angew. Chem., Int. Ed. Engl., 1982, 7, 540Google Scholar
  78. Thienpont, D., Arzneim.-Forsch., 1981, 31, 309Google Scholar
  79. Sircar, I., J. Med. Chem., 1985, 28, 1405Google Scholar
  80. Weishaar, R.E., Eur. J. Pharmacol., 1985, 119, 205Google Scholar
  81. Evans, D.B., Drug Dev. Res., 1986, 9, 143Google Scholar
  82. Steffen, R.P., New Cardiovasc. Drugs, 1986, 81Google Scholar
  83. Moos, W.H., J. Med. Chem., 1987, 30, 1963Google Scholar
  84. Leuke, D., Arzneim.-Forsch., 1967, 17, 317Google Scholar
  85. Kuhnert-Brandstaetter, M., Microchem. J., 1972, 17, 639Google Scholar
  86. Blazek, J., Cesk. Farm, 1975, 24, 174Google Scholar
  87. Shealy, Y.F., J. Pharm. Sci., 1968, 57, 83; 1975, 64, 177Google Scholar
  88. Hansch, C., Cancer Chemother. Rep., Part I, 1973, 57, 383Google Scholar
  89. Hill, D.L., Cancer Res., 1975, 35, 3106Google Scholar
  90. Koga, H., Chem. Pharm. Bull., 1974, 22, 482Google Scholar
  91. Cutbush, S.D., Acta Crystallogr., Sect. C, 1983, 39, 353Google Scholar
  92. Moore, E.C., Pharmacol. Ther., 1985, 27 167 (rev, cleric)Google Scholar
  93. Roby, T.O., Res. Vet. Sci., 1972, 13, 519Google Scholar
  94. Piskov, V.B., Khim.-Farm. Zh., 1974, 8, 17Google Scholar
  95. Aliu, Y.O., Am. J. Vet. Res., 1977, 38, 2001Google Scholar
  96. Rao, K.S., Indian Vet. J., 1980, 57, 283Google Scholar
  97. Wright, W.B., J. Med. Chem., 1966, 9, 852, 858Google Scholar
  98. Lien, E.J., J. Med. Chem., 1970, 13, 681Google Scholar
  99. Caroon, J.M., J. Med. Chem., 1982, 25, 666Google Scholar
  100. Chaples, C.B., J. Med. Chem., 1983, 26, 823 Google Scholar
  101. Carpy, A., Acta Crystallogr., Sect. C, 1984, 40, 1267Google Scholar
  102. Timmermans, P.B., J. Pharmacol. Exp. Ther., 1984, 228, 739Google Scholar
  103. El-Merzabani, M.M., Gann., 1955, 56, 589Google Scholar
  104. Okumoto, T., Chem. Pharm. Bull., 1976, 24, 1913Google Scholar
  105. Cain, B.F., J. Med. Chem., 1977, 20, 515Google Scholar
  106. Vesely, D.L., Oncology, 1979, 36, 122Google Scholar
  107. El-Merzabani, M.M., Pharmazie, 1983, 38, 110Google Scholar
  108. Leanza, W.J., J. Med. Chem., 1979, 22, 1435Google Scholar
  109. Shinkai, I., Tetrahedron Lett., 1982, 4903Google Scholar
  110. Kahan, F.M., J. Antimicrob. Chemother., 1983, 12 ( Suppl. D), IGoogle Scholar
  111. Oberholtzer, E.R., Anal. Profiles Drug Subst., 1988, 17, 73Google Scholar
  112. Schindler, W., Hely. Chim. Acta, 1954, 37, 472.Google Scholar
  113. Bickel, M.H., Biochem. Pharmacol., 1966, 15, 1155Google Scholar
  114. Buech, O., Med. Pharmacol. Exp., 1966, 15, 187Google Scholar
  115. Post, M.L., Acta Crystallogr., Sect. B, 1975, 31, 1008Google Scholar
  116. Kender, D.N., Anal. Profiles Drug Subst., 1985, 14, 37Google Scholar
  117. Craik, D.J., Chem. Pharm. Bull., 1987, 35, 188Google Scholar
  118. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 5355.Google Scholar
  119. Griffin, B.W., Metab. Clin. Exp., 1987, 36, 486Google Scholar
  120. Park, Y.H., J. Pharm. Sci., 1988, 77, 110Google Scholar
  121. Sterne, J., Therapie, 1965, 20, 89, 95Google Scholar
  122. Späth, E., Ber., 1933, 66, 1137Google Scholar
  123. Govindachari, T.R., Tetrahedron, 1968, 24, 753Google Scholar
  124. Basa, S.C., Chem. Ind. ( London ), 1970, 746Google Scholar
  125. Booer, M., Ghana J. Sci., 1970, 10, 82Google Scholar
  126. Murray, R.D.H., Tetrahedron, 1984, 40, 5225Google Scholar
  127. Leslie, G.B., J. Appl. Toxicol., 1982, 2, 265Google Scholar
  128. Durant, G.J., J. Med. Chem., 1985, 28, 1414Google Scholar
  129. Zacchei, A.G., Eur. J. Drug Metab. Pharmacokinet., 1977, 2, 37Google Scholar
  130. DeSolms, S.J., J. Med. Chem., 1978, 21, 437Google Scholar
  131. Wilhelmsson, C.E., Br. J. Clin. Pharmacol., 1979, 8, 261Google Scholar
  132. Woltersdorf, O.W., J. Labelled Compd. Radiopharm., 1980, 17, 635Google Scholar
  133. Blaine, E.H., Clin. Exp. Hypertens., 1982, 4, 161Google Scholar
  134. Dolling, U.H., J. Am. Chem. Soc., 1984, 106, 446Google Scholar
  135. Campbell, D.B., Curr. Med. Res. Opin., 1983, 8, 9Google Scholar
  136. Klunk, L.J., J. Clin. Pharmacol., 1983, 23, 377Google Scholar
  137. Pruss, T., Am. Heart J., 1983, 106, 208Google Scholar
  138. Amt, J., Naunyn-Schmiedeberg’s Arch. Pharmacol., 1985, 329, 101Google Scholar
  139. Bogeso, K.P., J. Med. Chem., 1985, 28, 1817Google Scholar
  140. Tachikawa, S., Arch. Int. Pharmacodyn. Ther., 1979, 238, 81Google Scholar
  141. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 15324.Google Scholar
  142. Takenaka, T., Arzneim.-Forsch., 1972, 22, 1864Google Scholar
  143. Murase, K., Chem. Pharm. Bull., 1976, 24, 552Google Scholar
  144. Bartsch, W., Arzneim.-Forsch., 1977, 27, 1022Google Scholar
  145. Anon., Drugs of Today, 1980, 16, 20Google Scholar
  146. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12849.Google Scholar
  147. Mattocks, A.R., J. Chem. Soc., 1961, 5400Google Scholar
  148. Mattocks, A.R., J. Chem. Soc. (C), 1967, 329Google Scholar
  149. Kugelman, M., Lloydia, 1976, 39, 125Google Scholar
  150. Jones, A.J., Aust. J. Chem., 1982, 35, 1173Google Scholar
  151. Suffness, M., Alkaloids (N.Y.), 1985, 25, 32Google Scholar
  152. Vedejs, E., J. Org. Chem., 1985, 50, 2170Google Scholar
  153. Zalkow, L.H., J. Med. Chem., 1985, 28, 687Google Scholar
  154. McCord, C.P., J. Ind. Hyg. Toxicol., 1942, 24 243 (lox)Google Scholar
  155. Brauer, G., Handbuch Prap. Anorg. Chem., 3rd Ed., 1975–1981, 867Google Scholar
  156. Sax, N.I., Dangerous Properties of Industrial Materials, 7th Ed., Van Nostrand-Reinhold, 1989, 1986.Google Scholar
  157. Nannini, G., Arzneim.-Forsch., 1973, 23, 1090Google Scholar
