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Synthesis of N-Substituted Derivatives of (5-Amino-2-methyl-1H-indol-3-yl)acetic Acid

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Chemistry of Heterocyclic Compounds Aims and scope

Abstract

A method has been developed for obtaining indole compounds containing an amino group in the benzene ring by the indolization of ethyl levulinate p-acetaminophenylhydrazone. A series of derivatives of (5-amino-2-methyl-1H-indol-3-yl)acetic acid at the 5-amino group has been synthesized.

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Authors and Affiliations

  1. Novomoskovsk Institute of the D. I. Mendeleev Russian University of Chemical Technology, Novomoskovsk, 301670

    S. A. Maklakov

  2. D. I. Mendeleev Russian University of Chemical Technology, Moscow, 125047

    Yu. I. Smushkevich

  3. Moscow K. A. Timiryazev Agricultural Academy, Moscow, 127550, Russia

    I. V. Magedov

Authors
  1. S. A. Maklakov
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  2. Yu. I. Smushkevich
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  3. I. V. Magedov
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Maklakov, S.A., Smushkevich, Y.I. & Magedov, I.V. Synthesis of N-Substituted Derivatives of (5-Amino-2-methyl-1H-indol-3-yl)acetic Acid. Chemistry of Heterocyclic Compounds 38, 539–542 (2002). https://doi.org/10.1023/A:1019500911047

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  • DOI: https://doi.org/10.1023/A:1019500911047

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