Abstract
Cyclization of 1-phenylpropane-1,2-dione monoarylhydrazones under Vilsmeier-Haack conditions gave 1-aryl-3-benzoyl-4-formylpyrazoles which were converted to 1-aryl-3-benzoyl-4-carboxypyrazoles using potassium permanganate in aqueous pyridine medium.
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Bratenko, M.K., Chornous, V.A. & Vovk, M.V. Polyfunctional Pyrazoles. 2. 1-Aryl-3-benzoyl-4-formyl- and 4-Carboxypyrazoles. Chemistry of Heterocyclic Compounds 37, 467–469 (2001). https://doi.org/10.1023/A:1017651904859
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DOI: https://doi.org/10.1023/A:1017651904859