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Synthesis and Antibacterial Activity of 9-Oxo-9,10-dihydroacridinecarboxylic Acids Esters Bearing a Triazole Fragment

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Abstract

An effective method for the synthesis of new acridine-9(10H)-one (acridone) derivatives containing 1,2,3-triazole fragment was developed. A number of new triazole-containing compounds were synthesized from propargyl acridone acetate and their antimicrobial activity was studied.

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Acknowledgments

This work was financially supported by the Ministry of Education and Science of Russia (project no. 4.9516.2017/BCh).

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Authors and Affiliations

  1. Kursk State University, ul. Radishcheva 33, Kursk, 305000, Russia

    T. N. Kudryavtseva, A. Yu. Lamanov & G. V. Nazarov

  2. Kursk State Medical University, Kursk, Russia

    L. G. Klimova

Authors
  1. T. N. Kudryavtseva
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  2. A. Yu. Lamanov
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  3. L. G. Klimova
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  4. G. V. Nazarov
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Corresponding author

Correspondence to T. N. Kudryavtseva.

Additional information

Original Russian Text © T.N. Kudryavtseva, A.Yu. Lamanov, L.G. Klimova, G.V. Nazarov, 2018, published in Zhurnal Obshchei Khimii, 2018, Vol. 88, No. 4, pp. 593–598.

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Kudryavtseva, T.N., Lamanov, A.Y., Klimova, L.G. et al. Synthesis and Antibacterial Activity of 9-Oxo-9,10-dihydroacridinecarboxylic Acids Esters Bearing a Triazole Fragment. Russ J Gen Chem 88, 676–681 (2018). https://doi.org/10.1134/S1070363218040102

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