  158. Tonani, R., Adv. Mass Spectrom., 1980, 8B, 1274Google Scholar
  159. Tremoli, E., Pharmacol. Res. Commun., 1981, 13, 847Google Scholar
  160. Bergamaschi, M., Pharmacol. Res. Commun., 1984, 16, 979Google Scholar
  161. Crow, M.J., Thromb. Res., 1985, 38, 303Google Scholar
  162. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12850.Google Scholar
  163. Pidevich, I.N., Farmakol. Toksikol., 1971, 34, 155Google Scholar
  164. Blankley, C.J., J. Med. Chem., 1987, 30, 992Google Scholar
  165. Shen, T.Y., J. Am. Chem. Soc., 1963, 85, 488.Google Scholar
  166. Yamamato, H., Chem. Pharm. Bull., 1968, 16, 17Google Scholar
  167. Bertazzoni, D., Boll. Chim. Farm., 1970, 109, 60Google Scholar
  168. Kistenmacher, T.J., J. Am. Chem. Soc., 1972, 94, 1340Google Scholar
  169. Shen, T.Y., Adv. Drug Res., 1977, 12, 89Google Scholar
  170. Singh, S.P., J. Heterocycl. Chem., 1978, 15, 13Google Scholar
  171. Helleberg, L., Clin. Pharmacokinet., 1981, 6, 245Google Scholar
  172. O’Brien, M., Anal. Profiles Drug Subst., 1984, 13, 211Google Scholar
  173. Kaneniwa, N., Chem. Pharm. Bull., 1985, 33, 3447Google Scholar
  174. Sauvaire, D., Drugs Exp. Clin. Res., 1987, 13, 247Google Scholar
  175. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 5116Google Scholar
  176. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2658.Google Scholar
  177. Buttinoni, A., Arzneim.-Forsch., 1973, 23, 1100Google Scholar
  178. Nannini, G., Arzneim.-Forsch., 1973, 23, 1090Google Scholar
  179. Tosolini, G.P., J. Pharm. Sci., 1974, 63, 1072Google Scholar
  180. Kametani, T., J. Heterocycl. Chem., 1978, 15, 369Google Scholar
  181. DeMunari, S., Tetrahedron Lett., 1980, 21, 2273Google Scholar
  182. Ghislandi, V., Farmaco, Ed. Sci., 1982, 37, 81Google Scholar
  183. Buttinoni, A., J. Pharm. Pharmacol., 1983, 35, 603Google Scholar
  184. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2659.Google Scholar
  185. Archibald, J.L., J. Med. Chem., 1971, 14, 1054Google Scholar
  186. Archibald, J.L., Br. J. Clin. Pharmacol., 1981, 12, 45Google Scholar
  187. Holmes, B., Drugs, 1986, 31, 467Google Scholar
  188. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 879.Google Scholar
  189. Safdy, M.E., J. Med. Chem., 1982, 25, 723Google Scholar
  190. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12851.Google Scholar
  191. Barchewitz, G., Therapie, 1974, 29, 57Google Scholar
  192. Gulland, J.M., J. Chem. Soc., 1936, 765Google Scholar
  193. Kinichi, I., Chem. Pharm. Bull., 1966, 14, 1377Google Scholar
  194. Green, D.P.L., Tetrahedron, 1970, 26, 1031Google Scholar
  195. Munns, A.R.I., Acta Crystallogr., Sect. B, 1970, 26, 1114Google Scholar
  196. Chenon, M.T., J. Am. Chem. Soc., 1975, 97, 4627Google Scholar
  197. Westhof, E., Z. Naturforsch., C, 1975, 30, 131Google Scholar
  198. Hawkes, G.E., J. Chem. Soc., Perkin Trans. 2, 1977, 1268 (N-15 nmr)Google Scholar
  199. Yamazaki, A., J. Heterocycl. Chem., 1978, 15, 353Google Scholar
  200. Aviado, D.M., J. Pharmacol., 1983, 14, 47Google Scholar
  201. Campoli-Richards, D.M., Drugs, 1986, 32, 383Google Scholar
  202. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 1551.Google Scholar
  203. Badgett, C.O., J. Am. Chem. Soc., 1947, 69, 2907Google Scholar
  204. Angyal, S.J., Adv. Carbohydr. Chem., 1959, 14, 135Google Scholar
  205. Angyal, S.J., J. Chem. Soc., 1961, 4116, 4122, 4718.Google Scholar
  206. Shvets, V.I., Tetrahedron, 1973, 29, 331.Google Scholar
  207. Isbrandt, L.R., J. Am. Chem. Soc., 1980, 102, 3144.Google Scholar
  208. Wells, W.W., Kirk-Othmer. Encycl. Chem. Technol., 3rd Ed., 1983, 24, 50Google Scholar
  209. Bleasdale, J.E., Eds., Inositol and Phosphoinositides: Metabolism and Regulation, Humane Press, Clifton, N.J., 1985Google Scholar
  210. Holub, B.J., Annu. Rev. Nutr., 1986, 6, 563Google Scholar
  211. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 540, 588, 8197Google Scholar
  212. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1056, 7877, 9243.Google Scholar
  213. Gauss, W., Angew. Chem., 1955, 67, 217Google Scholar
  214. Petersen, S., Medezin u. Chemie, 1956, 5, 163Google Scholar
  215. Akhtar, M.H., Can. J. Chem., 1975, 53, 2891Google Scholar
  216. Nicol, D.S.H., Nature (London), 1960, 187, 483Google Scholar
  217. Blundell, T.L., Adv. Protein Chem., 1972, 26, 279Google Scholar
  218. Butt, W.R., Hormone Chemistry, 1975, Wiley, New York, 2nd Ed., Vol. 1Google Scholar
  219. Geiger, R., Chem.-Ztg., Chem. App., 1976, 100, 111Google Scholar
  220. Sieber, P., Helv. Chim. Acta, 1977, 60, 27Google Scholar
  221. Goeddel, D.V., Proc. Natl. Acad. Sci. USA, 1979, 76, 106Google Scholar
  222. Meienhofer, J., Burger’s Medicinal Chemistry, 1979, (Wolff, M.E., Ed.), Wiley-Interscience, New York, 4th Ed., Part II, 813Google Scholar
  223. Morihara, K., Nature (London), 1979, 280, 412Google Scholar
  224. Williamson, K.L., Biochemistry, 1979, 18, 5965Google Scholar
  225. Blundell, T., FEBS Lett., 1980, 109, 167Google Scholar
  226. Duckworth, W.C., Endocr. Rev., 1981, 2, 210Google Scholar
  227. Gunning, J., Peptides (N.Y.), 1981, 4, 55Google Scholar
  228. Levine, R., Vitamin Horm. (N.Y.), 1982, 39, 145Google Scholar
  229. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 7201.Google Scholar
  230. Geiger, R., Hoppe-Seyler’s Z. Physiol. Chem., 1973, 354, 1285, 1521Google Scholar
  231. Caterson, I., Drugs, 1979, 17, 289Google Scholar
  232. Smith, G.D., Acta Crystallogr., Sect. B, 1982, 38, 3028Google Scholar
  233. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 7205.Google Scholar
