Russian Journal of Organic Chemistry

, Volume 47, Issue 10, pp 1527–1530 | Cite as

Polyfunctional imidazoles: IV. Synthesis of 2-aryl-4-chloro-1-methyl(aryl)-1H-imidazole-5-carbaldehydes

  • V. A. Chornous
  • A. N. Grozav
  • M. K. Bratenko
  • M. V. Vovk
Article

Abstract

2-Aroyl-2-[methyl(aryl)amino]acetamides reacted with the Vilsmeier-Haak reagent to give 2-aryl-4-chloro-1-methyl(aryl)-1H-imidazole-5-carbaldehydes.

Keywords

Benzoyl Chloride Anhydrous Acetonitrile Sodium Hydrogen Carbonate Glycinamides Phosphoryl Chloride 

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Copyright information

© Pleiades Publishing, Ltd. 2011

Authors and Affiliations

  • V. A. Chornous
    • 1
  • A. N. Grozav
    • 1
  • M. K. Bratenko
    • 1
  • M. V. Vovk
    • 2
  1. 1.Bukoviny State Medical UniversityChernovtsyUkraine
  2. 2.Institute of Organic ChemistryNational Academy of Sciences of UkraineKievUkraine

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