Abstract
The acylation of primary and secondary amines by 5-phenyltetrazol-2-ylacetyl chloride leads to the corresponding tetrazolylacetamides irrespective of the nature of the substituent in the structure of the amine.
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Putis, S.M., Zubarev, V.Y., Poplavskii, V.S. et al. Acylation of Amines with 5-Phenyltetrazol-2-ylacetyl Chloride. Chemistry of Heterocyclic Compounds 40, 854–861 (2004). https://doi.org/10.1023/B:COHC.0000044567.39872.b0
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DOI: https://doi.org/10.1023/B:COHC.0000044567.39872.b0