  234. Isaacs, A., Proc. R. Soc., London, Ser. B, 1957, 147, 258.Google Scholar
  235. Rubinstein, M., Proc. Natl. Acad. Sci. USA, 1979, 76, 640Google Scholar
  236. Tan, Y.H., J. Biol. Chem, 1979, 254, 8067Google Scholar
  237. Derynck, R., Nature (London), 1980, 285, 542Google Scholar
  238. Pestka, S., Ann. Rep. Med. Chem., 1981, 16, 229Google Scholar
  239. Wallace, D.M., Biochem. Biophys. Res. Commun., 1981, 100, 865Google Scholar
  240. Gray, P.W., Nature (London), 1982, 295, 503Google Scholar
  241. Pestka, S., UCLA Symp. Mol. Cell. Biol., 1982, 25, 81Google Scholar
  242. Vilcek, J., Lymphokines (N.Y.), 1985, 11, 1Google Scholar
  243. Pestka, S., Annu. Rev. Biochem., 1987, 56, 727Google Scholar
  244. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1683.Google Scholar
  245. Catabolin. Endogenous Pyrogen. Haematopoietin 1. Leucocyte Endogenous Mediator. Lymphocyte Activating Factor. ETAF. IL-1. LAFGoogle Scholar
  246. Cytokine peptide containing 152 amino acid residues. Isol. from neutrophils. Immunomodulator. Antitumour agent.Google Scholar
  247. Dinarello, C.A., Rev. Infect. Dis., 1984, 6, 51Google Scholar
  248. Benjamin, W.R., Annu. Rep. Med. Chem., 1985, 20, 173Google Scholar
  249. Gery, I., Methods Enzymol., 1985, 116 456 (rev, isol, props)Google Scholar
  250. Billiau, A., Int. Congr. Ser.-Excerpta Med., 1986, 715, 47Google Scholar
  251. Krakauer, T., CRC Crit. Rev. Immunol., 1986, 6, 245Google Scholar
  252. Maury, C.P.J., Acta Med. Scand., 1986, 220, 291Google Scholar
  253. Horohov, D.W., Drugs, 1987, 33, 289Google Scholar
  254. Auron, P.E., Lymphokines, 1988, 2, 33Google Scholar
  255. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 16853.Google Scholar
  256. Mier, J.W., Proc. Natl. Acad. Sci. U.S.A., 1980, 77, 6134Google Scholar
  257. Lahm, H.W., J. Chromatogr., 1985, 326, 357Google Scholar
  258. Mertelsmann, R., Immunobiology (Stuttgart), 1986, 172 400Google Scholar
  259. Fujishima, A., J. Mol. Biol., 1987, 197, 373Google Scholar
  260. Horohov, D.W., Drugs, 1987, 33, 289Google Scholar
  261. Rosenberg, S.A., Immunology Today, 1988, 9, 58Google Scholar
  262. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 16854.Google Scholar
  263. Ihle, J.N., Methods Enzymol., 1985, 116 540 (rev, isol, purifn)Google Scholar
  264. Schrader, J.W., Annu. Rev. Immunol., 1986, 4, 205Google Scholar
  265. Clark-Lewis, I., Lymphokines, 1988, 15, 1Google Scholar
  266. Yokota, T., Proc. Natl. Acad. Sci. U.S.A., 1986, 83, 5894Google Scholar
  267. Paul, W.E., Annu. Rev. Immunol., 1987, 5, 429Google Scholar
  268. Moeller, G., Ed., Immunol. Rev., 1988, 102 Google Scholar
  269. Azuma, C., Nucleic Acids Res., 1986, 14, 9149Google Scholar
  270. Moeller, G., Ed., Immunol. Rev., 1988, 102 Google Scholar
  271. Hirano, T., Proc. Natl. Acad. Sci. USA, 1985, 82, 5490Google Scholar
  272. Sehgal, P.B., Science, 1987, 235, 731Google Scholar
  273. Hirano, T., Med. Immunol., 1988, 15, 195Google Scholar
  274. Kishimoto, T., Annu. Rev. Immunol., 1988, 6, 485Google Scholar
  275. Medzihradszky, K., Recent Dev. Chem. Nat. Carbon Compd., 1976, 7, 117Google Scholar
  276. Thody, A.J., Adv. Drug Res., 1977, 11, 23Google Scholar
  277. Li, C.H., Horm. Proteins Pept., 1978, 5, 1Google Scholar
  278. Nikiforovich, G.V., FEES Lett., 1981, 126, 180Google Scholar
  279. Reith, M.E., Pharmacol. Ther., 1981, 12, 449Google Scholar
  280. Hammond, G.L., Int. J. Pept. Protein Res., 1983, 22, 161Google Scholar
  281. Kullmann, W., J. Protein Chem., 1983, 2, 289Google Scholar
  282. Hruby, V.J., Pept. Protein Res., 1984, 3, 1Google Scholar
  283. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 5936.Google Scholar
  284. Fleming, J.S., Arch. Int. Pharmacodyn. Ther., 1969, 178, 423Google Scholar
  285. Juby, P.F., J. Med. Chem., 1969, 12, 396Google Scholar
  286. Haworth, W.N., J. Chem. Soc., 1932, 2384.Google Scholar
  287. McDonald, E.J., Adv. Carbohydr. Chem., 1946, 2, 254Google Scholar
  288. Bacon, J.S.D., Biochem. J., 1951, 48, 114.Google Scholar
  289. Percival, E.G.V., Structural Carbohydr. Chem., 2nd Ed., 1962, 274Google Scholar
  290. Aspinall, G.O., Methods Carbohydr. Chem., 1965, 5, 157Google Scholar
  291. Ovodov, Yu.S., Dokl. Akad. Nauk SSSR, 1968, 178, 1338Google Scholar
  292. Kennedy, J.F., Carbohydr. Res., 1973, 26, 401.Google Scholar
  293. Marchessault, R.H., Can. J. Chem., 1980, 58, 2415Google Scholar
  294. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2137.Google Scholar
  295. Nakajo, M., J. Nucl. Med., 1983, 24, 672Google Scholar
  296. Chambon, C., J. Biophys. Med. Nucl., 1984, 8, 198Google Scholar
  297. Wieland, D.M., J. Med. Chem., 1984, 27, 149Google Scholar
  298. McEwan, A.J., Appl. Radiat. Isot., 1986, 37, 765Google Scholar
  299. Ertl, S., Nucl. Med. Commun., 1987, 8, 643Google Scholar
  300. Lindner, I., Arzneim.-Forsch., 1961, 11, 384Google Scholar
  301. Heide, M., Med. Klin., 1965, 60, 996Google Scholar
  302. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1559.Google Scholar
  303. Hoey, G.B., J. Med. Chem., 1966, 9, 964Google Scholar
  304. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1522, 1560.Google Scholar
  305. Felder, E., Heiv. Chim. Acta, 1965, 48, 259Google Scholar
  306. Grothuesmann, H.G., Arzneim.-Forsch., 1965, 15, 233.Google Scholar
  307. Zsebök, Z., Arzneim.-Forsch., 1967, 17, 1380Google Scholar
  308. Pitre, D., Anal. Profiles Drug Subst., 1986, 15, 337Google Scholar
  309. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1523, 1524, 1562.Google Scholar
  310. Lerner, H.H., Anal. Profiles Drug Subst., 1974, 3, 333Google Scholar
