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Acylation of Fischer’s Base with Methyl Aroylpyruvates

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Abstract

Methyl (Z)-4-aryl-2-hydroxy-4-oxobut-2-enoates (methyl aroylpyruvates) reacted with 1,3,3-trimethyl- 2-methylidene-2,3-dihydro-1H-indole (Fischer’s base) to give (2Z,5E)-1-aryl-3-hydroxy-5-(1,3,3-trimethyl-2,3-dihydro-1H-indol-2-ylidene)pent-2-ene-1,4-diones.

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Authors and Affiliations

  1. Institute of Technical Chemistry, Ural Branch, Russian Academy of Sciences, ul. Akad. Koroleva 3, Perm, 614013, Russia

    T. A. Rozdyalovskaya & V. V. Konovalova

  2. Perm National State Research University, ul. Bukireva 15, Perm, 614990, Russia

    M. V. Dmitriev

Authors
  1. T. A. Rozdyalovskaya
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  2. M. V. Dmitriev
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  3. V. V. Konovalova
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Corresponding author

Correspondence to V. V. Konovalova.

Additional information

Original Russian Text © T.A. Rozdyalovskaya, M.V. Dmitriev, V.V. Konovalova, 2018, published in Zhurnal Organicheskoi Khimii, 2018, Vol. 54, No. 1, pp. 139–141.

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Rozdyalovskaya, T.A., Dmitriev, M.V. & Konovalova, V.V. Acylation of Fischer’s Base with Methyl Aroylpyruvates. Russ J Org Chem 54, 139–142 (2018). https://doi.org/10.1134/S1070428018010141

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  • DOI: https://doi.org/10.1134/S1070428018010141

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