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N-Amination of Unsymmetrically Substituted Pyrimidines. Synthesis of Isomeric N-Aminopyrimidones

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

N-Amination of 6-amino-2-methyl-4-pyrimidone with O-(mesitylenesulfonyl)hydroxylamine leads to the 3-amino derivative. The isomeric 1,6-diamino-2-methyl-4-pyrimidone was obtained by the N-amination of the O-benzoyl derivative of the initial pyrimidone and removal of the benzoyl protection.

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REFERENCES

  1. Y. Tamura, J. Minamikawa, and M. Ikeda, Synthesis, 1 (1977).

  2. A. Yu. Ivanov, V. P. Tsyrenov, N. G. Antonov, P. S. Lobanov, and A. A. Potekhin, Khim. Geterotsikl. Soedin., 807 (2002).

  3. Z. Foldi, G. V. Fodar, I. Demjen, H. Szeker, and J. Halmos, Ber., 75, 755 (1942).

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Authors and Affiliations

  1. St. Petersburg State University, St. Petersburg, 198904, Petrodvorets, Russia

    M. B. Bodyagin, A. Yu. Ivanov, P. S. Lobanov & A. A. Potekhin

  2. Innsbruck University, A-6020, Austria

    K. Wurst & J. G. Schantl

Authors
  1. M. B. Bodyagin
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  2. A. Yu. Ivanov
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  3. K. Wurst
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  4. J. G. Schantl
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  5. P. S. Lobanov
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  6. A. A. Potekhin
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Bodyagin, M.B., Ivanov, A.Y., Wurst, K. et al. N-Amination of Unsymmetrically Substituted Pyrimidines. Synthesis of Isomeric N-Aminopyrimidones. Chemistry of Heterocyclic Compounds 39, 195–199 (2003). https://doi.org/10.1023/A:1023716424186

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  • DOI: https://doi.org/10.1023/A:1023716424186

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