  311. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6thGoogle Scholar
  312. Ed., Akademie-Verlag, Berlin, 1987, 5550 Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1525, 1526, 1563.Google Scholar
  313. Ferry, D.R., Naunyn-Schmiedeberg’s Arch. Pharmacol., 1984, 325, 186Google Scholar
  314. Glossmann, H., J. Cardiovasc. Pharmacol., 1985, 7, 520Google Scholar
  315. Hoppe, J.O., J. Am. Pharm. Assoc., 1959, 48, 368Google Scholar
  316. Yagupol’skii, L.M., Ukr. Khim. Zh., 1960, 26, 233Google Scholar
  317. Kracmar, J., Pharmazie, 1966, 21, 460Google Scholar
  318. Hoevel-Kestermann, H., Pharm. Acta Helv., 1972, 47, 394Google Scholar
  319. Novello, N.J., J. Biol. Chem, 1926, 67, 555Google Scholar
  320. Sinn, H., Int. J. Appl. Radiat. Isot., 1977, 28, 809Google Scholar
  321. Balthazor, T.M., J. Org. Chem., 1979, 44, 1447Google Scholar
  322. Dougan, H., Appl. Radiat. Isot., 1986, 37, 915Google Scholar
  323. Counsell, R.E., Steroids, 1970, 16, 317Google Scholar
  324. Couch, M.W., Steroids, 1976, 27, 451Google Scholar
  325. Bieirwaltes, W.H., Ther. Nucl. Med. (Symp.)Google Scholar
  326. Scott, K.N., J. Nucl. Med., 1977, 18, 492Google Scholar
  327. Scott, K.N., Can. J. Chem., 1979, 57, 27Google Scholar
  328. Owoyale, J.A., Steroids, 1981, 37, 133.Google Scholar
  329. Baughman, R.G., J. Agric. Food Chem., 1982, 30, 293Google Scholar
  330. Fogy, I., Int. J. Mass Spectrom. Ion Phys., 1983, 48 319.Google Scholar
  331. Agrochemical Handbook, Royal Society of Chemistry, London, 1983, A239. Pesticide Manual, 6th Ed., 304; 7th Ed., 319.Google Scholar
  332. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 3863.Google Scholar
  333. Sax, N.I., Dangerous Properties of Industrial Materials, 5th Ed., Van Nostrand-Reinhold, 1979, 745.Google Scholar
  334. Bougault, J., C. R. Hebd. Seances Acad. Sci., 1910, 150, 876.Google Scholar
  335. Hunsdiecker, H., Chem. Ber., 1942, 75, 291.Google Scholar
  336. Fox, R.B., J. Chem. Eng. Data, 1963, 8, 612.Google Scholar
  337. Laufer, P., Eur. J. Nucl. Med., 1981, 18, 1205Google Scholar
  338. Okada, R.D., J. Labelled Compd. Radiopharm., 1983, 8, 211Google Scholar
  339. Knapp, F.F., J. Med. Chem., 1984, 27, 94Google Scholar
  340. Lauer, W.M., J. Am. Chem. Soc., 1935, 57, 2361Google Scholar
  341. Block, E., J. Am. Chem. Soc., 1986, 108, 4568Google Scholar
  342. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6thEd., Akademie-Verlag, Berlin, 1987, 13.Google Scholar
  343. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1577.Google Scholar
  344. Cantarelli, G., Farmaco, Ed. Prat., 1979, 34, 393Google Scholar
  345. De Angelis, L., Drugs of Today, 1980, 16, 154Google Scholar
  346. Riva, M., Arzneim.-Forsch., 1983, 33 1091Google Scholar
  347. Hoppe, J.O. J. Am. Pharm. Assoc., 1959, 48 368Google Scholar
  348. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 812.Google Scholar
  349. Carlsen, L., Eur. J. Nucl. Med., 1982, 7, 280Google Scholar
  350. Holman, B.L., Invest. Radiol., 1982, 17, 206Google Scholar
  351. Lyall, D., Nucl. Med. Commun., 1985, 6, 485Google Scholar
  352. Cohen, M.B., Appl. Radiat. Isot., 1986, 37 749Google Scholar
  353. Mertens, J., Eur. J. Nucl. Med., 1987, 13, 380Google Scholar
  354. Felder, E., Farmaco, Ed. Sci., 1973, 28, 912, 925Google Scholar
  355. Rosati, G., Farmaco, Ed. Sci., 1973, 28, 996Google Scholar
  356. Pitre, D., Farmaco, Ed. Sci., 1974, 29, 793Google Scholar
  357. Pitre, D., Arch. Pharm. (Weinheim, Ger.), 1984, 317, 1037Google Scholar
  358. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1527, 1567.Google Scholar
  359. Klieger, E., Arch. Pharm. (Weinheim, Ger.), 1973, 306, 834Google Scholar
  360. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12855.Google Scholar
  361. Priewe, H., Chem. Ber., 1954, 87, 651Google Scholar
  362. Rosati, G., Boll. Chico. Farm., 1972, 111, 129Google Scholar
  363. Muetzel, W., Invest. Radiol., 1976, 11, 598Google Scholar
  364. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1528, 1529, 1569.Google Scholar
  365. Wolf, G.L., Invest. Radiol, 1981, 16, 320Google Scholar
  366. Edelson, J., J. Chromatogr., 1983, 274, 428Google Scholar
  367. Haavaldsen, J., Acta Pharm. Suec., 1983, 20, 219Google Scholar
  368. Edelson, J., J. Pharm. Sci., 1984, 73, 993.Google Scholar
  369. Kawada, T.K., Drug Intell. Clin. Pharm., 1985, 19, 525Google Scholar
  370. Shaw, D.D., Invest. Radiol, 1985, 20 (Suppl.), 10, 65, 84, 98Google Scholar
  371. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12856.Google Scholar
  372. Pitre, D., Chim. Ther., 1970, 5, 185Google Scholar
  373. Fumagalli, L., Pharmazie, 1975, 30, 78Google Scholar
  374. East Ger. Pat., 67 207, (1969); CA, 72, 106654Google Scholar
  375. Cassebaum, H., Pharmazie, 1972, 27, 391Google Scholar
  376. Bornschein, I., Pharmazie, 1974, 29, 730Google Scholar
  377. Counsell, R.E., J. Pharm. Sci., 1967, 56, 1042Google Scholar
  378. Counsell, R.E., J. Med. Chem., 1969, 12, 232Google Scholar
  379. Bakker, C.N.M., J. Labelled Compd. Radiopharm., 1979, 16, 917Google Scholar
  380. Goulding, R.W., J. Labelled Compd. Radiopharm., 1979, 16, 46Google Scholar
  381. Eakins, M.N., Int. J. Appl. Radiat. Isot., 1980, 31, 553Google Scholar
  382. Bubeck, B., Eur. J. Nucl. Med., 1981, 6, 227Google Scholar
  383. Felder, E., Farmaco, Ed. Sci., 1977, 32, 835Google Scholar
  384. Pitre, D., Farmaco, Ed. Sci., 1980, 35, 826Google Scholar
  385. Pitre, D., Invest. Radiol., 1980, 15, S301Google Scholar
  386. Clerici, A., Biomed. Mass Spectrom., 1982, 9, 257Google Scholar
  387. Ganazzoli, F., Acta Crystallogr., Sect. C, 1983, 39, 1570Google Scholar
  388. Felder, E., Anal. Profiles Drug Subst., 1988, 17, 115Google Scholar
  389. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 14037.Google Scholar
  390. Skjoeld, W., J. Chromatogr., 1986, 366, 299Google Scholar
  391. Michelet, A.A., Acta Radiol., 1987, 28, 329 Google Scholar
  392. Lewis, T.R., J. Am. Chem. Soc., 1949, 71, 3753Google Scholar
  393. Pitre, D., J. Med. Chem., 1968, 11, 406Google Scholar
  394. Pitre, D., Arch. Pharm. (Weinheim, Ger.), 1984, 317, 367Google Scholar
  395. Pitre, D., Anal. Profiles Drug Subst., 1985, 14, 181Google Scholar
  396. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6thGoogle Scholar
  397. Ed., Akademie-Verlag, Berlin, 1987, 1908 Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1570.Google Scholar
  398. Strain, W.H., J. Am. Chem. Soc., 1942, 64, 1436Google Scholar
  399. Baker, W., J. Chem. Soc. Ind., 1944, 63, 223 Google Scholar
  400. Liewendahl, K., Nucl.-Med., Suppl., 1968, 375 Google Scholar
  401. Kostin, V.N., Zh. Prikl. Khim. (Leningrad), 1977, 50, 2338Google Scholar
  402. Hansen, E.B., Br. J. Radiol., 1978, 51, 321Google Scholar
  403. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1571.Google Scholar
  404. Papa, D., J. Am. Chem. Soc., 1953, 75, 1107Google Scholar
  405. Stahl, E., Z. Anal. Chem., 1964, 200, 377 Google Scholar
  406. Mudge, G.H., J. Pharmacol. Exp. Ther., 1971, 178, 159Google Scholar
  407. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1572.Google Scholar
  408. Harwart, A., Arch. Exp. Pathol. Pharmacol., 1959, 237,186 Google Scholar
  409. Priewe, H., Chem. Ber., 1960, 93, 2347Google Scholar
  410. Cassebaum, H., Pharmazie, 1961, 16, 389Google Scholar
  411. Kimbel, K.H., Acta Radiol., 1961, 55, 305Google Scholar
  412. Sammul, O.R., J. Assoc. Off. Agric. Chem., 1964, 47, 918Google Scholar
  413. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1553.Google Scholar
  414. Felder, E., Farmaco, Ed. Sci., 1976, 31, 349Google Scholar
  415. Tirone, P., Farmaco, Ed. Sci., 1976, 31, 397, 437Google Scholar
  416. Pitre, D., Farmaco, Ed. Prat., 1976, 31, 516, 529, 540Google Scholar
  417. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 18652.Google Scholar
  418. Hoey, G.B., J. Med. Chem., 1966, 9, 964Google Scholar
  419. Rosenberg, F.J., Invest. Radiol., 1980, 15, S142Google Scholar
  420. Berk, R.N., Invest. Radiol., 1981, 16, 240Google Scholar
  421. Park, G.B., Drug Metab. Dispos., 1981, 9, 43Google Scholar
  422. Klieger, E., Arch. Pharm. (Weinheim, Ger.), 1973, 306, 834Google Scholar
  423. Siefert, H.M., Lymphology, 1980, 13, 150Google Scholar
  424. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12858.Google Scholar
  425. Hoey, G.B., J. Med. Chem., 1963, 6, 24Google Scholar
  426. Benness, G.T., Clin. Radiol., 1970, 21, 150Google Scholar
  427. Singh, G.B., Indian Drugs Pharm. Ind., 1980, 15, 35Google Scholar
  428. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 1530, 1531, 1575.Google Scholar
  429. Speck, U., Arzneim.-Forsch., 1978, 28, 2143, 2290Google Scholar
  430. Baehring-Kuhlmey, S.R., Drugs of Today, 1979, 15, 45Google Scholar
  431. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12859, 12860.Google Scholar
  432. Sarin, J.P.S, Phytochemistry, 1973, 12, 2461Google Scholar
  433. Schulz, W., Arzneim.-Forsch., 1976, 26, 960Google Scholar
  434. South African Pat., 6 707 766, (1968); CA, 70, 97033uGoogle Scholar
  435. Deckers, W., Postgrad. Med. J., 1975, 51 (suppl. 7), 76Google Scholar
  436. Pook, K.H., Justus Liebigs Ann. Chem., 1975, 1499Google Scholar
  437. Bauer, R., Arzneim.-Forsch., 1976, 26, 974Google Scholar
  438. Sarajana, L., Arzneim.-Forsch., 1976, 26, 985Google Scholar
  439. Bauer, R., Pharmacol. Biochem. Prop. Drug. Subst., 1979, 2, 489Google Scholar
  440. Massey, K.L., Drug. Intell. Clin. Pharm., 1985, 19, 5.Google Scholar
  441. Oates, J.A., New Engl. J. Med., 1988, 319, 486Google Scholar
  442. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 386Google Scholar
  443. Rice, L.M., J. Med. Chem., 1964, 7, 313Google Scholar
  444. Gluckman, M.I., Psychopharmacologia, 1969, 15, 169Google Scholar
  445. Lemberger, L., Biochem. Pharmacol., 1970, 19, 3021Google Scholar
  446. Miller, K.W., Experientia, 1970, 26, 863.Google Scholar
  447. Freeman, J.J., J. Pharmacol. Exp. Ther., 1972, 183, 307Google Scholar
  448. Rodgers, J.R., Acta Crystallogr., Sect. B, 1974, 30, 1970Google Scholar
  449. De Montigny, C., Mod. Prob. Pharmacopsychiatry, 1982, 18, 102Google Scholar
  450. Maxwell, R.A., Drug. Dev. Res., 1983, 3, 203Google Scholar
  451. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2518.Google Scholar
  452. Libermann, D., Bull. Soc. Chim. Fr., 1961, 1952.Google Scholar
  453. De Sagher, R.M., Biomed. Mass Spectrom., 1975, 2, 82Google Scholar
  454. De Sagher, R.M., Drug Metab. Dispos., 1975, 3, 423Google Scholar
  455. Fuicrand, P., Eur. J. Med. Chem.-Chim. Ther., 1978, 13, 177Google Scholar
  456. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2519.Google Scholar
  457. Martin, M., Eur. J. Med. Chem.-Chim. Ther., 1974, 9, 563Google Scholar
  458. Ju, H.-W., IEEE Trans. Nucl. Sci., 1977, NS-26 559Google Scholar
  459. Subramanian, G., Nuclearmedizin Suppl. (Stuttgart), 1978, 16, 136Google Scholar
  460. Williams, W., J. Nucl. Med., 1984, 25, 160Google Scholar
  461. Fox, H.H., J. Org. Chem., 1953, 18, 994.Google Scholar
  462. Yale, H.L., J. Am. Chem. Soc., 1953, 75, 1933.Google Scholar
  463. Davies, W.A., J. Clin. Exp. Psychopharmacol., 1958, 19, Suppl. 1, 1Google Scholar
  464. Randall, L.O., Ann. N.Y. Acad. Sci., 1959, 80, 626Google Scholar
  465. Spector, S., J. Pharmacol. Exp. Ther., 1960, 128, 15Google Scholar
  466. Coubeils, J.L., C.R. Hebd. Seances Acad. Sci., Ser. D, 1971, 273, 1164Google Scholar
  467. Kauffman, G.B., J. Chem. Educ. 1979, 56, 35Google Scholar
  468. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2520.Google Scholar
  469. Connors, T.A., Chem.-Biol. Interact., 1972, 5, 415.Google Scholar
  470. Tobe, M.L., J. Clin. Hematol. Oncol., 1977, 7, 114 Google Scholar
  471. Laverick, M., Br. J. Radiol., 1981, 54, 529Google Scholar
  472. Pendyala, L., Cancer Treat. Rep., 1982, 66, 509Google Scholar
  473. Barnard, C.F.J., J. Chem. Res. (S), 1983, 12, 302Google Scholar
  474. Chang, P., Drugs Future, 1985, 10, 561Google Scholar
  475. Harrap, K.R., Cancer Treat. Rev., 1985, 12A, 21Google Scholar
  476. Barnard, C.F.J., Chem. Br., 1986, 22, 1001Google Scholar
  477. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 18653.Google Scholar
  478. Mattioda, G., J. Med. Chem., 1975, 18, 553Google Scholar
  479. Dourish, C.T., Trends Pharmacol. Sci., 1986, 7, 212Google Scholar
  480. Goodwin, G.M., Psychopharmacology, 1986, 89, 382Google Scholar
  481. Rice, K.C., Nature (London), 1979, 278, 854Google Scholar
  482. Williams, E.F., Pharmacol., Biochem. Behay., 1981, 14, 487Google Scholar
  483. Skolnick, P., J. Neurochem., 1982, 39, 1142Google Scholar
  484. Jensen, B., Acta Crystallogr., Sect. C, 1988, 44, 1602Google Scholar
  485. Stefancich, G., Farmaco, Ed. Sci., 1985, 40, 237Google Scholar
  486. Domagala, J.M., J. Med. Chem., 1986, 29, 394Google Scholar
  487. Rackham, D.M., Org. Magn. Reson., 1978, 11, 424Google Scholar
  488. Chatfield, D.H., Xenobiotica, 1979, 9, 585Google Scholar
  489. Ross, W.J., J. Med. Chem., 1979, 22, 412Google Scholar
  490. Dawson, W., Br. J. Pharmacol., 1980, 71, 387Google Scholar
  491. Braeunlich, H., Pharmazie, 1964, 19, 650Google Scholar
  492. Bastos, W.P., Pharmacology, 1970, 4, 39.Google Scholar
  493. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 5622.Google Scholar
  494. Perjessy, A., Tetrahedron, 1971, 27, 6159Google Scholar
  495. Islam, A.M., Bull. Chem. Soc. Jpn., 1974, 47, 1274Google Scholar
  496. Fanelli, O., Arzneim.-Forsch., 1975, 25, 873Google Scholar
  497. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12866.Google Scholar
  498. Chubb, F.C., Can. J. Chem., 1959, 37, 1121Google Scholar
  499. Hokfelt, B. J. Med. Chem., 1962, 5 247Google Scholar
  500. Rosen, H., Toxicol. Appl. Pharmacol., 1966, 8, 13Google Scholar
  501. Ruelius, H.W., Arzneiur.-Forsch., 1970, 20, 115Google Scholar
  502. Gardner, T.S., J. Med. Chem., 1960, 2, 133Google Scholar
  503. Ho, B.T., J. Pharm. Sci., 1972, 61, 821Google Scholar
  504. Rudy, B.C., Anal. Profiles Drug Subst., 1973, 2, 295Google Scholar
  505. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2521.Google Scholar
  506. Dutcher, J.D., J. Am. Chem. Soc., 1946, 68, 419Google Scholar
  507. Gley, P., Compt. Rend. Soc. Biol., 1952, 146, 13Google Scholar
  508. Jeffreys, J.A.D., J. Chem. Soc., 1956, 4451Google Scholar
  509. Bick, I.R.C., J. Chem. Soc., 1961, 1896Google Scholar
  510. Battersby, A.R., J. Chem. Soc., 1965, 2239Google Scholar
  511. Baldas, J., J. Chem. Soc., Perkin Trans. 1, 1972, 599Google Scholar
  512. Dwuma-Badu, D., Phytochemistry, 1975, 14, 2520Google Scholar
  513. Galeffi, C., Gazz. Chim. Ital., 1978, 108, 97Google Scholar
  514. Marsaioli, A.J., Phytochemistry, 1978, 17, 1655Google Scholar
  515. Singh, R.S., J. Nat. Prod., 1981, 44, 664Google Scholar
  516. Godefroi, E.F., J. Med. Chem., 1969, 12, 784Google Scholar
  517. Kessler, H.J., Arzneim.-Forsch., 1979, 29, 1352Google Scholar
  518. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12868.Google Scholar
  519. Grana, E., Farmaco, Ed. Sci., 1969, 24, 1038Google Scholar
  520. Mardle, M.J., J. Med. Chem., 1974, 17, 513Google Scholar
  521. Lovgren, K., Acta Pharm. Suec., 1977, 14, 30Google Scholar
  522. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2070, 2071.Google Scholar
  523. Koepfli, J.B., J. Am. Chem. Soc., 1947, 69, 1837Google Scholar
  524. Jilek, J., Collect. Czech. Chem. Commun., 1984, 49, 2638Google Scholar
  525. Pacakova, V., J. Chromatogr., 1984, 298, 309Google Scholar
  526. Polakova, L., Acta Nerv. Super., 1984, 26, 9, 10, 14, 16, 17Google Scholar
  527. Polakova, L., Cesk. Farm., 1986, 35, 97, 255Google Scholar
  528. Protiva, M., Collect. Czech. Chem. Commun., 1986, 51, 698Google Scholar
  529. McAleer, W.J., J. Org. Chem., 1958, 23, 508Google Scholar
  530. Smith, L.L., J. Org. Chem., 1958, 23, 960Google Scholar
  531. Pechet, M.M., J. Clin. Invest., 1959, 38, 681Google Scholar
  532. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12869.Google Scholar
  533. Späth, E., Ber., 1939, 72, 52Google Scholar
  534. Perel’son, M.E., Khim. Prir. Soedin., 1966, 381Google Scholar
  535. Lee, K.-H., J. Pharm. Sci., 1969, 58, 681Google Scholar
  536. Perel’son, M.E., Khim. Prir. Soedin., 1971, 576Google Scholar
  537. Voigt, D., J. Prakt. Chem., 1977, 319, 767Google Scholar
  538. Bernstein, J.R., J. Chromatogr., 1985, 342, 228Google Scholar
  539. Hayes, J.S., J. Pharmacol. Exp. Ther., 1985, 233, 318Google Scholar
  540. Robertson, D.W., J. Med. Chem., 1985, 28, 717Google Scholar
  541. Jonas, R., Arch. Pharm. (Weinheim, Ger.), 1986, 319, 1150Google Scholar
  542. May, E.L., J. Org. Chem., 1952, 17, 1210Google Scholar
  543. Portoghese, P.S., J. Pharm. Sci., 1966, 55, 865Google Scholar
  544. Portoghese, P.S., Tetrahedron Lett., 1966, 6299 Google Scholar
  545. Portoghese, P.S., J. Med. Chem., 1970, 13, 626Google Scholar
  546. Ruemmler, R., Arch. Pharm. (Weinheim, Ger.), 1971, 304, 561Google Scholar
  547. Haller, R., Arch. Pharm. (Weinheim, Ger.), 1973, 306, 510Google Scholar
  548. Easton, N.R., J. Am. Chem. Soc., 1948, 70, 76Google Scholar
  549. Larsen, A.A., J. Am. Chem. Soc., 1948, 70, 4194Google Scholar
  550. Howe, E.E., J. Am. Chem. Soc., 1949, 71, 2935Google Scholar
  551. Walton, E., J. Chem. Soc., 1949, 648Google Scholar
  552. Eddy, N.B., J. Pharmacol. Exp. Ther., 1950, 98, 121Google Scholar
  553. Henkel, J.G., J. Med. Chem., 1974, 17, 124Google Scholar
  554. Shefter, E., J. Med. Chem., 1974, 17, 1037Google Scholar
  555. Portoghese, P.S., J. Med. Chem., 1982, 25, 684Google Scholar
  556. Gerardy, B.M., J. Labelled Compd. Radiopharm., 1985, 22, 5Google Scholar
  557. Tilford, C.H., J. Am. Chem. Soc., 1949, 71, 1705Google Scholar
  558. Sammul, O.R., J. Assoc. Off. Agr. Chem., 1964, 47, 918Google Scholar
  559. Meyer, H., Monatsh. Chem., 1912, 33, 400Google Scholar
  560. Ceriotti, G., Arch. Int. Pharmacodyn., 1953, 93, 105Google Scholar
  561. Ceriotti, G., Br. J. Pharmacol., 1953, 8, 356Google Scholar
  562. Bhat, T.N., Acta Crystallogr., Sect. B, 1974, 30, 2921Google Scholar
  563. Krishna Murti, C.R., Antibiotics (N.Y.), 1975, 3, 623Google Scholar
  564. Brewer, G.A., Anal. Profiles Drug Subst., 1977, 6, 183Google Scholar
  565. Takayama, K., Antibiotics (N.Y.), 1979, 5, 98Google Scholar
  566. Weber, W.W., Clin. Pharmacokinet., 1979, 4, 401Google Scholar
  567. Ed., Akademie-Verlag, Berlin, 1987, 438Google Scholar
  568. Sax, N.I. Dangerous Properties of Industrial Materials, 6th Ed., Van Nostrand-Reinhold, 1984, 1643.Google Scholar
  569. Bello, R., Arch. Farmacol. Toxicol., 1976, 2, 256Google Scholar
  570. Cadena, R., Arzneim.-Forsch., 1977, 27, 1457Google Scholar
  571. Mitjavila, M.T., Arzneim.-Forsch., 1977, 27, 1460Google Scholar
  572. Berthold, K., Acta Endocrinol. (Copenhagen), 1970, 63, 431Google Scholar
  573. Berthold, K., Arzneim.-Forsch., 1971, 21, 1510Google Scholar
  574. Beccari, E., Science, 1953, 118, 249Google Scholar
  575. Pratesi, P., Farmaco, Ed. Sci., 1960, 15, 3Google Scholar
  576. Payne, K.R., Ind. Chem., 1961, 37, 523Google Scholar
  577. Drost, R.H., Pharm. Weekbl., 1967, 102, 1379Google Scholar
  578. Brittain, R.T., Adv. Drug Res., 1970, 5, 197Google Scholar
  579. Riggin, R.M., Anal. Lett., 1974, 7, 791Google Scholar
  580. Pasaribu, S.J., Aust. J. Chem., 1978, 31, 2629Google Scholar
  581. Konzett, H., Trends Pharmacol. Sci., 1981, 2, 47Google Scholar
  582. Tariq, M., Anal. Profiles Drug Subst., 1985, 14, 391Google Scholar
  583. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 2126, 2127 Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2074, 2075.Google Scholar
  584. Janssen, P., Arch. Int. Pharmacodyn., 1955, 103, 82Google Scholar
  585. Santoro, R.S., Anal. Profiles Drug Subst., 1973, 2, 315; 1983, 12, 721Google Scholar
  586. Datta, N., J. Chem. Soc., Perkin Trans. 2, 1977, 781Google Scholar
  587. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 387.Google Scholar
  588. Gourevitch, A., Proc. Soc. Exptl. Biol. Med., 1961, 107, 455Google Scholar
  589. Glombitza, K.W., Justus Liebigs Ann. Chem., 1964, 673, 166Google Scholar
  590. Pfister, J.R., J. Med. Chem., 1972, 15, 1032Google Scholar
  591. Bergamaschi, M., Boll. Chim. Farm., 1972, 111, 667Google Scholar
  592. Vecchietti, V., Eur. J. Med. Chem., 1974, 9, 501Google Scholar
  593. Hafner, K., Justus Liebigs Ann. Chem., 1957, 606, 90Google Scholar
  594. Bellesia, F., J. Chem. Soc., Chem. Commun., 1976, 34.Google Scholar
  595. Harre, M., Chem. Ber., 1982, 115, 1437Google Scholar
  596. Plattner, P.A., Hely. Chim. Acta, 1949, 32, 2137, 2452Google Scholar
  597. gorm, F., Collect. Czech. Chem. Commun., 1951, 16, 168, 626Google Scholar
  598. Caujolle, F., Ann. Pharm. Fr., 1952, 10, 412Google Scholar
  599. Herz, A., Arzneim.-Forsch., 1953, 3, 253Google Scholar
  600. Jacob, T.M., Tetrahedron, 1964, 20, 2821 (uv, synth)Google Scholar
  601. Hoffmann, W., Tetrahedron Lett., 1975, 533Google Scholar
  602. Llinas, J.R., Can. J. Chem., 1975, 53, 2911Google Scholar
  603. Mukherjee, D., J. Am. Chem. Soc., 1979, 101, 251Google Scholar
  604. Fusetani, N., Experientia, 1981, 37, 680Google Scholar
  605. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6thGoogle Scholar
  606. Treibs, W., Justus Liebigs Ann. Chem., 1954, 586, 202Google Scholar
  607. Meier, W., Hely. Chim. Acta, 1963, 46, 1929Google Scholar
  608. Planz, G., Arzneim.-Forsch., 1973, 23, 281Google Scholar
  609. Schaefer, H., Arzneim.-Forsch., 1984, 34, 233Google Scholar
  610. Hertz, F., Arzneim.-Forsch., 1980, 30, 1549Google Scholar
  611. Hashimoto, A., Agric. Biol. Chem., 1970, 34, 1843Google Scholar
  612. Oritani, T., Agric. Biol. Chem., 1973, 37, 1695Google Scholar
  613. Leffingwell, J.C., Cosmet. Perfum., 1974, 89, 69Google Scholar
  614. Yamaguchi, S., Tetrahedron Lett., 1977, 89Google Scholar
  615. Nakatani, Y., Synthesis, 1978, 147Google Scholar
  616. Dauzonne, D., Org. Magn. Reson., 1981, 17, 18Google Scholar
  617. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 266.Google Scholar
  618. Sax, N.I., Dangerous Properties of Industrial Materials, 5th Ed., Van Nostrand-Reinhold, 1979, 791.Google Scholar
  619. Bulter, K., J. Med. Chem., 1967, 10, 891Google Scholar
  620. Weiss, G., Xenobiotica, 1981, 11, 207Google Scholar
  621. McKillop, A., Tetrahedron, 1983, 39 3797 Martindale, The Extra Pharmacopoeia, 28th/29th Eds.Google Scholar
  622. 1982/.
    Pharmaceutical Press, London, 12863.Google Scholar
  623. Meisenheimer, J., Ber., 1926, 59 1848 (oxide)Google Scholar
  624. Manske, R.H.F., Chem. Rev., 1942, 30, 145Google Scholar
  625. Narasimhan, N.S., Chem. Ind. ( London ), 1967, 120Google Scholar
  626. Gansow, O.A., J. Am. Chem. Soc., 1976, 98, 4250Google Scholar
  627. Johns, S.A., Aust J. Chem., 1976, 29, 1617Google Scholar
  628. Dyke, S.F., Chem. Heterocycl. Compd., 1981, 38, 1Google Scholar
  629. Kametani, T., Chem. Heterocycl. Compd., 1981, 38, 139Google Scholar
  630. Kirk-Othmer Encycl. Chem. Technol., 3rd Ed., 1982, 19, 499Google Scholar
  631. Wagner, H., Planta Med., 1986, 378Google Scholar
  632. Sax, N.I., Dangerous Properties of Industrial Materials, 6th Ed., Van Nostrand-Reinhold, 1984, 1669.Google Scholar
  633. Marchetti, E., Experientia, 1965, 21, 687Google Scholar
  634. Lenda, K., J. Liq. Chromatogr., 1981, 4, 863Google Scholar
  635. Kleine, M.W., Allergologie, 1986, 9, 330Google Scholar
  636. Lannom, H.K., Int. J. Pept. Protein Res., 1986, 28, 67Google Scholar
  637. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 2547.Google Scholar
  638. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 4031.Google Scholar
  639. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 6140.Google Scholar
  640. DiPasquale, G., Agents Actions, 1975, 5, 256Google Scholar
  641. Yakatan, G.J., Semin. Arthritis Rheum., 1982, 12, Suppl. 2, 153Google Scholar
  642. Zinnes, H., J. Med. Chem., 1982, 25, 12Google Scholar
  643. DiPasquale, G., Med. Actual., 1983, 19, 119Google Scholar
  644. Borondy, P.E., Drug Metab. Dispos., 1984, 12, 444 Google Scholar
  645. Dalla Croce, P., J. Chem. Res. (S), 1986, 150Google Scholar
  646. Svoboda, J., Collect. Czech. Chem. Commun., 1986, 51, 1133Google Scholar
  647. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 12873.Google Scholar
  648. Moed, H.D., Red. Tray. Chim. Pays-Bas, 1956, 75, 1215Google Scholar
  649. Data, P.G., Farmaco, Ed. Sci., 1973, 28, 611Google Scholar
  650. Negwer, M., Organic-Chemical Drugs and their Synonyms, 6th Ed., Akademie-Verlag, Berlin, 1987, 4903 Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 9246.Google Scholar
  651. Rieu, J.P., J. Pharm. Sci., 1980, 69, 49Google Scholar
  652. Cousse, H., J. Pharm. Sci., 1981, 70, 1245Google Scholar
  653. Roques, R., Acta Crystallogr., Sect. B, 1981, 37, 457Google Scholar
  654. Crasnier, F., Theochem., 1983, 14, 175Google Scholar
  655. Crawley, F.E., Eur. J. Drug Metab. Pharmacokinet, 1983, 8, 287Google Scholar
  656. Rynbrandt, R.H., J. Med. Chem., 1981, 24, 1507Google Scholar
  657. Linet, O.I., Drugs Exp. Clin. Res., 1984, 10, 263Google Scholar
  658. Heider, J.G., Transplant. Proc., 1987, 19, 96Google Scholar
  659. Tse, F.L.S., Eur. J. Clin. Pharmacol., 1987, 32, 361Google Scholar
  660. Heeres, J., J. Med. Chem., 1984, 27, 894Google Scholar
  661. Cauwenbergh, G., Drug Dev. Res., 1986, 8, 317Google Scholar
  662. Van Cauteren, H., Rev. Infect. Dis., 1987, 9, 543Google Scholar
  663. Mullen, G.B., HeIv. Chim. Acta, 1988, 71 718 (bibl)Google Scholar
  664. Martindale, The Extra Pharmacopoeia, 28th/29th Eds., 1982/1989, Pharmaceutical Press, London, 18657.Google Scholar
  665. Danswan, G.W., Arzneim.-Forsch., 1976, 26, 2190, 2193, 2197Google Scholar
  666. Chabala, J.C. et al, J. Med. Chem., 1980, 23, 1134Google Scholar
  667. U.S.P 4 199 569, (1980); CA, 93, 130559Google Scholar
  668. Campbell, W.C. et al, Science (Washington), 1983, 221, 823Google Scholar
  669. Calcott, P.H. et al, J. Antibiot., 1984, 37, 253Google Scholar
  670. Koch, H., Pharm. Int., 1984, 5, 55Google Scholar
  671. Fink, D.W., Anal. Profiles DrugSubst., 1988, 17, 155Google Scholar
  672. Baker, R. et al, Chem. Br., 1989, 25, 692Google Scholar

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© Springer Science+Business Media Dordrecht 1990

Authors and Affiliations

  • J. Elks
  • C. R. Ganellin

There are no affiliations available

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